FR2388795A1 - Nouveaux n-(1-(3-benzoylpropyl)-4-piperidyl)-sulfamides, procedes pour leur preparation et medicaments les renfermant - Google Patents
Nouveaux n-(1-(3-benzoylpropyl)-4-piperidyl)-sulfamides, procedes pour leur preparation et medicaments les renfermantInfo
- Publication number
- FR2388795A1 FR2388795A1 FR7812366A FR7812366A FR2388795A1 FR 2388795 A1 FR2388795 A1 FR 2388795A1 FR 7812366 A FR7812366 A FR 7812366A FR 7812366 A FR7812366 A FR 7812366A FR 2388795 A1 FR2388795 A1 FR 2388795A1
- Authority
- FR
- France
- Prior art keywords
- benzoylpropyl
- sulfamides
- piperidyl
- preparation
- new
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
L'invention a pour objet de nouveaux N-Ø1-(3-benzoylpropyl)-4-pipéridylõ-sulfamides. Ces composés répondent à la formule :
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19772718405 DE2718405A1 (de) | 1977-04-26 | 1977-04-26 | Neue n- eckige klammer auf 1-(3-benzoylpropyl)-4-piperidyl eckige klammer zu -sulfonsaeureamide und verfahren zu deren herstellung |
Publications (1)
Publication Number | Publication Date |
---|---|
FR2388795A1 true FR2388795A1 (fr) | 1978-11-24 |
Family
ID=6007245
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7812366A Withdrawn FR2388795A1 (fr) | 1977-04-26 | 1978-04-26 | Nouveaux n-(1-(3-benzoylpropyl)-4-piperidyl)-sulfamides, procedes pour leur preparation et medicaments les renfermant |
Country Status (23)
Country | Link |
---|---|
US (1) | US4145427A (fr) |
JP (1) | JPS53132579A (fr) |
AT (1) | AT364823B (fr) |
AU (1) | AU519705B2 (fr) |
BE (1) | BE866351A (fr) |
CA (1) | CA1097648A (fr) |
DE (1) | DE2718405A1 (fr) |
DK (1) | DK179278A (fr) |
ES (2) | ES469108A1 (fr) |
FI (1) | FI781177A (fr) |
FR (1) | FR2388795A1 (fr) |
GB (1) | GB1563989A (fr) |
GR (1) | GR64514B (fr) |
IL (1) | IL54574A (fr) |
IT (1) | IT1104811B (fr) |
LU (1) | LU79515A1 (fr) |
NL (1) | NL7804388A (fr) |
NO (1) | NO781450L (fr) |
NZ (1) | NZ187060A (fr) |
PH (1) | PH15717A (fr) |
PT (1) | PT67949B (fr) |
SE (1) | SE7804743L (fr) |
ZA (1) | ZA782340B (fr) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4246268A (en) * | 1979-02-09 | 1981-01-20 | Richardson-Merrell Inc. | Neuroleptic-4-(naphthylmethyl)piperidine derivatives |
NZ193654A (en) | 1979-05-16 | 1984-08-24 | Wuelfing Johann A | Naphthalene sulphonamido-alkyl-piperidines,pyrrolidines or piperazines and pharmaceutical compositions |
IE49998B1 (en) * | 1979-08-06 | 1986-01-22 | Merrell Dow Pharma | 4-(naphthalenyloxy)piperidine derivatives |
US4443462A (en) * | 1979-08-06 | 1984-04-17 | Merrell Dow Pharmaceuticals Inc. | Antipsychotic 4-(naphthalenyloxy)piperidine derivatives |
US5210090A (en) * | 1989-09-05 | 1993-05-11 | G. D. Searle & Co. | Substituted N-benzylpiperidine amides and cardiac regulatory compositions thereof |
WO2002022579A2 (fr) * | 2000-09-11 | 2002-03-21 | Sepracor, Inc. | Heterocycles sulfonamides antipsychotiques et leurs methodes d'utilisation |
EP1594840B1 (fr) * | 2003-02-17 | 2006-09-27 | F. Hoffmann-La Roche Ag | Dérivés de piperidine-benzenesulfonamide |
TW200630337A (en) | 2004-10-14 | 2006-09-01 | Euro Celtique Sa | Piperidinyl compounds and the use thereof |
US8247442B2 (en) * | 2006-03-29 | 2012-08-21 | Purdue Pharma L.P. | Benzenesulfonamide compounds and their use |
US8791264B2 (en) * | 2006-04-13 | 2014-07-29 | Purdue Pharma L.P. | Benzenesulfonamide compounds and their use as blockers of calcium channels |
US8937181B2 (en) * | 2006-04-13 | 2015-01-20 | Purdue Pharma L.P. | Benzenesulfonamide compounds and the use thereof |
CA2651732C (fr) * | 2006-05-18 | 2014-10-14 | Mannkind Corporation | Inhibiteurs de kinases intracellulaires |
