FI961199A0 - Substituerade tiazolo(3,2-alfa)azepinderivat - Google Patents
Substituerade tiazolo(3,2-alfa)azepinderivatInfo
- Publication number
- FI961199A0 FI961199A0 FI961199A FI961199A FI961199A0 FI 961199 A0 FI961199 A0 FI 961199A0 FI 961199 A FI961199 A FI 961199A FI 961199 A FI961199 A FI 961199A FI 961199 A0 FI961199 A0 FI 961199A0
- Authority
- FI
- Finland
- Prior art keywords
- group
- hydrogen atom
- lower alkyl
- alpha
- substituted
- Prior art date
Links
- 150000001538 azepines Chemical class 0.000 title 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 6
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000004414 alkyl thio group Chemical group 0.000 abstract 2
- 125000006239 protecting group Chemical group 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 102000004270 Peptidyl-Dipeptidase A Human genes 0.000 abstract 1
- 108090000882 Peptidyl-Dipeptidase A Proteins 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 230000007935 neutral effect Effects 0.000 abstract 1
- 125000003396 thiol group Chemical group [H]S* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Immunology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP6165481A JPH0827156A (ja) | 1994-07-18 | 1994-07-18 | アミノ酸誘導体の製造方法 |
| JP16548194 | 1994-07-18 | ||
| JP19918094A JP3444666B2 (ja) | 1994-08-24 | 1994-08-24 | （２ｓ， ３ｓ）−３− メチル−２− チオペンタン酸誘導体の製造方法 |
| JP19918094 | 1994-08-24 | ||
| JP30646894 | 1994-12-09 | ||
| JP6306468A JPH08165293A (ja) | 1994-12-09 | 1994-12-09 | 置換チアゾロ［３，２−ａ］アゼピン誘導体 |
| JP9501139 | 1995-06-07 | ||
| PCT/JP1995/001139 WO1996002549A1 (fr) | 1994-07-18 | 1995-06-07 | DERIVE DE THIAZOLO[3,2-α]AZEPINE A SUBSTITUTION |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI961199A0 true FI961199A0 (sv) | 1996-03-14 |
| FI961199A FI961199A (sv) | 1996-05-13 |
| FI110001B FI110001B (sv) | 2002-11-15 |
Family
ID=27322514
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI961199A FI110001B (sv) | 1994-07-18 | 1996-03-14 | 6-substituerade 5-oxo-oktahydrotiazolo[3,2-a]azepin-3-karboxylsyraderivat och förfarande för framställning av de samma samt deras användning |
| FI20011154A FI113656B (sv) | 1994-07-18 | 2001-06-01 | 6-amino-5-oxo-oktahydrotiazolo[3,2-a]azepin-3-karboxylsyraderivat användabara som mellanprodukt |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI20011154A FI113656B (sv) | 1994-07-18 | 2001-06-01 | 6-amino-5-oxo-oktahydrotiazolo[3,2-a]azepin-3-karboxylsyraderivat användabara som mellanprodukt |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US5789403A (sv) |
| EP (1) | EP0719779B1 (sv) |
| KR (1) | KR100284247B1 (sv) |
| CN (2) | CN1053908C (sv) |
| AT (1) | ATE254622T1 (sv) |
| AU (1) | AU694233B2 (sv) |
| CA (1) | CA2171334C (sv) |
| DE (1) | DE69532155T2 (sv) |
| DK (1) | DK0719779T3 (sv) |
| ES (1) | ES2210292T3 (sv) |
| FI (2) | FI110001B (sv) |
| HU (1) | HU225916B1 (sv) |
| MX (1) | MX9601017A (sv) |
| NO (1) | NO308077B1 (sv) |
| NZ (1) | NZ287557A (sv) |
| PT (1) | PT719779E (sv) |
| WO (1) | WO1996002549A1 (sv) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5650408A (en) * | 1995-06-07 | 1997-07-22 | Karanewsky; Donald S. | Thiazolo benzazepine containing dual action inhibitors |
| WO1998034636A1 (fr) * | 1997-02-05 | 1998-08-13 | Suntory Limited | Compositions medicinales pour traiter les cardiopathies induites par l'hypertrophie cardiaque |
| US9823092B2 (en) | 2014-10-31 | 2017-11-21 | Allegro Microsystems, Llc | Magnetic field sensor providing a movement detector |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA821904B (en) * | 1981-03-23 | 1983-01-26 | Merck & Co Inc | Bicyclic lactams as anthihypertensives |
