FR2949464B1 - Derives de thiadiazoles et d'oxadiazoles, leur preparation et leur application en therapeutique - Google Patents
Derives de thiadiazoles et d'oxadiazoles, leur preparation et leur application en therapeutiqueInfo
- Publication number
- FR2949464B1 FR2949464B1 FR0904137A FR0904137A FR2949464B1 FR 2949464 B1 FR2949464 B1 FR 2949464B1 FR 0904137 A FR0904137 A FR 0904137A FR 0904137 A FR0904137 A FR 0904137A FR 2949464 B1 FR2949464 B1 FR 2949464B1
- Authority
- FR
- France
- Prior art keywords
- oxadiazoles
- thiadiazoles
- derivatives
- preparation
- therapeutic application
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
- C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
- C07D285/135—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
- C07D271/07—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Child & Adolescent Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (27)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0904137A FR2949464B1 (fr) | 2009-09-01 | 2009-09-01 | Derives de thiadiazoles et d'oxadiazoles, leur preparation et leur application en therapeutique |
TW099102288A TW201031645A (en) | 2009-01-28 | 2010-01-27 | Thiadiazole and oxadiazole derivatives, preparation thereof and therapeutic use thereof |
CA2750742A CA2750742A1 (fr) | 2009-01-28 | 2010-01-27 | Derives de thiadiazoles et d'oxadiazoles, leur preparation et leur application en therapeutique |
ARP100100186A AR075177A1 (es) | 2009-01-28 | 2010-01-27 | Derivados de tiadiazoles y oxadiazoles, metodo de preparacion, intermediarios de sintesis, composiciones farmaceuticas que los contienen y uso de los mismos en el tratamiento de trastornos metabolicos, tales como obesidad y diabetes, entre otros. |
NZ594244A NZ594244A (en) | 2009-01-28 | 2010-01-27 | Thiadiazole and oxadiazole derivatives, preparation thereof, and therapeutic use thereof |
CN2010800142290A CN102365273A (zh) | 2009-01-28 | 2010-01-27 | 噻二唑与*二唑衍生物及其制备与其治疗用途 |
PCT/FR2010/050124 WO2010086551A1 (fr) | 2009-01-28 | 2010-01-27 | Dérivés de thiadiazoles et d'oxadiazoles, leur préparation et leur application en thérapeutique |
US13/145,665 US8546391B2 (en) | 2009-01-28 | 2010-01-27 | Thiadiazole and oxadiazole derivatives, preparation thereof and therapeutic use thereof |
MA34128A MA33069B1 (fr) | 2009-01-28 | 2010-01-27 | Dérivés de thiadiazoles et d'oxadiazoles, leur préparation et leur application en thérapeutique |
PE2011001392A PE20120362A1 (es) | 2009-01-28 | 2010-01-27 | Derivados de tiadiazoles y oxadiazoles, su preparacion y su aplicacion en terapia |
JP2011546921A JP2012516312A (ja) | 2009-01-28 | 2010-01-27 | チアジアゾールおよびオキサジアゾール誘導体、これらの調製ならびにこれらの治療用途 |
KR1020117019841A KR20110112845A (ko) | 2009-01-28 | 2010-01-27 | 티아디아졸 및 옥사디아졸 유도체, 그의 제조, 및 그의 치료 용도 |
MX2011007991A MX2011007991A (es) | 2009-01-28 | 2010-01-27 | Derivados de tiadiazoles y oxadiazoles, su preparacion y su uso en terapeutica. |
AU2010209545A AU2010209545A1 (en) | 2009-01-28 | 2010-01-27 | Thiadiazole and oxadiazole derivatives, preparation thereof, and therapeutic use thereof |
BRPI1007414-7A BRPI1007414A2 (pt) | 2009-01-28 | 2010-01-27 | derivados de tiadiazóis e de oxadiazóis, o respectivo preparo e a respectiva aplicação em terapêutica |