WO2008124118A1 (fr) * | 2007-04-09 | 2008-10-16 | Purdue Pharma L.P. | Composés benzènesulfonylés et leur utilisation |
ES2601856T3 (es) | 2007-06-08 | 2017-02-16 | Mannkind Corporation | Inhibidores de la IRE-1A |
WO2009040659A2 (fr) * | 2007-09-28 | 2009-04-02 | Purdue Pharma L.P. | Composés benzènesulfonamides et leurs utilisations |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1482099A (en) * | 1974-12-11 | 1977-08-03 | Wyeth John & Brother Ltd | Sulphonamido derivatives |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB948071A (en) * | 1959-05-01 | 1964-01-29 | May & Baker Ltd | New heterocyclic compounds |
US3932636A (en) * | 1972-08-12 | 1976-01-13 | Pfizer Inc. | 2 And 3-substituted-4-(heterocyclic-amino-sulfonyl)benzene sulfonamides as cerebral vasodilators |
US3932649A (en) * | 1972-08-12 | 1976-01-13 | Pfizer Inc. | 2 And 3-substituted-4-(heterocyclic-amino-sulfonyl)benzene sulfonamides as cerebral vasodilators |
US3932647A (en) * | 1973-08-09 | 1976-01-13 | Pfizer Inc. | Cyclic N-substituted derivatives of 1,4-benzene disulphonamide |
-
1977
- 1977-04-26 DE DE19772718405 patent/DE2718405A1/de not_active Withdrawn
-
1978
- 1978-04-13 PH PH21001A patent/PH15717A/en unknown
- 1978-04-14 US US05/896,575 patent/US4145427A/en not_active Expired - Lifetime
- 1978-04-14 AT AT0261578A patent/AT364823B/de not_active IP Right Cessation
- 1978-04-18 FI FI781177A patent/FI781177A/fi not_active Application Discontinuation
- 1978-04-20 GR GR56039A patent/GR64514B/el unknown
- 1978-04-24 LU LU79515A patent/LU79515A1/de unknown
- 1978-04-24 IT IT49045/78A patent/IT1104811B/it active
- 1978-04-24 JP JP4866778A patent/JPS53132579A/ja active Pending
- 1978-04-24 NZ NZ187060A patent/NZ187060A/xx unknown
- 1978-04-24 PT PT67949A patent/PT67949B/pt unknown
- 1978-04-25 DK DK179278A patent/DK179278A/da not_active Application Discontinuation
- 1978-04-25 NL NL7804388A patent/NL7804388A/xx not_active Application Discontinuation
- 1978-04-25 SE SE7804743A patent/SE7804743L/xx unknown
- 1978-04-25 BE BE187089A patent/BE866351A/fr unknown
- 1978-04-25 ES ES469108A patent/ES469108A1/es not_active Expired
- 1978-04-25 ZA ZA00782340A patent/ZA782340B/xx unknown
- 1978-04-25 GB GB16308/78A patent/GB1563989A/en not_active Expired
- 1978-04-25 NO NO781450A patent/NO781450L/no unknown
- 1978-04-25 CA CA301,885A patent/CA1097648A/fr not_active Expired
- 1978-04-25 IL IL54574A patent/IL54574A/xx unknown
- 1978-04-26 AU AU35453/78A patent/AU519705B2/en not_active Expired
- 1978-04-26 FR FR7812366A patent/FR2388795A1/fr not_active Withdrawn
- 1978-08-08 ES ES472448A patent/ES472448A1/es not_active Expired
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1482099A (en) * | 1974-12-11 | 1977-08-03 | Wyeth John & Brother Ltd | Sulphonamido derivatives |
Also Published As
Publication number | Publication date |
---|---|
SE7804743L (sv) | 1978-10-27 |
IT7849045A0 (it) | 1978-04-24 |
ES469108A1 (es) | 1978-11-16 |
NO781450L (no) | 1978-10-27 |
LU79515A1 (de) | 1979-05-25 |
AU519705B2 (en) | 1981-12-17 |
BE866351A (fr) | 1978-10-25 |
IL54574A0 (en) | 1978-07-31 |
PT67949B (de) | 1980-06-16 |
GR64514B (en) | 1980-04-09 |
AT364823B (de) | 1981-11-25 |
ES472448A1 (es) | 1979-05-01 |
PH15717A (en) | 1983-03-18 |
IL54574A (en) | 1981-09-13 |
DE2718405A1 (de) | 1978-11-02 |
NZ187060A (en) | 1980-11-28 |
AU3545378A (en) | 1979-11-01 |
FI781177A (fi) | 1978-10-27 |
PT67949A (de) | 1978-05-01 |
US4145427A (en) | 1979-03-20 |
ATA261578A (de) | 1981-04-15 |
GB1563989A (en) | 1980-04-02 |
ZA782340B (en) | 1979-12-27 |
NL7804388A (nl) | 1978-10-30 |
CA1097648A (fr) | 1981-03-17 |
DK179278A (da) | 1978-10-27 |
JPS53132579A (en) | 1978-11-18 |
