FR2208651A1 - Piperazinyl carbonyloxy-dithiino pyrrols as tranquillisers - anticonvulsants and spasmolytics from aryloxycarbonates of dithiinopyrrols and piperazines - Google Patents
Piperazinyl carbonyloxy-dithiino pyrrols as tranquillisers - anticonvulsants and spasmolytics from aryloxycarbonates of dithiinopyrrols and piperazinesInfo
- Publication number
- FR2208651A1 FR2208651A1 FR7243054A FR7243054A FR2208651A1 FR 2208651 A1 FR2208651 A1 FR 2208651A1 FR 7243054 A FR7243054 A FR 7243054A FR 7243054 A FR7243054 A FR 7243054A FR 2208651 A1 FR2208651 A1 FR 2208651A1
- Authority
- FR
- France
- Prior art keywords
- dithiinopyrrols
- aryloxycarbonates
- tranquillisers
- pyrrols
- spasmolytics
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- XBRAPGITUVXBKT-UHFFFAOYSA-N 5H-dithiino[4,3-b]pyrrol-3-yl piperazine-1-carboxylate Chemical class N1(CCNCC1)C(=O)OC1=CC2=C(C=CN2)SS1 XBRAPGITUVXBKT-UHFFFAOYSA-N 0.000 title 1
- 229940125681 anticonvulsant agent Drugs 0.000 title 1
- 239000001961 anticonvulsive agent Substances 0.000 title 1
- 150000004885 piperazines Chemical class 0.000 title 1
- 230000002048 spasmolytic effect Effects 0.000 title 1
- WEVYAHXRMPXWCK-UHFFFAOYSA-N Acetonitrile Chemical compound CC#N WEVYAHXRMPXWCK-UHFFFAOYSA-N 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 239000002253 acid Substances 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000004593 naphthyridinyl group Chemical group N1=C(C=CC2=CC=CN=C12)* 0.000 abstract 1
- 125000002098 pyridazinyl group Chemical group 0.000 abstract 1
- 125000004076 pyridyl group Chemical group 0.000 abstract 1
- 125000005493 quinolyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/08—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (39)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7243054A FR2208651A1 (en) | 1972-12-04 | 1972-12-04 | Piperazinyl carbonyloxy-dithiino pyrrols as tranquillisers - anticonvulsants and spasmolytics from aryloxycarbonates of dithiinopyrrols and piperazines |
| AR251345A AR207555A1 (es) | 1972-12-04 | 1973-01-01 | Procedimiento para preparar aril-6-piperazinocarboniloxi-5 oxo-7 tetrahidro-2,3,6,7 ditiino(1,4)(2,3-c)pirroles |
| NL7316162.A NL164037C (nl) | 1972-12-04 | 1973-11-26 | Werkwijze ter bereiding van 1,4-dithiino- -2,3-cpyrrool-derivaten en van farmaceutische preparaten die deze derivaten bevatten. |
| OA55074A OA04515A (fr) | 1972-12-04 | 1973-11-29 | Nouveaux dérivés du dithiino[1,4] [2,3-c] pyrrole et leur procédé de préparation. |
| IE2178/73A IE38561B1 (en) | 1972-12-04 | 1973-12-03 | 1,4-dithiino 2,3-cpyrrole derivatives |
| MX684773U MX4845E (es) | 1972-12-04 | 1973-12-03 | Procedimiento mejorado para la preparacion de los derivados de (1,4) (2,3-c) ditiino pirrol |
| CH1691273A CH590867A5 (enExample) | 1972-12-04 | 1973-12-03 | |
| IL43734A IL43734A (en) | 1972-12-04 | 1973-12-03 | 5-(piperazin-1-yl)carbonyloxy-6-substituted 7-oxo-2,3,6,7-tetrahydro-1,4-dithiino(2,3-c)pyrrole derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same |
| LU68924A LU68924A1 (enExample) | 1972-12-04 | 1973-12-03 | |
