GB1168361A - Hydroxyphenyl Substituted Cyclic and Acyclic Amidines and derivatives thereof - Google Patents
Hydroxyphenyl Substituted Cyclic and Acyclic Amidines and derivatives thereofInfo
- Publication number
- GB1168361A GB1168361A GB52098/67A GB5209867A GB1168361A GB 1168361 A GB1168361 A GB 1168361A GB 52098/67 A GB52098/67 A GB 52098/67A GB 5209867 A GB5209867 A GB 5209867A GB 1168361 A GB1168361 A GB 1168361A
- Authority
- GB
- United Kingdom
- Prior art keywords
- methyl
- hydrogen
- derivatives
- compositions
- ethylene
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- -1 Acyclic Amidines Chemical class 0.000 title abstract 2
- 125000004122 cyclic group Chemical group 0.000 title 1
- 125000004464 hydroxyphenyl group Chemical group 0.000 title 1
- 239000001257 hydrogen Substances 0.000 abstract 4
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 4
- 239000000203 mixture Substances 0.000 abstract 3
- VGGSQFUCUMXWEO-UHFFFAOYSA-N Ethene Chemical compound C=C VGGSQFUCUMXWEO-UHFFFAOYSA-N 0.000 abstract 2
- 239000005977 Ethylene Substances 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 230000000507 anthelmentic effect Effects 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 2
- 150000002431 hydrogen Chemical group 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 125000003903 2-propenyl group Chemical group [H]C([*])([H])C([H])=C([H])[H] 0.000 abstract 1
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
- 108010003272 Hyaluronate lyase Proteins 0.000 abstract 1
- 102000001974 Hyaluronidases Human genes 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
- 229910052794 bromium Inorganic materials 0.000 abstract 1
- 239000002775 capsule Substances 0.000 abstract 1
- 125000001589 carboacyl group Chemical group 0.000 abstract 1
- 229910052801 chlorine Inorganic materials 0.000 abstract 1
- 239000000460 chlorine Substances 0.000 abstract 1
- 239000003651 drinking water Substances 0.000 abstract 1
- 235000020188 drinking water Nutrition 0.000 abstract 1
- 239000003937 drug carrier Substances 0.000 abstract 1
- 229960002773 hyaluronidase Drugs 0.000 abstract 1
- PNDPGZBMCMUPRI-UHFFFAOYSA-N iodine Chemical compound II PNDPGZBMCMUPRI-UHFFFAOYSA-N 0.000 abstract 1
- 229960005015 local anesthetics Drugs 0.000 abstract 1
- 231100000252 nontoxic Toxicity 0.000 abstract 1
- 230000003000 nontoxic effect Effects 0.000 abstract 1
- 238000007911 parenteral administration Methods 0.000 abstract 1
- 239000000843 powder Substances 0.000 abstract 1
- 125000003258 trimethylene group Chemical group [H]C([H])([*:2])C([H])([H])C([H])([H])[*:1] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C243/00—Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
- C07C243/24—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids
- C07C243/26—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids with acylating carboxyl groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C243/34—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids with acylating carboxyl groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of a carbon skeleton further substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C259/00—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
- C07C259/12—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. N-hydroxyamidines
- C07C259/14—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. N-hydroxyamidines having carbon atoms of hydroxamidine groups bound to hydrogen atoms or to acyclic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/42—Unsaturated compounds containing hydroxy or O-metal groups
- C07C59/52—Unsaturated compounds containing hydroxy or O-metal groups a hydroxy or O-metal group being bound to a carbon atom of a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C65/00—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C65/01—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups
- C07C65/03—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups monocyclic and having all hydroxy or O-metal groups bound to the ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D233/22—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D233/24—Radicals substituted by nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US66425867A | 1967-08-30 | 1967-08-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1168361A true GB1168361A (en) | 1969-10-22 |
Family
ID=24665273
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB52098/67A Expired GB1168361A (en) | 1967-08-30 | 1967-11-15 | Hydroxyphenyl Substituted Cyclic and Acyclic Amidines and derivatives thereof |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US3579510A (cg-RX-API-DMAC7.html) |
| JP (1) | JPS4813108B1 (cg-RX-API-DMAC7.html) |
| BR (1) | BR6801003D0 (cg-RX-API-DMAC7.html) |
| DE (1) | DE1793050C3 (cg-RX-API-DMAC7.html) |
| DK (2) | DK123710B (cg-RX-API-DMAC7.html) |
| FR (2) | FR1584069A (cg-RX-API-DMAC7.html) |
| GB (1) | GB1168361A (cg-RX-API-DMAC7.html) |
| IL (1) | IL30383A (cg-RX-API-DMAC7.html) |
| NL (1) | NL162074C (cg-RX-API-DMAC7.html) |
| NO (1) | NO126440B (cg-RX-API-DMAC7.html) |
| SE (1) | SE349579B (cg-RX-API-DMAC7.html) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3930001A (en) * | 1971-11-30 | 1975-12-30 | Pfizer | 2-(Substituted)-5,6-dihydro-4H-1,4-thiazines used for the control of rice blast |
| US3890443A (en) * | 1973-09-17 | 1975-06-17 | Pfizer | 2-(Substituted) thiazolines for the control of rice blast |
| US4490388A (en) * | 1981-02-27 | 1984-12-25 | Torii & Co., Ltd. | Amidine compound and anticomplement agent comprising same |
| DE3211301A1 (de) * | 1982-03-26 | 1983-09-29 | Bayer Ag, 5090 Leverkusen | Cyclische amidine, verfahren zu ihrer herstellung und die verwendung cyclischer amidine als katalysatoren fuer die haertung von epoxidharzen |
| WO1995007100A1 (en) * | 1993-09-10 | 1995-03-16 | Petrovax L.L.C. | Compounds for the prevention and treatment of helminth infections |
-
1967
- 1967-08-30 US US664258A patent/US3579510A/en not_active Expired - Lifetime
- 1967-11-15 GB GB52098/67A patent/GB1168361A/en not_active Expired
-
1968
- 1968-07-17 IL IL30383A patent/IL30383A/xx unknown
- 1968-07-24 SE SE10100/68A patent/SE349579B/xx unknown
- 1968-07-24 NO NO2927/68A patent/NO126440B/no unknown
- 1968-07-26 NL NL6810601.A patent/NL162074C/xx not_active IP Right Cessation
- 1968-07-27 DE DE1793050A patent/DE1793050C3/de not_active Expired
- 1968-07-29 DK DK366168AA patent/DK123710B/da not_active IP Right Cessation
- 1968-07-29 BR BR201003/68A patent/BR6801003D0/pt unknown
- 1968-07-30 JP JP43053411A patent/JPS4813108B1/ja active Pending
- 1968-07-30 FR FR1584069D patent/FR1584069A/fr not_active Expired
- 1968-10-30 FR FR172006A patent/FR7991M/fr not_active Expired
-
1970
- 1970-02-20 DK DK85470AA patent/DK126785B/da unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BR6801003D0 (pt) | 1973-07-03 |
| NO126440B (cg-RX-API-DMAC7.html) | 1973-02-05 |
| DE1793050A1 (de) | 1971-12-16 |
| DE1793050C3 (de) | 1975-09-11 |
| SE349579B (cg-RX-API-DMAC7.html) | 1972-10-02 |
| FR1584069A (cg-RX-API-DMAC7.html) | 1969-12-12 |
| US3579510A (en) | 1971-05-18 |
| NL162074B (nl) | 1979-11-15 |
| NL162074C (nl) | 1980-04-15 |
| JPS4813108B1 (cg-RX-API-DMAC7.html) | 1973-04-25 |
| IL30383A0 (en) | 1968-09-26 |
| FR7991M (cg-RX-API-DMAC7.html) | 1970-06-08 |
| IL30383A (en) | 1973-02-28 |
| DE1793050B2 (de) | 1975-01-23 |
| NL6810601A (cg-RX-API-DMAC7.html) | 1969-03-04 |
| DK123710B (da) | 1972-07-24 |
| DK126785B (da) | 1973-08-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| PE20 | Patent expired after termination of 20 years |