GB1458185A - Carboxyl and tetrazolyl cerivatives of thioxanthones methods for their preparation and compositions containing them - Google Patents
Carboxyl and tetrazolyl cerivatives of thioxanthones methods for their preparation and compositions containing themInfo
- Publication number
- GB1458185A GB1458185A GB4143372A GB4143372A GB1458185A GB 1458185 A GB1458185 A GB 1458185A GB 4143372 A GB4143372 A GB 4143372A GB 4143372 A GB4143372 A GB 4143372A GB 1458185 A GB1458185 A GB 1458185A
- Authority
- GB
- United Kingdom
- Prior art keywords
- group
- tetrazolyl
- alkyl
- carboxyl
- carbon atoms
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 125000003831 tetrazolyl group Chemical group 0.000 title abstract 5
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 title abstract 4
- 239000000203 mixture Substances 0.000 title 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 4
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- -1 5-tetrazolyl Chemical group 0.000 abstract 2
- 230000002378 acidificating effect Effects 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 206010020751 Hypersensitivity Diseases 0.000 abstract 1
- 239000002841 Lewis acid Substances 0.000 abstract 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 150000007513 acids Chemical class 0.000 abstract 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 125000004442 acylamino group Chemical group 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 230000009435 amidation Effects 0.000 abstract 1
- 238000007112 amidation reaction Methods 0.000 abstract 1
- 150000001408 amides Chemical class 0.000 abstract 1
- LTYMSROWYAPPGB-UHFFFAOYSA-N diphenyl sulfide Chemical class C=1C=CC=CC=1SC1=CC=CC=C1 LTYMSROWYAPPGB-UHFFFAOYSA-N 0.000 abstract 1
- 230000032050 esterification Effects 0.000 abstract 1
- 238000005886 esterification reaction Methods 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 150000007517 lewis acids Chemical class 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
- YRHRIQCWCFGUEQ-UHFFFAOYSA-N thioxanthen-9-one Chemical class C1=CC=C2C(=O)C3=CC=CC=C3SC2=C1 YRHRIQCWCFGUEQ-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
- C07D335/04—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D335/10—Dibenzothiopyrans; Hydrogenated dibenzothiopyrans
- C07D335/12—Thioxanthenes
- C07D335/14—Thioxanthenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 9
- C07D335/16—Oxygen atoms, e.g. thioxanthones
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Priority Applications (22)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB4143372A GB1458185A (en) | 1972-09-06 | 1972-09-06 | Carboxyl and tetrazolyl cerivatives of thioxanthones methods for their preparation and compositions containing them |
| AU60035/73A AU488547B2 (en) | 1973-09-05 | Sulphur ring compounds | |
| ZA00737106A ZA737106B (en) | 1972-09-06 | 1973-09-05 | Sulphur ring compounds |
| ES418514A ES418514A1 (es) | 1972-09-06 | 1973-09-05 | Un metodo para preparar compuestos triciclicos sustituidos con tetrazolilo. |
| HU73WE00000497A HU172110B (hu) | 1972-09-06 | 1973-09-05 | Sposob poluchenija triciklicheskikh soedinenij sery i farmacevticheskikh preparatov soderzhahhikh takie soedinenija |
| DE19732344799 DE2344799A1 (de) | 1972-09-06 | 1973-09-05 | Schwefelhaltige tricyclische verbindungen und diese enthaltende arzneimittel |
| IL43162A IL43162A0 (en) | 1972-09-06 | 1973-09-05 | Pharmaceutical compositions containing tricyclic sulphur compounds,certain such novel compounds and their preparation |
| NL7312253A NL7312253A (enrdf_load_stackoverflow) | 1972-09-06 | 1973-09-06 | |
