FR2361880A1 - Nouvelles 4-amino piperidines, leurs procedes d'obtention et les compositions pharmaceutiques en renfermant - Google Patents
Nouvelles 4-amino piperidines, leurs procedes d'obtention et les compositions pharmaceutiques en renfermantInfo
- Publication number
- FR2361880A1 FR2361880A1 FR7612671A FR7612671A FR2361880A1 FR 2361880 A1 FR2361880 A1 FR 2361880A1 FR 7612671 A FR7612671 A FR 7612671A FR 7612671 A FR7612671 A FR 7612671A FR 2361880 A1 FR2361880 A1 FR 2361880A1
- Authority
- FR
- France
- Prior art keywords
- new
- processes
- pharmaceutical compositions
- compositions containing
- amino piperidines
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 150000003053 piperidines Chemical class 0.000 title 1
- BCIIMDOZSUCSEN-UHFFFAOYSA-N piperidin-4-amine Chemical class NC1CCNCC1 BCIIMDOZSUCSEN-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C321/00—Thiols, sulfides, hydropolysulfides or polysulfides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/34—Sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La présente invention a pour objet de nouvelles 4-amino pipéridines et plus particulierement les 1-aryl alcoyl 4-amino pipéridines répondant à la formule générale :
Priority Applications (14)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7612671A FR2361880A1 (fr) | 1976-04-29 | 1976-04-29 | Nouvelles 4-amino piperidines, leurs procedes d'obtention et les compositions pharmaceutiques en renfermant |
BE177109A BE854072A (fr) | 1976-04-29 | 1977-04-28 | Nouvelles aminopiperidines, leur preparation et leur emploi comme medicament |
JP4983377A JPS52133989A (en) | 1976-04-29 | 1977-04-28 | Novel aminopiperidines and method of their preparation and medical composition thereof |
IL51966A IL51966A (en) | 1976-04-29 | 1977-04-28 | 1-(phenyl(or thienyl)amino(or thio)alkyl)-4-(n-alkanoyl-n-phenyl)amino piperidine derivatives,their preparation and pharmalceutical compositions containing them |
AU24648/77A AU508575B2 (en) | 1976-04-29 | 1977-04-28 | Aminopiperidines |
NL7704760A NL7704760A (nl) | 1976-04-29 | 1977-04-29 | Werkwijze voor de bereiding van 4-aminopiperi- dinen, werkwijze voor de bereiding van een ge- neesmiddel met antihypertensieve werking en een dergelijk geneesmiddel. |
AT306177A AT361924B (de) | 1976-04-29 | 1977-04-29 | Verfahren zur herstellung von neuen arylalkyl- piperidinen und von deren salzen |
DE2719211A DE2719211C3 (de) | 1976-04-29 | 1977-04-29 | 1-(2-Phenylamino-äthyl)-4-(N-phenyl-N-propionylamino)-piperidine, Verfahren zu ihrer Herstellung und sie enthaltende Arzneimittel |
ES458307A ES458307A1 (es) | 1976-04-29 | 1977-04-29 | Un procedimiento de preparacion de nuevas 4-amino-piperidi- nas sustituidas en el nitrogeno del ciclo piperidico por unacadena aril-alcoilica o sus sales. |
GB18027/77A GB1544191A (en) | 1976-04-29 | 1977-04-29 | Acylaminopiperidines processes for their preparation and pharmaceutical compositions containing them |
CH540977A CH620679A5 (fr) | 1976-04-29 | 1977-04-29 | |
JP5869378A JPS549282A (en) | 1976-04-29 | 1978-05-17 | Novel aminopiperidines*its preparation*and medical compositions |
US05/948,536 US4246267A (en) | 1976-04-29 | 1978-10-04 | Aminopiperidines, their production and the pharmaceutical compositions incorporating them |
AT686079A AT361926B (de) | 1976-04-29 | 1979-10-22 | Verfahren zur herstellung von neuen arylthio- alkylpiperidinen und von deren salzen |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7612671A FR2361880A1 (fr) | 1976-04-29 | 1976-04-29 | Nouvelles 4-amino piperidines, leurs procedes d'obtention et les compositions pharmaceutiques en renfermant |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2361880A1 true FR2361880A1 (fr) | 1978-03-17 |
FR2361880B1 FR2361880B1 (fr) | 1978-12-15 |
Family
ID=9172434
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7612671A Granted FR2361880A1 (fr) | 1976-04-29 | 1976-04-29 | Nouvelles 4-amino piperidines, leurs procedes d'obtention et les compositions pharmaceutiques en renfermant |
Country Status (12)
Country | Link |
---|---|
US (1) | US4246267A (fr) |
JP (2) | JPS52133989A (fr) |
AT (1) | AT361924B (fr) |
AU (1) | AU508575B2 (fr) |
