FR2745569B1 - Composes apparentes a la famille des amidiniums, compositions pharmaceutiques les contenant et leurs applications - Google Patents

Composes apparentes a la famille des amidiniums, compositions pharmaceutiques les contenant et leurs applications

Info

Publication number
FR2745569B1
FR2745569B1 FR9602604A FR9602604A FR2745569B1 FR 2745569 B1 FR2745569 B1 FR 2745569B1 FR 9602604 A FR9602604 A FR 9602604A FR 9602604 A FR9602604 A FR 9602604A FR 2745569 B1 FR2745569 B1 FR 2745569B1
Authority
FR
France
Prior art keywords
amidinium
family
applications
pharmaceutical compositions
compositions containing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
FR9602604A
Other languages
English (en)
Other versions
FR2745569A1 (fr
Inventor
Jean Marie Lehn
Jean Pierre Vigneron
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Centre National de la Recherche Scientifique CNRS
Original Assignee
Centre National de la Recherche Scientifique CNRS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR9602604A priority Critical patent/FR2745569B1/fr
Application filed by Centre National de la Recherche Scientifique CNRS filed Critical Centre National de la Recherche Scientifique CNRS
Priority to AU19304/97A priority patent/AU723998B2/en
Priority to HU9902465A priority patent/HU228072B1/hu
Priority to KR1019980706784A priority patent/KR19990087372A/ko
Priority to DK97907154T priority patent/DK0888379T3/da
Priority to SI9730098T priority patent/SI0888379T1/xx
Priority to CA002248186A priority patent/CA2248186C/fr
Priority to BRPI9707889A priority patent/BRPI9707889B8/pt
Priority to JP53067797A priority patent/JP4271260B2/ja
Priority to AT97907154T priority patent/ATE198599T1/de
Priority to IL12592697A priority patent/IL125926A/en
Priority to PT97907154T priority patent/PT888379E/pt
Priority to US09/125,825 priority patent/US6143729A/en
Priority to DE69703878T priority patent/DE69703878T2/de
Priority to ES97907154T priority patent/ES2154453T3/es
Priority to CZ19982772A priority patent/CZ295225B6/cs
Priority to SK1182-98A priority patent/SK283575B6/sk
Priority to PCT/FR1997/000364 priority patent/WO1997031935A1/fr
Priority to EP97907154A priority patent/EP0888379B1/fr
Publication of FR2745569A1 publication Critical patent/FR2745569A1/fr
Publication of FR2745569B1 publication Critical patent/FR2745569B1/fr
Application granted granted Critical
Priority to NO19983691A priority patent/NO311806B1/no
Priority to US09/706,619 priority patent/US6316422B1/en
Priority to GR20000402653T priority patent/GR3035205T3/el
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0055Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of at least three carbon atoms which may or may not be branched, e.g. cholane or cholestane derivatives, optionally cyclised, e.g. 17-beta-phenyl or 17-beta-furyl derivatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Liposomes
    • A61K9/1271Non-conventional liposomes, e.g. PEGylated liposomes, liposomes coated with polymers
    • A61K9/1272Non-conventional liposomes, e.g. PEGylated liposomes, liposomes coated with polymers with substantial amounts of non-phosphatidyl, i.e. non-acylglycerophosphate, surfactants as bilayer-forming substances, e.g. cationic lipids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
FR9602604A 1996-03-01 1996-03-01 Composes apparentes a la famille des amidiniums, compositions pharmaceutiques les contenant et leurs applications Expired - Lifetime FR2745569B1 (fr)

Priority Applications (22)