| CS736213A CS188902B2 (en) | 1972-09-06 | 1973-09-06 | Method of producing derivatives of thioxanthone |
| JP48100727A JPS5829309B2 (ja) | 1972-09-06 | 1973-09-06 | コウアレルギ−セイサンカンシキカゴウブツノ セイゾウホウホウ |
| IE1590/73A IE38329B1 (en) | 1972-09-06 | 1973-09-06 | Carboxyl and tetrazolyl derivatives of thioxanthones methods for their preparation and compisitions containing them |
| BE135398A BE804554A (fr) | 1972-09-06 | 1973-09-06 | Composes cycliques sulfures |
| FR7332118A FR2197607B1 (enrdf_load_stackoverflow) | 1972-09-06 | 1973-09-06 | |
| CH1282773A CH614203A5 (en) | 1972-09-06 | 1973-09-06 | Process for the preparation of thioxanthone derivatives |
| CA180,382A CA1023365A (en) | 1972-09-06 | 1973-09-06 | Sulphur ring compounds |
| DK54975A DK54975A (enrdf_load_stackoverflow) | 1972-09-06 | 1975-02-14 | |
| CS758021A CS188948B2 (en) | 1972-09-06 | 1975-11-26 | Process for preparing derivatives of thioxanthone |
| CS758020A CS188947B2 (en) | 1972-09-06 | 1975-11-26 | Method of producing derivatives of thioxanthone |
| ES443476A ES443476A1 (es) | 1972-09-06 | 1975-12-13 | Un metodo de preparar una composicion farmaceutica que com- prende una tioxantona sustituida con carboxi. |
| FR7600805A FR2289184A1 (fr) | 1972-09-06 | 1976-01-14 | Medicament contenant un derive de carboxy-thioxanthone |
| CA266,840A CA1023269A (en) | 1972-09-06 | 1976-11-30 | Pharmaceutical composition containing sulphur ring compound |
| JP57225769A JPS5919955B2 (ja) | 1972-09-06 | 1982-12-22 | 抗アレルギ−性三環式化合物の製造方法 |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB4143372A GB1458185A (en) | 1972-09-06 | 1972-09-06 | Carboxyl and tetrazolyl cerivatives of thioxanthones methods for their preparation and compositions containing them |
| GB3341073 | 1973-07-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1458185A true GB1458185A (en) | 1976-12-08 |
Family
ID=26261859
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB4143372A Expired GB1458185A (en) | 1972-09-06 | 1972-09-06 | Carboxyl and tetrazolyl cerivatives of thioxanthones methods for their preparation and compositions containing them |
Country Status (10)
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4348530A (en) | 1980-02-05 | 1982-09-07 | Ciba-Geigy Corporation | Thioxanthonecarboxylic acids, esters, thioesters and amides with reactive functional groups |
| US4367324A (en) | 1980-02-05 | 1983-01-04 | Ciba-Geigy Corporation | Photocrosslinkable polymers with thioxanthone and imidyl groupings in side chains |
| US4385182A (en) | 1980-05-06 | 1983-05-24 | Ciba-Geigy Corporation | Thioxanthonecarboxylic acids and thioxanthonecarboxylic acid derivatives |
| GB2119364A (en) * | 1979-05-18 | 1983-11-16 | Ciba Geigy Ag | Phenylthio-phthalic acids and their production |
| US4623656A (en) | 1984-01-05 | 1986-11-18 | Morton Harfenist | Method for inhibiting monoamine oxidase-A and treating depression by administering 3-N-methyl-thioxanthen-9-one carboxamide 10,10-dioxide |
| US4737514A (en) * | 1984-01-05 | 1988-04-12 | Burroughs Wellcome Co. | Method for treating depression with thioxanthen-9-one derivatives |
| US11618742B2 (en) | 2018-02-16 | 2023-04-04 | Adeka Corporation | Radical polymerization initiator, composition containing same, cured product of composition, production method for cured product, and compound |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS55122785A (en) * | 1979-03-15 | 1980-09-20 | Yoshitomi Pharmaceut Ind Ltd | Preparation of benzopyranopyridine derivative |
| US4564578A (en) * | 1982-11-25 | 1986-01-14 | Ciba-Geigy Corporation | Novel thioxanthones substituted by alpha-aminoalkyl groups |