IT1104811B (it) | 1985-10-28 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
FR2372810A1 (fr) | Nouvelles aminoalcoylimidazolidinones, procedes pour leur preparation et leur utilisation en tant que medicaments | |
FR2394534A1 (fr) | Nouveaux 1-aryloxy-2-hydroxy-3-alcoyleneaminopropanes, procedes pour leur preparation et medicaments les renfermant | |
FR2400512A1 (fr) | Nouveaux nitro-imidazoles, leur preparation et leur application en tant que medicaments | |
FR2383922A1 (fr) | Nouvelles 4-acylamino-phenyl-ethanolamines, procede pour leur preparation et leur utilisation en tant que medicaments | |
FR2390420A1 (fr) | Nouveaux derives cyclopeptidiques, leur preparation et leur application comme medicaments | |
FR2377418A1 (fr) | Nouveaux derives steroides 4,9-dieniques 11b-substitues, leur procede de preparation et leur application comme medicaments | |
FR2388795A1 (fr) | Nouveaux n-(1-(3-benzoylpropyl)-4-piperidyl)-sulfamides, procedes pour leur preparation et medicaments les renfermant | |
FR2397403A1 (fr) | Nouveaux derives de 1-acyl 2-cyano-aziridine, procede pour leur preparation et compositions pharmaceutiques contenant ces composes | |
FR2444681A1 (fr) | Nouvelles 1,4-dihydropyridines, leur preparation et leur application comme medicaments | |
FR2391215A1 (fr) | Nouvelles imidazoazines et imidazodiazines, leur preparation et leur application en tant que medicaments | |
FR2392991A1 (fr) | Nouvelles 5,11-dihydro-6h-pyrido(2,3-b) (1,4) benzodiazepin-6-ones substituees en position 11, procedes pour leur preparation et medicaments renfermant ces composes | |
FR2361398A1 (fr) | Nouvelles 6-aryl-4h-s-triazolo-(3,4c)-thieno(2,3e)-1,4-diazepines, leur preparation et leur utilisation en tant que medicaments | |
FR2377419A1 (fr) | Nouveaux derives steroides 11b-substitues 1,3,5 (10) trieniques, leur procede de preparation et leur application comme medicament | |
FR2392993A1 (fr) | Nouvelles 5,11-dihydro-6h-pyrido(2,3-b) (1,4) benzadiazepin-6-ones, procedes pour leur preparation et medicaments renfermant ces composes | |
FR2423485A1 (fr) | Nouvelles 1,3-diaryl-2-imino-imidazolidines et 1,3-diaryl-2-imino-hexahydro-pyrimidines substituees, procedes de preparation de ces composes et medicaments les contenant | |
FR2378014A1 (fr) | Nouveaux derives aminoalcoxyphenyles, leur preparation et leur utilisation en tant que medicaments | |
FR2379533A1 (fr) | Tetrazolylcarbamoylquinoleines utilisables comme medicaments et leur preparation | |
FR2355007A1 (fr) | (3-alcoyle inferieur-amino-2-r, 10 propoxy pyridines substituees, leur preparation et leur application en tant que medicaments | |
FR2361371A1 (fr) | Nouvelles 2-phenylamino imidazolines-(2) substituees, leurs sels d'addition avec des acides, les medicaments les renfermant et procedes pour leur preparation | |
FR2417503A1 (fr) | Nouvelles 2-phenylimino-imidazolidines substituees, leurs sels d'addition avec des acides, medicaments les renfermant et procedes pour leur preparation | |
FR2370745A1 (fr) | Nouveaux derives de la morphanthridine, leur preparation et leur application comme medicaments | |
FR2398069A1 (fr) | Nouvelles imidazo-isoquinoleine-diones, procedes pour leur preparation et leur utilisation en tant que medicaments | |
FR2383944A1 (fr) | Derives de bis-benzimidazolyle substitues, leur procede de preparation et leur application en therapeutique | |
FR2400017A1 (fr) | Nouveaux acides 2-pyridyl- et 2-pyrimidylaminobenzoiques, leur preparation et leur utilisation en tant que medicaments | |
FR2379542A1 (fr) | Nouveaux 1,1-dioxydes de 2,5-dihydro-1,2-thiazino (5,6-b) indole-3-carboxamides, procedes pour leur preparation et medicaments les renfermant |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |