GB201018996D0 - Novel ROCK inhibitors - Google Patents
Novel ROCK inhibitorsInfo
- Publication number
- GB201018996D0 GB201018996D0 GB201018996A GB201018996A GB201018996D0 GB 201018996 D0 GB201018996 D0 GB 201018996D0 GB 201018996 A GB201018996 A GB 201018996A GB 201018996 A GB201018996 A GB 201018996A GB 201018996 D0 GB201018996 D0 GB 201018996D0
- Authority
- GB
- United Kingdom
- Prior art keywords
- rock inhibitors
- novel rock
- novel
- inhibitors
- rock
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- 239000003112 inhibitor Substances 0.000 title 1
- 239000011435 rock Substances 0.000 title 1
Priority Applications (23)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB201018996A GB201018996D0 (en) | 2010-11-10 | 2010-11-10 | Novel ROCK inhibitors |
| CN201180011949.6A CN102884049B (zh) | 2010-11-10 | 2011-03-04 | 用作rock抑制剂的杂环酰胺 |
| EA201201201A EA031616B1 (ru) | 2010-03-02 | 2011-03-04 | Новые ингибиторы rock |
| CN2013102026660A CN103316000A (zh) | 2010-11-10 | 2011-03-04 | 用作rock抑制剂的杂环酰胺 |
| KR1020127025686A KR101794009B1 (ko) | 2010-03-02 | 2011-03-04 | Ｒｏｃｋ 저해제로서 헤테로고리 아미드 |
| SG2012059739A SG183285A1 (en) | 2010-03-02 | 2011-03-04 | Heterocyclic amides as rock inhibitors |
| AU2011222900A AU2011222900B2 (en) | 2010-03-02 | 2011-03-04 | Heterocyclic amides as ROCK inhibitors |
| DK11712789.4T DK2542528T3 (da) | 2010-03-02 | 2011-03-04 | Heterocykliske amider som rock-inhibitorer |
| ES11712789T ES2426410T3 (es) | 2010-03-02 | 2011-03-04 | Amidas heterocíclicas como inhibidores de la ROCK |
| BR112012021889-1A BR112012021889B1 (pt) | 2010-03-02 | 2011-03-04 | Compostos de amidas heterocíclicas e composição que as compreende para a prevenção ou o tratamento de doenças oculares |
| US13/582,195 US8815873B2 (en) | 2010-03-02 | 2011-03-04 | Heterocyclic amides as rock inhibitors |
| CA2791338A CA2791338C (en) | 2010-03-02 | 2011-03-04 | Heterocyclic amides as rock inhibitors |
| PL11712789T PL2542528T3 (pl) | 2010-03-02 | 2011-03-04 | Heterocykliczne amidy jako inhibitory ROCK |
| PCT/EP2011/053343 WO2011107608A1 (en) | 2010-03-02 | 2011-03-04 | Heterocyclic amides as rock inhibitors |
| JP2012555446A JP5710650B2 (ja) | 2010-11-10 | 2011-03-04 | Ｒｏｃｋ阻害剤としての複素環アミド |
| EP11712789.4A EP2542528B1 (en) | 2010-03-02 | 2011-03-04 | Heterocyclic amides as rock inhibitors |
| PT117127894T PT2542528E (pt) | 2010-03-02 | 2011-03-04 | Aminas heterociclicas como inibidores rock |
| MX2012010174A MX2012010174A (es) | 2010-03-02 | 2011-03-04 | Inhibidores novedosos de rock. |
| EP13165882.5A EP2626348A1 (en) | 2010-03-02 | 2011-03-04 | Heterocyclic amides as rock inhibitors |
| NZ602191A NZ602191A (en) | 2010-03-02 | 2011-03-04 | Heterocyclic amides as rock inhibitors |
| ZA2012/06450A ZA201206450B (en) | 2010-03-02 | 2012-08-28 | Heterocyclic amides as rock inhibitors |
| IL221676A IL221676A (en) | 2010-03-02 | 2012-08-28 | Affluent heterocycles as rock inhibitors |
| US13/897,524 US8912209B2 (en) | 2010-03-02 | 2013-05-20 | Rock inhibitors |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB201018996A GB201018996D0 (en) | 2010-11-10 | 2010-11-10 | Novel ROCK inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB201018996D0 true GB201018996D0 (en) | 2010-12-22 |