EA201170983A EA201170983A1 (ru) | 2009-01-28 | 2010-01-27 | Производные тиадиазолов и оксадиазолов, их получение и их применение в терапии |
EP10707597.0A EP2391611B1 (fr) | 2009-01-28 | 2010-01-27 | Dérivés de thiadiazoles et d'oxadiazoles, leur préparation et leur application en thérapeutique |
UY0001032405A UY32405A (es) | 2009-01-28 | 2010-01-28 | Derivados de tiadiazoles y oxadiazoles, su preparacion y su aplicacion en terapia |
TN2011000353A TN2011000353A1 (fr) | 2009-01-28 | 2011-07-15 | Derives de thiadiazoles et d'oxadiazoles, leur preparation et leur application en therapeutique |
IL214260A IL214260A0 (en) | 2009-01-28 | 2011-07-24 | Thiadiazole and oxadiazole derivatives, preparation thereof, and therapeutic use thereof |
EC2011011224A ECSP11011224A (es) | 2009-01-28 | 2011-07-25 | Derivados de tiadiazoles y oxadiazoles, su preparaciòn y su aplicaciòn en terapia |
CR20110403A CR20110403A (es) | 2009-01-28 | 2011-07-26 | Derivados de tiadiazoles y oxadiazoles, su preparación y su aplicación en terapia |
NI201100149A NI201100149A (es) | 2009-01-28 | 2011-07-27 | Derivados de tiadiazoles y oxadiazoles, su preparación y su aplicación en terapia. |
ZA2011/05525A ZA201105525B (en) | 2009-01-28 | 2011-07-27 | Thiadiazole and oxadiazole derivatives,preparation thereof,and therapeutic use thereof |
CL2011001839A CL2011001839A1 (es) | 2009-01-28 | 2011-07-28 | Compuestos derivados de tiadiazoles y oxadiazoles, inhibidores de la biosintesis de trigliceridos; procedimiento de preparacion; compuestos intermediarios; composicion farmaceutica; y uso para el tratamiento y/o la prevencion de obesidad, dislipidemia, afecciones de alteracion de la glucosa en ayunas, diabetes de tipo 2, entre otras. |
DO2011000245A DOP2011000245A (es) | 2009-01-28 | 2011-07-28 | Derivados de tiadiazoles y oxadiazoles, su preparacion y su aplicacion en terapeutica |
CO11094698A CO6400221A2 (es) | 2009-01-28 | 2011-07-28 | Derivados de tidiazoles y oxadiazoles, su preparación y su aplicación en terapia |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0904137A FR2949464B1 (fr) | 2009-09-01 | 2009-09-01 | Derives de thiadiazoles et d'oxadiazoles, leur preparation et leur application en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2949464A1 FR2949464A1 (fr) | 2011-03-04 |
FR2949464B1 true FR2949464B1 (fr) | 2011-09-30 |
Family
ID=41821879
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR0904137A Expired - Fee Related FR2949464B1 (fr) | 2009-01-28 | 2009-09-01 | Derives de thiadiazoles et d'oxadiazoles, leur preparation et leur application en therapeutique |
Country Status (1)
Country | Link |
---|---|
FR (1) | FR2949464B1 (fr) |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2007236049A1 (en) * | 2006-04-07 | 2007-10-18 | High Point Pharmaceuticals, Llc | 11beta-hydroxysteroid dehydrogenase type 1 active compounds |
JP2011500563A (ja) * | 2007-10-10 | 2011-01-06 | メルク・シャープ・エンド・ドーム・コーポレイション | ジフェニル置換されたシクロアルカン |
-
2009
- 2009-09-01 FR FR0904137A patent/FR2949464B1/fr not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
FR2949464A1 (fr) | 2011-03-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PLFP | Fee payment |
Year of fee payment: 7 |
|
ST | Notification of lapse |
Effective date: 20170531 |