| PH15282A PH10402A (en) | 1972-12-04 | 1973-12-03 | 1,4-dithino(2,3-c)pyrrole derivatives and pharmaceutical compositions containing the same |
| DK652573A DK145781C (da) | 1972-12-04 | 1973-12-03 | Analogifremgangsmaade til fremstilling af ditiino(1,4)(2,3-c)pyrrolderivater |
| HURO762A HU166918B (enExample) | 1972-12-04 | 1973-12-03 | |
| SU7301974547A SU576942A3 (ru) | 1972-12-04 | 1973-12-03 | Способ получени производных дитиино (1,4) (2,3-с) пиррола или их солей |
| CH1350576A CH589092A5 (enExample) | 1972-12-04 | 1973-12-03 | |
| ZA739139A ZA739139B (en) | 1972-12-04 | 1973-12-03 | 1,4-dithiino(2,3-c)pyrrole derivatives |
| US05/421,060 US3948917A (en) | 1972-12-04 | 1973-12-03 | 1,4-Dithiino(2,3-c)pyrrole derivatives |
| CA187,271A CA989841A (fr) | 1972-12-04 | 1973-12-03 | Derives du dithiino (1,4)(2,3-c) pyrrole, leur preparation et les compositions qui les contiennent |
| SE7316302A SE398351B (sv) | 1972-12-04 | 1973-12-03 | Forfarande for framstellning av ditino-(1,4)-(2,3-c)pyrrol-piperazinderivat |
| BE138458A BE808152A (fr) | 1972-12-04 | 1973-12-03 | Nouveaux derives du dithiino (1,4) (2,3-c) pyrrole, leur preparation et les compositions qui les contiennent |
| NO734609A NO138850C (no) | 1972-12-04 | 1973-12-03 | Analogifremgangsmaater for fremstilling av nye terapeutisk aktive derivater av ditiino(1,4)(2,3-c)pyrrol |
| JP48135675A JPS52959B2 (enExample) | 1972-12-04 | 1973-12-03 | |
| DD175050A DD108301A5 (enExample) | 1972-12-04 | 1973-12-03 | |
| ES421130A ES421130A1 (es) | 1972-12-04 | 1973-12-04 | Procedimiento para preparar derivados de ditiino (1,4) (2, 3-c) pirrol. |
| FI3721/73A FI54712C (fi) | 1972-12-04 | 1973-12-04 | Foerfarande foer framstaellning av terapeutiskt aktiva 5-((4-metylpiperazin-1-yl)karbonyloxi)-7-oxo-2,3,6,7-tetrahydroditiino (1,4)2,3-c)pyrroler |
| YU3124/73A YU40969B (en) | 1972-12-04 | 1973-12-04 | Process for obtaining new dithiino-(1,4)(2,3-c)-pyrrole derivtives |
| CS738348A CS209410B2 (en) | 1972-12-04 | 1973-12-04 | Method of making the new derivatives of the 1,4 dithiino(2,3-c)-pyrrole |
| CY959A CY959A (en) | 1972-12-04 | 1973-12-04 | 1,4-dithino(2,3-c)pyrrole derivatives |
| DE19732360362 DE2360362C3 (de) | 1972-12-04 | 1973-12-04 | 5-Hydroxy -7-oxo-2,3,6,7tetrahydro -1,4-dlthiino eckige Klammer auf 2,3-c eckige Klammer zu pyrrolderWate, Hire Herstellung und diese enthaltende pharmazeutische Zusammensetzungen |
| GB5604373A GB1397060A (en) | 1972-12-04 | 1973-12-04 | 1,4-dighiino 2,3-c pyrrole derivatives |
| AT1015273A AT330789B (de) | 1972-12-04 | 1973-12-04 | Verfahren zur herstellung von neuen (1,4) ditihiino (2,3-c) pyrrolderivaten und von deren saureadditionssalzen |
| AR255085A AR205094A1 (es) | 1972-12-04 | 1974-01-01 | Procedimiento para preparar derivados de ((piperazinil-1) carboniloxi)-5 oxo-7 tetrahidro-2,3,6,7 ditiino (1,4) (2,3-c) pirrol de formula general |
| ES423586A ES423586A1 (es) | 1972-12-04 | 1974-02-23 | Procedimiento para preparar derivados de ditiino (1,4) (2,3-c) pirrol. |
