FR2937972B1 - Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique - Google Patents

Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique

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Publication number
FR2937972B1
FR2937972B1 FR0857496A FR0857496A FR2937972B1 FR 2937972 B1 FR2937972 B1 FR 2937972B1 FR 0857496 A FR0857496 A FR 0857496A FR 0857496 A FR0857496 A FR 0857496A FR 2937972 B1 FR2937972 B1 FR 2937972B1
Authority
FR
France
Prior art keywords
cosmetics
preparation
human medicine
oxoazetidine derivatives
oxoazetidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0857496A
Other languages
English (en)
Other versions
FR2937972A1 (fr
Inventor
Peter Claire Bouix
Itaru Suzuki
Nicolas Rodeville
Pascale Mauvais
Jean Claude Pascal
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Galderma Research and Development SNC
Original Assignee
Galderma Research and Development SNC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR0857496A priority Critical patent/FR2937972B1/fr
Application filed by Galderma Research and Development SNC filed Critical Galderma Research and Development SNC
Priority to US13/127,643 priority patent/US8871187B2/en
Priority to JP2011533761A priority patent/JP5798486B2/ja
Priority to BRPI0916069A priority patent/BRPI0916069C1/pt
Priority to RU2011122637/04A priority patent/RU2569886C2/ru
Priority to ARP090104265A priority patent/AR074275A1/es
Priority to RU2015141009A priority patent/RU2671189C1/ru
Priority to CN201410498368.5A priority patent/CN104387372B/zh
Priority to AU2009312818A priority patent/AU2009312818B2/en
Priority to CA2738785A priority patent/CA2738785C/fr
Priority to EP09744417.8A priority patent/EP2342194B1/fr
Priority to KR1020117012910A priority patent/KR101689042B1/ko
Priority to CN2009801446981A priority patent/CN102203081A/zh
Priority to MX2011004068A priority patent/MX2011004068A/es
Priority to PCT/EP2009/064646 priority patent/WO2010052253A1/fr
Publication of FR2937972A1 publication Critical patent/FR2937972A1/fr
Application granted granted Critical
Publication of FR2937972B1 publication Critical patent/FR2937972B1/fr
Priority to US14/497,600 priority patent/US9630949B2/en
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q17/00—Barrier preparations; Preparations brought into direct contact with the skin for affording protection against external influences, e.g. sunlight, X-rays or other harmful rays, corrosive materials, bacteria or insect stings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q17/00—Barrier preparations; Preparations brought into direct contact with the skin for affording protection against external influences, e.g. sunlight, X-rays or other harmful rays, corrosive materials, bacteria or insect stings
    • A61Q17/04—Topical preparations for affording protection against sunlight or other radiation; Topical sun tanning preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/004—Aftersun preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/007—Preparations for dry skin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/008—Preparations for oily skin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/02—Preparations for care of the skin for chemically bleaching or whitening the skin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/04—Preparations for care of the skin for chemically tanning the skin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/08—Anti-ageing preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q5/00—Preparations for care of the hair
    • A61Q5/10—Preparations for permanently dyeing the hair
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/74—Biological properties of particular ingredients
    • A61K2800/78—Enzyme modulators, e.g. Enzyme agonists
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
FR0857496A 2008-11-04 2008-11-04 Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique Expired - Fee Related FR2937972B1 (fr)

Priority Applications (16)

Application Number Priority Date Filing Date Title
FR0857496A FR2937972B1 (fr) 2008-11-04 2008-11-04 Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique
EP09744417.8A EP2342194B1 (fr) 2008-11-04 2009-11-04 Dérivés d'oxoazétidine, procédé pour la préparation de ceux-ci et utilisation de ceux-ci dans la médecine humaine et dans les cosmétiques
BRPI0916069A BRPI0916069C1 (pt) 2008-11-04 2009-11-04 composto, usos de um composto, composição farmacêutica, composição cosmética e usos cosméticos de uma composição
RU2011122637/04A RU2569886C2 (ru) 2008-11-04 2009-11-04 Производные оксоазетидина, способ их получения и их применения в медицине и косметологии
ARP090104265A AR074275A1 (es) 2008-11-04 2009-11-04 Derivados de oxoacetidina, procedimiento para su preparacion y su uso como moduladores de la melanocortina
RU2015141009A RU2671189C1 (ru) 2008-11-04 2009-11-04 Производные оксоазетидина, способ их получения и их применения в медицине и косметологии
CN201410498368.5A CN104387372B (zh) 2008-11-04 2009-11-04 氧代吖丁啶衍生物、其制备方法及其在人类医药和美容品中的用途
AU2009312818A AU2009312818B2 (en) 2008-11-04 2009-11-04 Oxoazetidine derivatives, process for the preparation thereof and use thereof in human medicine and in cosmetics
US13/127,643 US8871187B2 (en) 2008-11-04 2009-11-04 Oxoazetidine derivatives, process for the preparation thereof and use thereon in human medicine and in cosmetics
JP2011533761A JP5798486B2 (ja) 2008-11-04 2009-11-04 オキソアゼチジン誘導体、その調製方法、ならびにヒト医薬および化粧品におけるその使用
KR1020117012910A KR101689042B1 (ko) 2008-11-04 2009-11-04 옥소아제티딘 유도체, 이의 제조 방법 및 인간 약물 및 화장품에서의 이의 용도
CN2009801446981A CN102203081A (zh) 2008-11-04 2009-11-04 氧代吖丁啶衍生物、其制备方法及其在人类医药和美容品中的用途
MX2011004068A MX2011004068A (es) 2008-11-04 2009-11-04 Derivados de oxoazetidina, procesos para la preparacion de los mismos y usos de los mismos en medicina humana y en cosmeticos.
PCT/EP2009/064646 WO2010052253A1 (fr) 2008-11-04 2009-11-04 Dérivés d'oxoazétidine, procédé pour la préparation de ceux-ci et utilisation de ceux-ci dans la médecine humaine et dans les cosmétiques
CA2738785A CA2738785C (fr) 2008-11-04 2009-11-04 Derives d'oxoazetidine, procede pour la preparation de ceux-ci et utilisation de ceux-ci dans la medecine humaine et dans les cosmetiques
US14/497,600 US9630949B2 (en) 2008-11-04 2014-09-26 Oxoazetidine derivatives, process for the preparation thereof and use thereof in human medicine and in cosmetics

