GB1330072A - Oestradiol derivative and a process for its manufacture - Google Patents
Oestradiol derivative and a process for its manufactureInfo
- Publication number
- GB1330072A GB1330072A GB1042871*[A GB1042871A GB1330072A GB 1330072 A GB1330072 A GB 1330072A GB 1042871 A GB1042871 A GB 1042871A GB 1330072 A GB1330072 A GB 1330072A
- Authority
- GB
- United Kingdom
- Prior art keywords
- methyl
- estradiol
- ethynyl
- april
- manufacture
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/168—Steroids
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/184—Hormones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general
Landscapes
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Polymers & Plastics (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Husbandry (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Food Science & Technology (AREA)
- General Health & Medical Sciences (AREA)
- Endocrinology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Steroid Compounds (AREA)
Abstract
1330072 The 3-cyclopentyl ether of 7α-methyl- 17α - ethynyl - estradiol CIBA - GEIGY AG 21 April 1971 [24 April 1970] 10428/71 Heading C2U The title compound is prepared by etherification of 7α-methyl-17α-ethynyl-estradiol, by reacting the diol or a salt thereof with a reactive ester of cyclopentanol, or by ethynylation with an acetylene metal compound of 3-cyclopentyloxy - 7α - methyl - 17 - oxo - #<SP>1,3,5(10)</SP> - estratriene. The novel steroid is stated to have estrogenic, uterotropic and blastocyte implantation inhibiting action, and it may be made up into pharmaceutical and veterinary compositions with suitable carriers. Specification 1,330,071 is referred to.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH621870A CH536291A (en) | 1970-04-24 | 1970-04-24 | Process for the production of a new, highly estrogenic steroid |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1330072A true GB1330072A (en) | 1973-09-12 |
Family
ID=4306140
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB1042871*[A Expired GB1330072A (en) | 1970-04-24 | 1971-04-21 | Oestradiol derivative and a process for its manufacture |
Country Status (19)
| Country | Link |
|---|---|
| AT (2) | AT306261B (en) |
| BE (1) | BE766183A (en) |
| CA (1) | CA921022A (en) |
| CH (2) | CH536291A (en) |
| CS (2) | CS161776B2 (en) |
| DE (1) | DE2118997A1 (en) |
| DK (2) | DK129580B (en) |
| ES (2) | ES390460A1 (en) |
| FI (1) | FI48826C (en) |
| FR (1) | FR2092081B1 (en) |
| GB (1) | GB1330072A (en) |
| HU (1) | HU162383B (en) |
| IE (1) | IE35146B1 (en) |
| IL (1) | IL36653A (en) |
| NL (1) | NL7105577A (en) |
| PL (2) | PL71122B1 (en) |
| SE (1) | SE373576B (en) |
| SU (2) | SU383287A3 (en) |
| ZA (1) | ZA712524B (en) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1434174A (en) * | 1963-12-24 | 1966-04-08 | Ciba Geigy | Process for the preparation of new steroids of the estrane series |
| BE755689A (en) * | 1969-09-03 | 1971-03-03 | Upjohn Co | NEW 7 BETA-ALKYL-19- NORTESTOSTERONES MANUFACTURING PROCESS |
-
1970
- 1970-04-24 CH CH621870A patent/CH536291A/en not_active IP Right Cessation
- 1970-04-24 CH CH1870172A patent/CH536293A/en not_active IP Right Cessation
-
1971
- 1971-04-19 CA CA110655A patent/CA921022A/en not_active Expired
- 1971-04-19 IL IL36653A patent/IL36653A/en unknown
- 1971-04-20 DE DE19712118997 patent/DE2118997A1/en active Pending
- 1971-04-20 IE IE490/71A patent/IE35146B1/en unknown
- 1971-04-20 ZA ZA712524A patent/ZA712524B/en unknown
- 1971-04-21 GB GB1042871*[A patent/GB1330072A/en not_active Expired
- 1971-04-22 ES ES390460A patent/ES390460A1/en not_active Expired
- 1971-04-22 PL PL1971147686A patent/PL71122B1/pl unknown
- 1971-04-22 HU HUCI1105A patent/HU162383B/hu unknown
- 1971-04-22 PL PL1971178220A patent/PL83828B1/pl unknown
- 1971-04-22 FR FR7114321A patent/FR2092081B1/fr not_active Expired
- 1971-04-23 SE SE7105302A patent/SE373576B/en unknown
- 1971-04-23 BE BE766183A patent/BE766183A/en unknown
- 1971-04-23 AT AT351071A patent/AT306261B/en not_active IP Right Cessation
- 1971-04-23 FI FI711130A patent/FI48826C/en active
- 1971-04-23 AT AT234272A patent/AT315394B/en not_active IP Right Cessation
- 1971-04-23 SU SU1649254A patent/SU383287A3/ru active
- 1971-04-23 CS CS1883A patent/CS161776B2/cs unknown
- 1971-04-23 DK DK197071AA patent/DK129580B/en unknown
- 1971-04-23 NL NL7105577A patent/NL7105577A/xx unknown
- 1971-04-23 SU SU711649254D patent/SU399116A3/ru active
- 1971-04-23 CS CS2985A patent/CS161775B2/cs unknown
-
1972
- 1972-08-18 DK DK412072AA patent/DK128316B/en unknown
-
1973
- 1973-07-16 ES ES416953A patent/ES416953A1/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| AT315394B (en) | 1974-05-27 |
| PL71122B1 (en) | 1974-04-30 |
| DE2118997A1 (en) | 1971-11-11 |
| FR2092081A1 (en) | 1972-01-21 |
| FI48826B (en) | 1974-09-30 |
| IE35146B1 (en) | 1975-11-26 |
| AT306261B (en) | 1973-04-10 |
| IE35146L (en) | 1971-10-24 |
| SE373576B (en) | 1975-02-10 |
| CH536291A (en) | 1973-04-30 |
| CS161775B2 (en) | 1975-06-10 |
| DK128316B (en) | 1974-04-08 |
| IL36653A (en) | 1974-07-31 |
| BE766183A (en) | 1971-10-25 |
| ZA712524B (en) | 1972-01-26 |
| FR2092081B1 (en) | 1974-10-18 |
| IL36653A0 (en) | 1971-06-23 |
| DK129580C (en) | 1975-04-28 |
| ES416953A1 (en) | 1976-03-16 |
| CH536293A (en) | 1973-04-30 |
| CA921022A (en) | 1973-02-13 |
| ES390460A1 (en) | 1974-07-01 |
| PL83828B1 (en) | 1976-02-28 |
| HU162383B (en) | 1973-02-28 |
| SU399116A3 (en) | 1973-09-27 |
| SU383287A3 (en) | 1973-05-25 |
| NL7105577A (en) | 1971-10-26 |
| DK129580B (en) | 1974-10-28 |
| CS161776B2 (en) | 1975-06-10 |
| FI48826C (en) | 1975-01-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| PCNP | Patent ceased through non-payment of renewal fee |