| SU2112820A SU548209A3 (ru) | 1972-12-04 | 1975-03-17 | Способ получени производных дитиино (1,4) (2,3-с) пиррола или их солей |
| US05/589,871 US3966931A (en) | 1972-12-04 | 1975-06-24 | 1,4-Dithino[2,3-c]pyrrole compositions |
| AT591675A AT330790B (de) | 1972-12-04 | 1975-07-30 | Verfahren zur herstellung von neuen (1,4) dithiino (2,3-c) pyrrolderivaten und von deren saureadditionssalzen |
| CS763589A CS209411B2 (cs) | 1972-12-04 | 1976-05-28 | Způsob výroby nových derivátů l,4-dithiino[2,3-c]pyrrolu |
| KE2864A KE2864A (en) | 1972-12-04 | 1978-08-03 | 1, 4-dithiino (2,3,-c) pyrrole derivatives |
| HK502/78A HK50278A (en) | 1972-12-04 | 1978-09-07 | 1,4-dithiino(2,3-c)pyrrole derivatives |
| YU02382/81A YU238281A (en) | 1972-12-04 | 1981-10-02 | Process for obtaining new derivatives of dithiino(1,4)(2,3-c)pyrroles |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7243054A FR2208651A1 (en) | 1972-12-04 | 1972-12-04 | Piperazinyl carbonyloxy-dithiino pyrrols as tranquillisers - anticonvulsants and spasmolytics from aryloxycarbonates of dithiinopyrrols and piperazines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2208651A1 true FR2208651A1 (en) | 1974-06-28 |
| FR2208651B1 FR2208651B1 (enExample) | 1975-11-28 |
Family
ID=9108153
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7243054A Granted FR2208651A1 (en) | 1972-12-04 | 1972-12-04 | Piperazinyl carbonyloxy-dithiino pyrrols as tranquillisers - anticonvulsants and spasmolytics from aryloxycarbonates of dithiinopyrrols and piperazines |
Country Status (3)
| Country | Link |
|---|---|
| BE (1) | BE808152A (enExample) |
| FR (1) | FR2208651A1 (enExample) |
| ZA (1) | ZA739139B (enExample) |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2141634A1 (de) * | 1970-08-19 | 1972-02-24 | Rhone-Poulenc S.A., Paris | Neue Isoindolinderivate, ihre Herstellung und Zusammensetzungen, die diese enthalten |
| FR2117740A1 (enExample) * | 1970-12-14 | 1972-07-28 | Rhone Poulenc Sa | |
| DE2221939A1 (de) * | 1971-05-04 | 1972-11-23 | Rhone Poulenc Sa | Neue Derivate des Isoindolins,Verfahren zu deren Herstellung und diese enthaltende medizinische Zusammensetzungen |
-
1972
- 1972-12-04 FR FR7243054A patent/FR2208651A1/fr active Granted
-
1973
- 1973-12-03 ZA ZA739139A patent/ZA739139B/xx unknown
- 1973-12-03 BE BE138458A patent/BE808152A/xx not_active IP Right Cessation
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2141634A1 (de) * | 1970-08-19 | 1972-02-24 | Rhone-Poulenc S.A., Paris | Neue Isoindolinderivate, ihre Herstellung und Zusammensetzungen, die diese enthalten |
| FR2117740A1 (enExample) * | 1970-12-14 | 1972-07-28 | Rhone Poulenc Sa | |
| DE2221939A1 (de) * | 1971-05-04 | 1972-11-23 | Rhone Poulenc Sa | Neue Derivate des Isoindolins,Verfahren zu deren Herstellung und diese enthaltende medizinische Zusammensetzungen |
Also Published As
| Publication number | Publication date |
|---|---|
| FR2208651B1 (enExample) | 1975-11-28 |
| ZA739139B (en) | 1974-11-27 |
| BE808152A (fr) | 1974-06-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| CD | Change of name or company name | ||
| TP | Transmission of property |