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FR0857496A FR2937972B1 (fr) 2008-11-04 2008-11-04 Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique

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AR (1) AR074275A1 (fr)
AU (1) AU2009312818B2 (fr)
BR (1) BRPI0916069C1 (fr)
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MX (1) MX2011004068A (fr)
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FR2969494B1 (fr) * 2010-12-22 2013-11-08 Expanscience Lab Extrait de parties aeriennes de gynandropsis gynandra ou cleome gynandra et compositions cosmetiques, dermatologiques le comprenant
FR2981933B1 (fr) * 2011-11-02 2013-11-15 Galderma Res & Dev Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique
FR2984167B1 (fr) 2011-12-16 2014-01-17 Galderma Res & Dev Association d'un agoniste des recepteurs des prostaglandines et d'un agoniste du recepteur mc1r pour le traitement et/ou la prevention de desordres de la pigmentation
EP2825187A1 (fr) 2012-03-15 2015-01-21 Galderma Research & Development Combinaison d'un agoniste du récepteur mc1r et d'uvb dans le traitement et/ou la prévention de troubles de la pigmentation
FR2992317B1 (fr) 2012-06-22 2016-05-13 Diverchim Procede de preparation de peptides chiraux
FR3027900B1 (fr) * 2014-11-05 2018-02-23 Centre National De La Recherche Scientifique Utilisation de derives halogenes de l'histidine a titre de sel d'electrolyte dans une cellule photovoltaique a colorants
CA2968836A1 (fr) 2016-06-13 2017-12-13 Gilead Sciences, Inc. Composes modulant fxr (nr1h4)
AU2018215619A1 (en) * 2017-02-01 2019-08-08 Clinuvel Pharmaceuticals Ltd Alpha-MSH analogues used in the treatment of xeroderma pigmentosum
PL3600309T3 (pl) 2017-03-28 2022-11-07 Gilead Sciences, Inc. Skojarzenia terapeutyczne do leczenia chorób wątroby
JP2022519906A (ja) 2019-02-19 2022-03-25 ギリアード サイエンシーズ， インコーポレイテッド Ｆｘｒアゴニストの固体形態
US20220096648A1 (en) 2020-09-14 2022-03-31 Regeneron Pharmaceuticals, Inc. Antibody-drug conjugates comprising glp1 peptidomimetics and uses thereof
US20230330254A1 (en) 2022-03-11 2023-10-19 Regeneron Pharmaceuticals, Inc. Anti-glp1r antibody-tethered drug conjugates comprising glp1 peptidomimetics and uses thereof

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CA2738785C (fr) 2017-05-16
CN104387372B (zh) 2018-06-26
JP2012507491A (ja) 2012-03-29
KR101689042B1 (ko) 2016-12-22
US9630949B2 (en) 2017-04-25
CN102203081A (zh) 2011-09-28
JP5798486B2 (ja) 2015-10-21
BRPI0916069B8 (pt) 2019-12-17
AU2009312818B2 (en) 2014-11-06
EP2342194B1 (fr) 2018-08-08
US8871187B2 (en) 2014-10-28
WO2010052253A1 (fr) 2010-05-14
AU2009312818A1 (en) 2010-05-14
RU2011122637A (ru) 2012-12-20
RU2671189C1 (ru) 2018-10-30
CN104387372A (zh) 2015-03-04
BRPI0916069A2 (pt) 2015-11-10
MX2011004068A (es) 2011-05-31
EP2342194A1 (fr) 2011-07-13
BRPI0916069B1 (pt) 2019-11-05
CA2738785A1 (fr) 2010-05-14
RU2569886C2 (ru) 2015-12-10
US20150045559A1 (en) 2015-02-12
FR2937972A1 (fr) 2010-05-07
KR20110088555A (ko) 2011-08-03
AR074275A1 (es) 2011-01-05
US20110274638A1 (en) 2011-11-10
BRPI0916069C1 (pt) 2021-05-25

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