| US4415496A (en) * | 1981-03-23 | 1983-11-15 | Merck & Co., Inc. | Bicyclic lactams |
| US4617301A (en) * | 1983-06-22 | 1986-10-14 | Merck & Co., Inc. | Sulfoxide and sulfone derivatives of bicyclic lactams as antihypertensives |
| JPS6056790A (ja) * | 1983-09-03 | 1985-04-02 | 山陽科学株式会社 | 荷役用マット |
| RU2124503C1 (ru) * | 1992-05-18 | 1999-01-10 | И.Р.Сквибб энд Санз, Инк. | Гетероциклические азотсодержащие производные карбоновой кислоты, способ их получения и фармацевтическая композиция |
| JP3420766B2 (ja) * | 1992-10-30 | 2003-06-30 | メレルダウファーマス−ティカルズ インコーポレイテッド | エンケファリナーゼ及びａｃｅの阻害剤として有用な新規なメルカプトアセチルアミド二環式ラクタム誘導体類 |
| US5650408A (en) * | 1995-06-07 | 1997-07-22 | Karanewsky; Donald S. | Thiazolo benzazepine containing dual action inhibitors |
-
1995
- 1995-06-07 US US08/612,864 patent/US5789403A/en not_active Expired - Lifetime
- 1995-06-07 DE DE69532155T patent/DE69532155T2/de not_active Expired - Fee Related
- 1995-06-07 WO PCT/JP1995/001139 patent/WO1996002549A1/ja active IP Right Grant
- 1995-06-07 AT AT95921127T patent/ATE254622T1/de not_active IP Right Cessation
- 1995-06-07 CA CA002171334A patent/CA2171334C/en not_active Expired - Fee Related
- 1995-06-07 NZ NZ287557A patent/NZ287557A/en not_active IP Right Cessation
- 1995-06-07 KR KR1019960701358A patent/KR100284247B1/ko not_active IP Right Cessation
- 1995-06-07 EP EP95921127A patent/EP0719779B1/en not_active Expired - Lifetime
- 1995-06-07 PT PT95921127T patent/PT719779E/pt unknown
- 1995-06-07 HU HU9600679A patent/HU225916B1/hu not_active IP Right Cessation
- 1995-06-07 CN CN95190779A patent/CN1053908C/zh not_active Expired - Fee Related
- 1995-06-07 MX MX9601017A patent/MX9601017A/es not_active IP Right Cessation
- 1995-06-07 DK DK95921127T patent/DK0719779T3/da active
- 1995-06-07 AU AU26301/95A patent/AU694233B2/en not_active Ceased
- 1995-06-07 ES ES95921127T patent/ES2210292T3/es not_active Expired - Lifetime
-
1996
- 1996-03-14 FI FI961199A patent/FI110001B/sv active
- 1996-03-14 NO NO19961051A patent/NO308077B1/no not_active IP Right Cessation
-
1998
- 1998-05-27 US US09/085,729 patent/US6051705A/en not_active Expired - Fee Related
-
1999
- 1999-10-28 CN CNB991236092A patent/CN1170832C/zh not_active Expired - Fee Related
-
2001
- 2001-06-01 FI FI20011154A patent/FI113656B/sv not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| NZ287557A (en) | 1997-04-24 |
| CA2171334C (en) | 2008-10-21 |
| US5789403A (en) | 1998-08-04 |
| FI20011154A (sv) | 2001-06-01 |
| CN1170832C (zh) | 2004-10-13 |
| CN1262275A (zh) | 2000-08-09 |
| ES2210292T3 (es) | 2004-07-01 |
| KR960704898A (ko) | 1996-10-09 |
| PT719779E (pt) | 2004-04-30 |
| DK0719779T3 (da) | 2004-03-22 |
| EP0719779A1 (en) | 1996-07-03 |
| US6051705A (en) | 2000-04-18 |
| ATE254622T1 (de) | 2003-12-15 |
| EP0719779B1 (en) | 2003-11-19 |
| NO961051D0 (no) | 1996-03-14 |
| CN1053908C (zh) | 2000-06-28 |
| FI113656B (sv) | 2004-05-31 |
| HU225916B1 (en) | 2007-12-28 |
| NO961051L (no) | 1996-05-10 |
| AU694233B2 (en) | 1998-07-16 |
| FI961199A (sv) | 1996-05-13 |
| NO308077B1 (no) | 2000-07-17 |
| HUT76477A (en) | 1997-09-29 |
| DE69532155D1 (de) | 2003-12-24 |
| FI110001B (sv) | 2002-11-15 |
| WO1996002549A1 (fr) | 1996-02-01 |
| DE69532155T2 (de) | 2004-08-19 |
| HU9600679D0 (en) | 1996-05-28 |
| CN1134152A (zh) | 1996-10-23 |
| AU2630195A (en) | 1996-02-16 |
| CA2171334A1 (en) | 1996-02-01 |
| KR100284247B1 (ko) | 2001-10-24 |
| MX9601017A (es) | 1997-10-31 |
| EP0719779A4 (en) | 1996-12-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC | Transfer of assignment of patent |
Owner name: EISAI R&D MANAGEMENT CO., LTD. Free format text: EISAI R&D MANAGEMENT CO., LTD. |