| EP0150891A1 (en) * | 1984-01-05 | 1985-08-07 | The Wellcome Foundation Limited | Tricyclic compounds, processes for their preparation, compositions containing such compounds and their use in medicine |
| CN101906095B (zh) * | 2010-07-06 | 2013-08-14 | 天津久日化学股份有限公司 | 噻吨酮-4-羧酸酯及制备方法和光引发剂组合物与应用 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE793954A (fr) * | 1972-07-19 | 1973-07-12 | Syntex Corp | Acides thioxanthone-carboxyliques et leurs derives |
-
1972
- 1972-09-06 GB GB4143372A patent/GB1458185A/en not_active Expired
-
1973
- 1973-09-05 DE DE19732344799 patent/DE2344799A1/de not_active Ceased
- 1973-09-05 ES ES418514A patent/ES418514A1/es not_active Expired
- 1973-09-05 IL IL43162A patent/IL43162A0/xx unknown
- 1973-09-06 FR FR7332118A patent/FR2197607B1/fr not_active Expired
- 1973-09-06 IE IE1590/73A patent/IE38329B1/xx unknown
- 1973-09-06 JP JP48100727A patent/JPS5829309B2/ja not_active Expired
- 1973-09-06 NL NL7312253A patent/NL7312253A/xx not_active Application Discontinuation
- 1973-09-06 CA CA180,382A patent/CA1023365A/en not_active Expired
- 1973-09-06 CH CH1282773A patent/CH614203A5/xx not_active IP Right Cessation
-
1975
- 1975-12-13 ES ES443476A patent/ES443476A1/es not_active Expired
-
1976
- 1976-01-14 FR FR7600805A patent/FR2289184A1/fr active Granted
Cited By (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2119364A (en) * | 1979-05-18 | 1983-11-16 | Ciba Geigy Ag | Phenylthio-phthalic acids and their production |
| US4505794A (en) * | 1979-05-18 | 1985-03-19 | Ciba-Geigy Corporation | Thioxanthonecarboxylic acid esters, thioesters and amides |
| US4348530A (en) | 1980-02-05 | 1982-09-07 | Ciba-Geigy Corporation | Thioxanthonecarboxylic acids, esters, thioesters and amides with reactive functional groups |
| US4367324A (en) | 1980-02-05 | 1983-01-04 | Ciba-Geigy Corporation | Photocrosslinkable polymers with thioxanthone and imidyl groupings in side chains |
| US4594400A (en) * | 1980-02-05 | 1986-06-10 | Ciba-Geigy Corporation | Thioxanthonecarboxylic acids, esters thioesters and amides with reactive functional groups and polymers prepared therefrom and having thioxanthone radicals as side chains |
| US4385182A (en) | 1980-05-06 | 1983-05-24 | Ciba-Geigy Corporation | Thioxanthonecarboxylic acids and thioxanthonecarboxylic acid derivatives |
| US4623656A (en) | 1984-01-05 | 1986-11-18 | Morton Harfenist | Method for inhibiting monoamine oxidase-A and treating depression by administering 3-N-methyl-thioxanthen-9-one carboxamide 10,10-dioxide |
| US4737514A (en) * | 1984-01-05 | 1988-04-12 | Burroughs Wellcome Co. | Method for treating depression with thioxanthen-9-one derivatives |
| US11618742B2 (en) | 2018-02-16 | 2023-04-04 | Adeka Corporation | Radical polymerization initiator, composition containing same, cured product of composition, production method for cured product, and compound |
Also Published As
| Publication number | Publication date |
|---|---|
| IE38329B1 (en) | 1978-02-15 |
| DE2344799A1 (de) | 1974-03-21 |
| NL7312253A (enrdf_load_stackoverflow) | 1974-03-08 |
| JPS4992072A (enrdf_load_stackoverflow) | 1974-09-03 |
| ES418514A1 (es) | 1977-01-01 |
| IL43162A0 (en) | 1973-11-28 |
| CH614203A5 (en) | 1979-11-15 |
| FR2197607A1 (enrdf_load_stackoverflow) | 1974-03-29 |
| FR2289184A1 (fr) | 1976-05-28 |
| AU6003573A (en) | 1975-03-06 |
| FR2197607B1 (enrdf_load_stackoverflow) | 1977-01-28 |
| CA1023365A (en) | 1977-12-27 |
| JPS5829309B2 (ja) | 1983-06-22 |
| ES443476A1 (es) | 1977-08-16 |
| IE38329L (en) | 1974-03-06 |
| FR2289184B1 (enrdf_load_stackoverflow) | 1979-09-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| PCNP | Patent ceased through non-payment of renewal fee |