BE (1) | BE854072A (fr) |
CH (1) | CH620679A5 (fr) |
DE (1) | DE2719211C3 (fr) |
ES (1) | ES458307A1 (fr) |
FR (1) | FR2361880A1 (fr) |
GB (1) | GB1544191A (fr) |
IL (1) | IL51966A (fr) |
NL (1) | NL7704760A (fr) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4584303A (en) * | 1984-04-09 | 1986-04-22 | The Boc Group, Inc. | N-aryl-N-(4-piperidinyl)amides and pharmaceutical compositions and method employing such compounds |
GR1000662B (el) * | 1988-07-01 | 1992-09-25 | Janssen Pharmaceutica Nv | Μεθοδος παρασκευης cis-ν-(3-μεθοξυ-4-πιπεριδινυλο)βενζαμιδιων. |
US5106983A (en) * | 1990-04-30 | 1992-04-21 | The United States Of America As Represented By The Secretary Of The Army | Process of making carfentanil and related analgesics |
FR2676054B1 (fr) * | 1991-05-03 | 1993-09-03 | Sanofi Elf | Nouveaux composes n-alkylenepiperidino et leurs enantiomeres, procede pour leur preparation et compositions pharmaceutiques les contenant. |
US5466691A (en) * | 1991-08-09 | 1995-11-14 | Yoshitomi Pharmaceutical Industries, Ltd. | Thiophene compound |
SE9902987D0 (sv) * | 1999-08-24 | 1999-08-24 | Astra Pharma Prod | Novel compounds |
GB0011838D0 (en) * | 2000-05-17 | 2000-07-05 | Astrazeneca Ab | Chemical compounds |
GB0104050D0 (en) | 2001-02-19 | 2001-04-04 | Astrazeneca Ab | Chemical compounds |
GB0107228D0 (en) | 2001-03-22 | 2001-05-16 | Astrazeneca Ab | Chemical compounds |
SE0103818D0 (sv) * | 2001-11-15 | 2001-11-15 | Astrazeneca Ab | Chemical compounds |
SE0301369D0 (sv) | 2003-05-09 | 2003-05-09 | Astrazeneca Ab | Chemical compounds |
JP2008502651A (ja) * | 2004-06-18 | 2008-01-31 | ノイロサーチ アクティーゼルスカブ | モノアミン神経伝達物質再取込み阻害剤としての、新規アルキル置換ピペリジン誘導体及びその使用 |
CN113214139B (zh) * | 2020-02-03 | 2022-03-04 | 江苏谛奇医药科技有限公司 | 哌啶酰胺类衍生物及其制备方法、其药物组合物、其单晶培养方法及其应用 |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3218327A (en) * | 1963-10-02 | 1965-11-16 | Parke Davis & Co | alpha-naphthylamine alkyl piperidine compounds |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2846437A (en) * | 1955-09-12 | 1958-08-05 | Sterling Drug Inc | Lower alkyl 4-phenyl-1-(substituted-alkyl) piperidine-4-carboxylates and preparationthereof |
US3479346A (en) * | 1961-08-08 | 1969-11-18 | Sterling Drug Inc | N-acyl-n- (and n,n-bis-) ((1-piperidyl)-lower-alkyl)amines |
US3869463A (en) * | 1973-01-17 | 1975-03-04 | Wyeth John & Brother Ltd | N-phenyl derivatives of alkanoylamido piperidines |
-
1976
- 1976-04-29 FR FR7612671A patent/FR2361880A1/fr active Granted
-
1977
- 1977-04-28 BE BE177109A patent/BE854072A/fr unknown
- 1977-04-28 IL IL51966A patent/IL51966A/xx unknown
- 1977-04-28 AU AU24648/77A patent/AU508575B2/en not_active Expired
- 1977-04-28 JP JP4983377A patent/JPS52133989A/ja active Pending
- 1977-04-29 NL NL7704760A patent/NL7704760A/xx not_active Application Discontinuation
- 1977-04-29 DE DE2719211A patent/DE2719211C3/de not_active Expired
- 1977-04-29 CH CH540977A patent/CH620679A5/fr not_active IP Right Cessation
- 1977-04-29 ES ES458307A patent/ES458307A1/es not_active Expired
- 1977-04-29 GB GB18027/77A patent/GB1544191A/en not_active Expired
- 1977-04-29 AT AT306177A patent/AT361924B/de not_active IP Right Cessation
-
1978
- 1978-05-17 JP JP5869378A patent/JPS549282A/ja active Pending
- 1978-10-04 US US05/948,536 patent/US4246267A/en not_active Expired - Lifetime
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3218327A (en) * | 1963-10-02 | 1965-11-16 | Parke Davis & Co | alpha-naphthylamine alkyl piperidine compounds |
Also Published As
Publication number | Publication date |
---|---|
IL51966A (en) | 1981-01-30 |
AU2464877A (en) | 1978-11-02 |
CH620679A5 (fr) | 1980-12-15 |
FR2361880B1 (fr) | 1978-12-15 |
GB1544191A (en) | 1979-04-11 |
US4246267A (en) | 1981-01-20 |
AU508575B2 (en) | 1980-03-27 |
BE854072A (fr) | 1977-10-28 |
ATA306177A (de) | 1980-09-15 |
IL51966A0 (en) | 1977-06-30 |
DE2719211B2 (de) | 1980-10-09 |
JPS549282A (en) | 1979-01-24 |
JPS52133989A (en) | 1977-11-09 |
NL7704760A (nl) | 1977-11-01 |
DE2719211A1 (de) | 1977-11-03 |
ES458307A1 (es) | 1978-02-16 |
AT361924B (de) | 1981-04-10 |
DE2719211C3 (de) | 1982-01-07 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |