GB0602632D0 - Preparation Of A Solid Dosage From Comprising Tacrolimus And/Or Sirolimus - Google Patents
Preparation Of A Solid Dosage From Comprising Tacrolimus And/Or SirolimusInfo
- Publication number
- GB0602632D0 GB0602632D0 GB0602632A GB0602632A GB0602632D0 GB 0602632 D0 GB0602632 D0 GB 0602632D0 GB 0602632 A GB0602632 A GB 0602632A GB 0602632 A GB0602632 A GB 0602632A GB 0602632 D0 GB0602632 D0 GB 0602632D0
- Authority
- GB
- United Kingdom
- Prior art keywords
- sirolimus
- tacrolimus
- preparation
- solid dosage
- dosage
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- QJJXYPPXXYFBGM-LFZNUXCKSA-N Tacrolimus Chemical compound C1C[C@@H](O)[C@H](OC)C[C@@H]1\C=C(/C)[C@@H]1[C@H](C)[C@@H](O)CC(=O)[C@H](CC=C)/C=C(C)/C[C@H](C)C[C@H](OC)[C@H]([C@H](C[C@H]2C)OC)O[C@@]2(O)C(=O)C(=O)N2CCCC[C@H]2C(=O)O1 QJJXYPPXXYFBGM-LFZNUXCKSA-N 0.000 title 1
- ZAHRKKWIAAJSAO-UHFFFAOYSA-N rapamycin Natural products COCC(O)C(=C/C(C)C(=O)CC(OC(=O)C1CCCCN1C(=O)C(=O)C2(O)OC(CC(OC)C(=CC=CC=CC(C)CC(C)C(=O)C)C)CCC2C)C(C)CC3CCC(O)C(C3)OC)C ZAHRKKWIAAJSAO-UHFFFAOYSA-N 0.000 title 1
- QFJCIRLUMZQUOT-HPLJOQBZSA-N sirolimus Chemical compound C1C[C@@H](O)[C@H](OC)C[C@@H]1C[C@@H](C)[C@H]1OC(=O)[C@@H]2CCCCN2C(=O)C(=O)[C@](O)(O2)[C@H](C)CC[C@H]2C[C@H](OC)/C(C)=C/C=C/C=C/[C@@H](C)C[C@@H](C)C(=O)[C@H](OC)[C@H](O)/C(C)=C/[C@@H](C)C(=O)C1 QFJCIRLUMZQUOT-HPLJOQBZSA-N 0.000 title 1
- 229960002930 sirolimus Drugs 0.000 title 1
- 239000007787 solid Substances 0.000 title 1
- 229960001967 tacrolimus Drugs 0.000 title 1
- QJJXYPPXXYFBGM-SHYZHZOCSA-N tacrolimus Natural products CO[C@H]1C[C@H](CC[C@@H]1O)C=C(C)[C@H]2OC(=O)[C@H]3CCCCN3C(=O)C(=O)[C@@]4(O)O[C@@H]([C@H](C[C@H]4C)OC)[C@@H](C[C@H](C)CC(=C[C@@H](CC=C)C(=O)C[C@H](O)[C@H]2C)C)OC QJJXYPPXXYFBGM-SHYZHZOCSA-N 0.000 title 1
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0602632A GB0602632D0 (en) | 2006-02-08 | 2006-02-08 | Preparation Of A Solid Dosage From Comprising Tacrolimus And/Or Sirolimus |
PCT/GB2007/000422 WO2007091059A1 (en) | 2006-02-08 | 2007-02-06 | Preparation and composition of a solid dosage form containing tacrolimus and/or sirolimus |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0602632A GB0602632D0 (en) | 2006-02-08 | 2006-02-08 | Preparation Of A Solid Dosage From Comprising Tacrolimus And/Or Sirolimus |
Publications (1)
Publication Number | Publication Date |
---|---|
GB0602632D0 true GB0602632D0 (en) | 2006-03-22 |
Family
ID=36119804
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GB0602632A Ceased GB0602632D0 (en) | 2006-02-08 | 2006-02-08 | Preparation Of A Solid Dosage From Comprising Tacrolimus And/Or Sirolimus |
Country Status (2)
Country | Link |
---|---|
GB (1) | GB0602632D0 (en) |
WO (1) | WO2007091059A1 (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013022201A1 (en) * | 2011-08-11 | 2013-02-14 | Dong-A Pharm. Co., Ltd. | Process of preparing a stabilized and solubilized formulation of sirolimus derivatives |
HUP1400075A2 (en) | 2014-02-14 | 2015-08-28 | Druggability Technologies Ip Holdco Jersey Ltd | Complexes of sirolimus and its derivatives, process for the preparation thereof and pharmaceutical composition containing them |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8608080D0 (en) * | 1986-04-02 | 1986-05-08 | Fujisawa Pharmaceutical Co | Solid dispersion composition |
ZA9710927B (en) * | 1996-12-06 | 1998-06-15 | Fujisawa Pharmaceutical Co | Pharmaceutical composition. |
CN1133424C (en) * | 1997-06-13 | 2004-01-07 | 惠氏公司 | Rapamycin formulations for oral administration |
-
2006
- 2006-02-08 GB GB0602632A patent/GB0602632D0/en not_active Ceased
-
2007
- 2007-02-06 WO PCT/GB2007/000422 patent/WO2007091059A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
WO2007091059A1 (en) | 2007-08-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
AT | Applications terminated before publication under section 16(1) |