GB1183135A - 2,4-Benzodiazepines, process for their manufacture and Compositions containing them - Google Patents
2,4-Benzodiazepines, process for their manufacture and Compositions containing themInfo
- Publication number
- GB1183135A GB1183135A GB1694368A GB1694368A GB1183135A GB 1183135 A GB1183135 A GB 1183135A GB 1694368 A GB1694368 A GB 1694368A GB 1694368 A GB1694368 A GB 1694368A GB 1183135 A GB1183135 A GB 1183135A
- Authority
- GB
- United Kingdom
- Prior art keywords
- aliphatic
- araliphatic
- heteroaryl
- aromatic
- residue
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/04—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US63049767A | 1967-04-13 | 1967-04-13 | |
US69442167A | 1967-12-29 | 1967-12-29 |
Publications (1)
Publication Number | Publication Date |
---|---|
GB1183135A true GB1183135A (en) | 1970-03-04 |
Family
ID=27091165
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GB1694368A Expired GB1183135A (en) | 1967-04-13 | 1968-04-09 | 2,4-Benzodiazepines, process for their manufacture and Compositions containing them |
Country Status (5)
Country | Link |
---|---|
BE (1) | BE713698A (de) |
CH (3) | CH523264A (de) |
DE (1) | DE1770135A1 (de) |
FR (2) | FR1588463A (de) |
GB (1) | GB1183135A (de) |
Cited By (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU639821B2 (en) * | 1990-09-10 | 1993-08-05 | Sanofi | Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents |
EP0597540A1 (de) * | 1992-11-10 | 1994-05-18 | Sterling Winthrop Inc. | Aryl und Hetaryl annelierte 2,4-Diazocine als anti-arryhthmische Wirkstoffe |
US5380721A (en) * | 1990-09-10 | 1995-01-10 | Sterling Winthrop Inc. | Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents |
WO1996019440A1 (en) * | 1994-12-20 | 1996-06-27 | The Wellcome Foundation Limited | Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase |
JP2009513656A (ja) * | 2005-10-27 | 2009-04-02 | シェーリング コーポレイション | 複素環式アスパルチルプロテアーゼインヒビター |
CN101671307A (zh) * | 2003-12-15 | 2010-03-17 | 先灵公司 | 杂环天冬氨酰蛋白酶抑制剂 |
-
1968
- 1968-03-25 CH CH257971A patent/CH523264A/de not_active IP Right Cessation
- 1968-03-25 CH CH258071A patent/CH527828A/de not_active IP Right Cessation
- 1968-03-25 CH CH435768A patent/CH511863A/de not_active IP Right Cessation
- 1968-04-05 DE DE19681770135 patent/DE1770135A1/de active Pending
- 1968-04-09 GB GB1694368A patent/GB1183135A/en not_active Expired
- 1968-04-11 FR FR1588463D patent/FR1588463A/fr not_active Expired
- 1968-04-12 BE BE713698D patent/BE713698A/xx unknown
- 1968-07-02 FR FR157515A patent/FR7495M/fr not_active Expired
Cited By (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU639821B2 (en) * | 1990-09-10 | 1993-08-05 | Sanofi | Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents |
US5380721A (en) * | 1990-09-10 | 1995-01-10 | Sterling Winthrop Inc. | Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents |
US5624922A (en) * | 1990-09-10 | 1997-04-29 | Sterling Winthrop Inc. | Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents |
EP0597540A1 (de) * | 1992-11-10 | 1994-05-18 | Sterling Winthrop Inc. | Aryl und Hetaryl annelierte 2,4-Diazocine als anti-arryhthmische Wirkstoffe |
WO1996019440A1 (en) * | 1994-12-20 | 1996-06-27 | The Wellcome Foundation Limited | Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase |
US5866612A (en) * | 1994-12-20 | 1999-02-02 | Glaxo Wellcome Inc. | Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase |
USRE37438E1 (en) | 1994-12-20 | 2001-11-06 | Glaxo Wellcome Inc. | Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase |
CN101671307A (zh) * | 2003-12-15 | 2010-03-17 | 先灵公司 | 杂环天冬氨酰蛋白酶抑制剂 |
CN102627609A (zh) * | 2003-12-15 | 2012-08-08 | 先灵公司 | 杂环天冬氨酰蛋白酶抑制剂 |
CN101671307B (zh) * | 2003-12-15 | 2014-05-14 | 默沙东公司 | 杂环天冬氨酰蛋白酶抑制剂 |
CN102627609B (zh) * | 2003-12-15 | 2016-05-04 | 默沙东公司 | 杂环天冬氨酰蛋白酶抑制剂 |
JP2009513656A (ja) * | 2005-10-27 | 2009-04-02 | シェーリング コーポレイション | 複素環式アスパルチルプロテアーゼインヒビター |
Also Published As
Publication number | Publication date |
---|---|
BE713698A (de) | 1968-10-14 |
FR1588463A (de) | 1970-04-17 |
DE1770135A1 (de) | 1971-09-23 |
CH527828A (de) | 1972-09-15 |
CH523264A (de) | 1972-05-31 |
FR7495M (de) | 1969-12-08 |
CH511863A (de) | 1971-08-31 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PS | Patent sealed | ||
PLNP | Patent lapsed through nonpayment of renewal fees |