GB1463520A - Process for the production of imidazolines - Google Patents

Process for the production of imidazolines

Info

Publication number
GB1463520A
GB1463520A GB3914374A GB3914374A GB1463520A GB 1463520 A GB1463520 A GB 1463520A GB 3914374 A GB3914374 A GB 3914374A GB 3914374 A GB3914374 A GB 3914374A GB 1463520 A GB1463520 A GB 1463520A
Authority
GB
United Kingdom
Prior art keywords
formula
positions
compound
quinoxaline
aminoethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB3914374A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
PFIZER Ltd
Original Assignee
PFIZER Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by PFIZER Ltd filed Critical PFIZER Ltd
Priority to GB3914374A priority Critical patent/GB1463520A/en
Priority to SE7509271A priority patent/SE7509271L/xx
Priority to AU84305/75A priority patent/AU489162B2/en
Priority to CA234,270A priority patent/CA1043791A/en
Priority to DE19752538620 priority patent/DE2538620A1/de
Priority to JP50105862A priority patent/JPS51149291A/ja
Priority to LU73327A priority patent/LU73327A1/xx
Priority to FI752487A priority patent/FI752487A7/fi
Priority to BE159796A priority patent/BE833135A/xx
Priority to ES440760A priority patent/ES440760A1/es
Priority to DK398775A priority patent/DK398775A/da
Priority to NL7510473A priority patent/NL7510473A/xx
Priority to FR7527324A priority patent/FR2283899A1/fr
Publication of GB1463520A publication Critical patent/GB1463520A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
GB3914374A 1974-09-06 1974-09-06 Process for the production of imidazolines Expired GB1463520A (en)

Priority Applications (13)

Application Number Priority Date Filing Date Title
GB3914374A GB1463520A (en) 1974-09-06 1974-09-06 Process for the production of imidazolines
SE7509271A SE7509271L (sv) 1974-09-06 1975-08-25 Sett att framstella kinoxalin- och kinazolinderivat
AU84305/75A AU489162B2 (en) 1974-09-06 1975-08-27 Process for preparing imidazolinylamnquinoxalines
CA234,270A CA1043791A (en) 1974-09-06 1975-08-27 Process for preparing imidazolinylaminoquinoxalines
DE19752538620 DE2538620A1 (de) 1974-09-06 1975-08-29 Verfahren zur herstellung von chinoxalin- und chinazolinderivaten
JP50105862A JPS51149291A (en) 1974-09-06 1975-09-01 Preparation method of imidazolinylaminoquinoxaline and quinazolines
LU73327A LU73327A1 (enExample) 1974-09-06 1975-09-04
FI752487A FI752487A7 (enExample) 1974-09-06 1975-09-04
BE159796A BE833135A (fr) 1974-09-06 1975-09-05 Procede de preparation de derives de quinoxaline, et quinazoline
ES440760A ES440760A1 (es) 1974-09-06 1975-09-05 Procedimiento para preparar derivados de quinoxalina y qui- nazolina.
DK398775A DK398775A (da) 1974-09-06 1975-09-05 Fremgangsmade til fremstilling af derivater af quinoxalin og quinazolin
NL7510473A NL7510473A (nl) 1974-09-06 1975-09-05 Werkwijze ter bereiding van chinoxalinederivaten.
FR7527324A FR2283899A1 (fr) 1974-09-06 1975-09-05 Procede de preparation de derives de quinazoline

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB3914374A GB1463520A (en) 1974-09-06 1974-09-06 Process for the production of imidazolines

Publications (1)

Publication Number Publication Date
GB1463520A true GB1463520A (en) 1977-02-02

Family

ID=10407882

Family Applications (1)

Application Number Title Priority Date Filing Date
GB3914374A Expired GB1463520A (en) 1974-09-06 1974-09-06 Process for the production of imidazolines

Country Status (12)

Country Link
JP (1) JPS51149291A (enExample)
BE (1) BE833135A (enExample)
CA (1) CA1043791A (enExample)
DE (1) DE2538620A1 (enExample)
DK (1) DK398775A (enExample)
ES (1) ES440760A1 (enExample)
FI (1) FI752487A7 (enExample)
FR (1) FR2283899A1 (enExample)
GB (1) GB1463520A (enExample)
LU (1) LU73327A1 (enExample)
NL (1) NL7510473A (enExample)
SE (1) SE7509271L (enExample)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5552403A (en) * 1993-10-13 1996-09-03 Allergan Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US6323204B1 (en) 1993-10-13 2001-11-27 Allergan Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US7265117B2 (en) 2004-05-06 2007-09-04 Alcon, Inc. Topical brimonidine tartrate formulations that lack chlorine dioxide