Application Number Priority Date Filing Date Title
FR9602604A FR2745569B1 (fr) 1996-03-01 1996-03-01 Composes apparentes a la famille des amidiniums, compositions pharmaceutiques les contenant et leurs applications
ES97907154T ES2154453T3 (es) 1996-03-01 1997-02-28 Compuestos pertenecientes a la familia de los amidiniums, composiciones farmaceuticas que les contienen y sus aplicaciones.
HU9902465A HU228072B1 (en) 1996-03-01 1997-02-28 New cholesterol amidinium derivatives, pharmaceutical compositions containing same, and uses thereof
CZ19982772A CZ295225B6 (cs) 1996-03-01 1997-02-28 Amidiniový derivát a farmaceutický prostředek tento derivát obsahující
SI9730098T SI0888379T1 (en) 1996-03-01 1997-02-28 Compounds related to the amidinium family, pharmaceutical compositions containing same, and uses thereof
CA002248186A CA2248186C (fr) 1996-03-01 1997-02-28 Composes apparentes a la famille des amidiniums, compositions pharmaceutiques les contenant et leurs applications
BRPI9707889A BRPI9707889B8 (pt) 1996-03-01 1997-02-28 composto e seus sais, composição farmacêutica, utilização do composto.
JP53067797A JP4271260B2 (ja) 1996-03-01 1997-02-28 アミジニウムファミリーに属する化合物、該化合物を含有する医薬組成物及びその使用
AT97907154T ATE198599T1 (de) 1996-03-01 1997-02-28 Guanidinium-verbindungen, pharmazeutische präparate davon und ihre verwendungen
IL12592697A IL125926A (en) 1996-03-01 1997-02-28 Compounds related to the amidinium family, pharmaceutical preparations containing them and their uses
PT97907154T PT888379E (pt) 1996-03-01 1997-02-28 Compostos analogos a familia dos amidinios composicoes farmaceuticas que os contem e suas aplicacoes
US09/125,825 US6143729A (en) 1996-03-01 1997-02-28 Compounds related to the amidinium family, pharmaceutical compositions containing same, and uses thereof
AU19304/97A AU723998B2 (en) 1996-03-01 1997-02-28 Compounds related to the amidinium family, pharmaceutical compositions containing same, and uses thereof
KR1019980706784A KR19990087372A (ko) 1996-03-01 1997-02-28 아미디늄류 관련 화합물, 이를 함유한 약학조성물, 및 이의용도
DK97907154T DK0888379T3 (da) 1996-03-01 1997-02-28 Forbindelser tilhørende amidinium-familien, farmaceutiske præparater indeholdende disse forbindelser og anvendelsen deraf
SK1182-98A SK283575B6 (sk) 1996-03-01 1997-02-28 Zlúčeniny amidíniového typu, farmaceutické prostriedky, ktoré ich obsahujú, a ich použitie
PCT/FR1997/000364 WO1997031935A1 (fr) 1996-03-01 1997-02-28 Composes apparentes a la famille des amidiniums, compositions pharmaceutiques les contenant et leurs applications
EP97907154A EP0888379B1 (fr) 1996-03-01 1997-02-28 Composes apparentes a la famille des amidiniums, compositions pharmaceutiques les contenant et leurs applications
DE69703878T DE69703878T2 (de) 1996-03-01 1997-02-28 Guanidinium-verbindungen, pharmazeutische präparate davon und ihre verwendungen
NO19983691A NO311806B1 (no) 1996-03-01 1998-08-12 Forbindelser tilhörende amidiniumfamilien, farmasöytiske preparater inneholdende disse samt anvendelse derav
US09/706,619 US6316422B1 (en) 1996-03-01 2000-11-06 Compounds related to the amidinium family, pharmaceutical compositions containing same, and uses thereof
GR20000402653T GR3035205T3 (en) 1996-03-01 2001-01-11 Compounds related to the amidinium family, pharmaceutical compositions containing same, and uses thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9602604A FR2745569B1 (fr) 1996-03-01 1996-03-01 Composes apparentes a la famille des amidiniums, compositions pharmaceutiques les contenant et leurs applications

Publications (2)

Publication Number Publication Date
FR2745569A1 FR2745569A1 (fr) 1997-09-05
FR2745569B1 true FR2745569B1 (fr) 1998-05-07

Family

ID=9489760

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9602604A Expired - Lifetime FR2745569B1 (fr) 1996-03-01 1996-03-01 Composes apparentes a la famille des amidiniums, compositions pharmaceutiques les contenant et leurs applications

Country Status (1)

Country Link
FR (1) FR2745569B1 (fr)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5283185A (en) * 1991-08-28 1994-02-01 University Of Tennessee Research Corporation Method for delivering nucleic acids into cells
JPH09508099A (ja) * 1993-12-20 1997-08-19 ユニヴェルシテ リブル ドゥ ブリュッセル 細胞中に少なくとも一つの分子を導入できる化合物
US5777153A (en) * 1994-07-08 1998-07-07 Gilead Sciences, Inc. Cationic lipids

Also Published As

Publication number Publication date
FR2745569A1 (fr) 1997-09-05

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