Family
ID=43414658
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB201018996A Ceased GB201018996D0 (en) | 2010-03-02 | 2010-11-10 | Novel ROCK inhibitors |
Country Status (3)
| Country | Link |
|---|---|
| JP (1) | JP5710650B2 (enExample) |
| CN (2) | CN102884049B (enExample) |
| GB (1) | GB201018996D0 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG11201400058PA (en) * | 2011-08-31 | 2014-03-28 | Amakem Nv | Novel rock kinase inhibitors |
| CN108047193A (zh) * | 2017-12-31 | 2018-05-18 | 佛山市赛维斯医药科技有限公司 | 烷氧噻吩酰胺类rock抑制剂、制备方法及其用途 |
| CN108047195A (zh) * | 2017-12-31 | 2018-05-18 | 佛山市赛维斯医药科技有限公司 | 一种含丙二醇腈基噻吩酰胺类化合物及其用途 |
| CN108191821A (zh) * | 2017-12-31 | 2018-06-22 | 佛山市赛维斯医药科技有限公司 | 一种含甲基萘和腈基噻吩酰胺类结构的rock抑制剂及用途 |
| CN108129452A (zh) * | 2017-12-31 | 2018-06-08 | 佛山市赛维斯医药科技有限公司 | 一种含异丙基萘和丙二醇硝基噻吩酰胺类化合物及其用途 |
| CN107915717A (zh) * | 2017-12-31 | 2018-04-17 | 佛山市赛维斯医药科技有限公司 | 一类含异丙基萘和丙二醇噻吩酰胺类化合物及其用途 |
| CN108047194A (zh) * | 2017-12-31 | 2018-05-18 | 佛山市赛维斯医药科技有限公司 | 含甲基萘和丙二醇噻吩酰胺类化合物、制备方法及其用途 |
| CN108101885A (zh) * | 2017-12-31 | 2018-06-01 | 佛山市赛维斯医药科技有限公司 | 含异丙胺和硝基噻吩酰胺类结构化合物、其制备方法及用途 |
| CN107935986A (zh) * | 2017-12-31 | 2018-04-20 | 佛山市赛维斯医药科技有限公司 | 异丙胺和卤代噻吩酰胺类结构化合物、其制备方法及用途 |
| CN107935987A (zh) * | 2017-12-31 | 2018-04-20 | 佛山市赛维斯医药科技有限公司 | 含甲基萘和噻吩酰胺结构的rock抑制剂、制备方法及其用途 |
| CN108191820A (zh) * | 2017-12-31 | 2018-06-22 | 佛山市赛维斯医药科技有限公司 | 一种含异丙胺和噻吩酰胺类结构的化合物 |
| CN114956977B (zh) * | 2022-06-09 | 2024-03-26 | 朗捷睿(苏州)生物科技有限公司 | 一种联苯类化合物、药物组合物及其制备方法和应用 |
| CN120569383A (zh) * | 2023-01-13 | 2025-08-29 | 武汉朗来科技发展有限公司 | 一种rock抑制剂中间体的制备方法 |
| CN119569655B (zh) * | 2024-11-21 | 2025-11-11 | 西北大学 | 含吡唑甲酰胺基的苯甲酸氟甲基硫酯类化合物及其制备方法与应用 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007006547A1 (en) * | 2005-07-11 | 2007-01-18 | Devgen N.V. | Amide derivatives as kinase inhibitors |
| CN101248046A (zh) * | 2005-07-11 | 2008-08-20 | 德福根有限公司 | 作为激酶抑制剂的酰胺衍生物 |
| CN101287707A (zh) * | 2005-10-13 | 2008-10-15 | 德福根有限公司 | 激酶抑制剂 |
| JP2009536947A (ja) * | 2006-05-12 | 2009-10-22 | バーテックス ファーマシューティカルズ インコーポレイテッド | Ｒｏｃｋプロテインキナーゼの選択的阻害剤およびその使用方法 |
| MX2010002272A (es) * | 2007-08-27 | 2010-08-09 | Abbott Gmbh & Co Kg | 4-(4-piridinil)-benzamidas y su uso como moduladores de la actividad de rho-cinasa (rock). |
| EP2331507A2 (en) * | 2008-09-18 | 2011-06-15 | Astellas Pharma Inc. | Heterocyclic carboxamide compounds |
-
2010
- 2010-11-10 GB GB201018996A patent/GB201018996D0/en not_active Ceased
-
2011
- 2011-03-04 CN CN201180011949.6A patent/CN102884049B/zh not_active Expired - Fee Related
- 2011-03-04 CN CN2013102026660A patent/CN103316000A/zh active Pending
- 2011-03-04 JP JP2012555446A patent/JP5710650B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP2013527136A (ja) | 2013-06-27 |
| CN102884049A (zh) | 2013-01-16 |
| CN102884049B (zh) | 2016-08-24 |
| CN103316000A (zh) | 2013-09-25 |
| JP5710650B2 (ja) | 2015-04-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AT | Applications terminated before publication under section 16(1) |