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5326763A (en) * 1989-10-12 1994-07-05 Allergan, Inc. Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US5077292A (en) * 1989-10-12 1991-12-31 Allergan, Inc. (2-imidazolin-2-ylamino) tetrahydroquinoxalines and methods for using same
US5198442A (en) * 1989-10-12 1993-03-30 Allergan, Inc. (2-imidazolin-2-ylamino) quinoxaline derivatives and methods for using same
US5204347A (en) * 1989-10-12 1993-04-20 Allergan, Inc. Methods for using (2-imidazolin-2-ylamino) tetrahydroquinoxalines
US5112822A (en) * 1989-10-12 1992-05-12 Allergan, Inc. (2-imidazolin-2-ylamino) quinoxaline derivatives and methods for using same
US5021416A (en) * 1989-10-31 1991-06-04 Allergan, Inc. Method for using (2-imidazolin-2-ylamino) quinoxalines to reduce or maintain intraocular pressure
US5130441A (en) * 1990-02-06 1992-07-14 Allergan, Inc. Method for producing amino-2-imidazoline derivatives
US5237072A (en) * 1990-02-06 1993-08-17 Allergan, Inc. Method for producing amino-2-imidazoline derivatives
RU2285003C1 (ru) * 2005-04-29 2006-10-10 Федеральное государственное унитарное предприятие "Центр по химии лекарственных средств" (ФГУП ЦХЛС-ВНИХФИ) Способ получения 5-бром-6-[(2-имидазолин-2-ил)амино]хиноксалина l-тартрата
ES2818073T3 (es) 2013-12-24 2021-04-09 Sentiss Pharma Private Ltd Solución oftálmica de tartrato de brimonidina tópica
JP6339364B2 (ja) * 2013-12-27 2018-06-06 カズマパートナーズ株式会社 無定形ブリモニジン酒石酸塩及びその製造方法
JP6270603B2 (ja) * 2014-04-14 2018-01-31 カズマパートナーズ株式会社 ブリモニジン酒石酸塩の新規多形及びその製造方法
UA129938C2 (uk) 2020-04-29 2025-09-17 Сентісс Фарма Прайвет Лімітед Офтальмологічні композиції, що містять комбінацію бринзоламіду та бримонідину

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE795970A (fr) * 1972-02-29 1973-08-27 Pfizer Nouveaux derives de quinoleine, quinoxaline et quinazoline er composition pharmaceutiques les contenant

Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5552403A (en) * 1993-10-13 1996-09-03 Allergan Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US5561132A (en) * 1993-10-13 1996-10-01 Allergan Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US5587376A (en) * 1993-10-13 1996-12-24 Allergan Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US5703077A (en) * 1993-10-13 1997-12-30 Allergan Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US5714486A (en) * 1993-10-13 1998-02-03 Allergan Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US5756503A (en) * 1993-10-13 1998-05-26 Allergan Methods for using (2-imidazolin-2-ylamino) Quinoxaline derivatives
US5773440A (en) * 1993-10-13 1998-06-30 Allergan Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US6323204B1 (en) 1993-10-13 2001-11-27 Allergan Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US7265117B2 (en) 2004-05-06 2007-09-04 Alcon, Inc. Topical brimonidine tartrate formulations that lack chlorine dioxide

Also Published As

Publication number Publication date
SE7509271L (sv) 1975-12-29
DK398775A (da) 1976-03-07
FI752487A7 (enExample) 1976-03-07
ES440760A1 (es) 1977-04-01
BE833135A (fr) 1976-03-05
CA1043791A (en) 1978-12-05
NL7510473A (nl) 1976-03-09
JPS51149291A (en) 1976-12-22
DE2538620A1 (de) 1976-03-18
AU8430575A (en) 1977-03-03
LU73327A1 (enExample) 1977-05-11
FR2283899A1 (fr) 1976-04-02

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Legal Events

Date Code Title Description
PS Patent sealed [section 19, patents act 1949]
PCNP Patent ceased through non-payment of renewal fee