GR3004124T3 - - Google Patents

Info

Publication number
GR3004124T3
GR3004124T3 GR910402151T GR910402151T GR3004124T3 GR 3004124 T3 GR3004124 T3 GR 3004124T3 GR 910402151 T GR910402151 T GR 910402151T GR 910402151 T GR910402151 T GR 910402151T GR 3004124 T3 GR3004124 T3 GR 3004124T3
Authority
GR
Greece
Prior art keywords
solid dispersion
dispersion composition
octacos
tetraone
azatricyclo
Prior art date
Application number
GR910402151T
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GR3004124T3 publication Critical patent/GR3004124T3/el

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
GR910402151T 1986-04-02 1992-03-24 GR3004124T3 (el)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868608080A GB8608080D0 (en) 1986-04-02 1986-04-02 Solid dispersion composition

Publications (1)

Publication Number Publication Date
GR3004124T3 true GR3004124T3 (el) 1993-03-31

Family

ID=10595572

Family Applications (1)

Application Number Title Priority Date Filing Date
GR910402151T GR3004124T3 (el) 1986-04-02 1992-03-24

Country Status (16)

Country Link
US (1) US4916138A (el)
EP (1) EP0240773B1 (el)
JP (1) JPS62277321A (el)
KR (2) KR950007209B1 (el)
AT (1) ATE73327T1 (el)
CA (1) CA1302279C (el)
DE (1) DE3777223D1 (el)
DK (1) DK174979B1 (el)
ES (1) ES2032397T3 (el)
GB (1) GB8608080D0 (el)
GR (1) GR3004124T3 (el)
HK (1) HK6397A (el)
IE (1) IE59712B1 (el)
MX (1) MX9202945A (el)
RU (1) RU1826977C (el)
UA (1) UA13209A (el)

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US5250678A (en) 1991-05-13 1993-10-05 Merck & Co., Inc. O-aryl, O-alkyl, O-alkenyl and O-alkynylmacrolides having immunosuppressive activity
US5565560A (en) * 1991-05-13 1996-10-15 Merck & Co., Inc. O-Aryl,O-alkyl,O-alkenyl and O-alkynylmacrolides having immunosuppressive activity
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US5189042A (en) * 1991-08-22 1993-02-23 Merck & Co. Inc. Fluoromacrolides having immunosuppressive activity
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US20050113460A1 (en) * 1999-04-30 2005-05-26 The Regents Of The University Of Michigan Compositions and methods relating to novel compounds and targets thereof
US20040176358A1 (en) * 1999-04-30 2004-09-09 The Regents Of The University Of Michigan Compositions and methods relating to novel compounds and targets thereof
US20030119029A1 (en) * 1999-04-30 2003-06-26 Regents Of The University Of Michigan Compositions and methods relating to novel benzodiazepine compounds and targets thereof
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US6989131B2 (en) * 2002-03-12 2006-01-24 Uop Llc Catalytic reactor with integral evaporator
JP4796300B2 (ja) * 2002-08-29 2011-10-19 ファイザー インコーポレイテッド モチライド化合物
CN1819817A (zh) * 2003-07-09 2006-08-16 株式会社钟根堂 一种泰克利玛的固体分散体
BRPI0413927B8 (pt) 2003-08-29 2021-05-25 Lifecycle Pharma As composição farmacêutica compreendendo tacrolimus, forma de dosagem, uso da composição, e, método para a preparação da composição
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US20090275099A1 (en) * 2004-04-27 2009-11-05 Regents Of The University Of Michigan Methods and compositions for treating diseases and conditions associated with mitochondrial function
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AU2008226532B2 (en) 2007-03-09 2011-09-22 The Regents Of The University Of Michigan Compositions and methods relating to novel compounds and targets thereof
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Also Published As

Publication number Publication date
DK140487A (da) 1987-10-03
EP0240773A1 (en) 1987-10-14
CA1302279C (en) 1992-06-02
HK6397A (en) 1997-01-24
JPS62277321A (ja) 1987-12-02
IE59712B1 (en) 1994-03-23
IE870843L (en) 1987-10-02
DK140487D0 (da) 1987-03-18
KR890001626A (ko) 1989-03-28
RU1826977C (ru) 1993-07-07
KR870010073A (ko) 1987-11-30
MX9202945A (es) 1992-07-01
KR950007209B1 (ko) 1995-07-04
UA13209A (uk) 1997-02-28
DE3777223D1 (de) 1992-04-16
KR950007210B1 (ko) 1995-07-04
EP0240773B1 (en) 1992-03-11
ES2032397T3 (es) 1993-02-16
DK174979B1 (da) 2004-04-05
ATE73327T1 (de) 1992-03-15
GB8608080D0 (en) 1986-05-08
US4916138A (en) 1990-04-10
JPH0536411B2 (el) 1993-05-31

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