FI960795A - Uudet tiofeeniyhdisteet, menetelmä niiden valmistamiseksi ja niitä sisältävät farmaseuttiset koostumukset - Google Patents

Uudet tiofeeniyhdisteet, menetelmä niiden valmistamiseksi ja niitä sisältävät farmaseuttiset koostumukset Download PDF

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Publication number
FI960795A
FI960795A FI960795A FI960795A FI960795A FI 960795 A FI960795 A FI 960795A FI 960795 A FI960795 A FI 960795A FI 960795 A FI960795 A FI 960795A FI 960795 A FI960795 A FI 960795A
Authority
FI
Finland
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
thiophene compounds
alkyl
Prior art date
Application number
FI960795A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI960795A0 (fi
Inventor
Michel Wierzbicki
Frederic Sauveur
Jacqueline Bonnet
Charles Tordjman
Original Assignee
Adir
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adir filed Critical Adir
Publication of FI960795A0 publication Critical patent/FI960795A0/fi
Publication of FI960795A publication Critical patent/FI960795A/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/24Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
FI960795A 1995-02-23 1996-02-21 Uudet tiofeeniyhdisteet, menetelmä niiden valmistamiseksi ja niitä sisältävät farmaseuttiset koostumukset FI960795A (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9502061A FR2730996B1 (fr) 1995-02-23 1995-02-23 Nouveaux composes du thiophene, leur procede de preparation et les compositions pharmaceutiques les renfermant

Publications (2)

Publication Number Publication Date
FI960795A0 FI960795A0 (fi) 1996-02-21
FI960795A true FI960795A (fi) 1996-08-24

Family

ID=9476411

Family Applications (1)

Application Number Title Priority Date Filing Date
FI960795A FI960795A (fi) 1995-02-23 1996-02-21 Uudet tiofeeniyhdisteet, menetelmä niiden valmistamiseksi ja niitä sisältävät farmaseuttiset koostumukset

Country Status (18)

Country Link
US (2) US5705525A (ja)
EP (1) EP0728755B1 (ja)
JP (1) JPH08253470A (ja)
CN (1) CN1058965C (ja)
AT (1) ATE200488T1 (ja)
AU (1) AU697832B2 (ja)
CA (1) CA2170097C (ja)
CY (1) CY2262B1 (ja)
DE (1) DE69612416T2 (ja)
DK (1) DK0728755T3 (ja)
ES (1) ES2158255T3 (ja)
FI (1) FI960795A (ja)
FR (1) FR2730996B1 (ja)
GR (1) GR3036192T3 (ja)
NO (1) NO314997B1 (ja)
NZ (1) NZ286045A (ja)
PT (1) PT728755E (ja)
ZA (1) ZA961472B (ja)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2305414A1 (en) * 1997-10-03 1999-04-15 Merck Frosst Canada & Co. Aryl thiophene derivatives as pde iv inhibitors
AUPR283801A0 (en) * 2001-02-01 2001-03-01 Australian National University, The Chemical compounds and methods
FR2860792B1 (fr) * 2003-10-10 2006-02-24 Sanofi Synthelabo Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutique
CN112724127B (zh) * 2019-10-28 2023-02-17 中国科学院上海药物研究所 五元杂环氧代羧酸类化合物及其医药用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0055471A1 (en) * 1980-12-29 1982-07-07 E.I. Du Pont De Nemours And Company Antiinflammatory 4,5-diaryl-alpha,alpha-bis(polyhalomethyl)-2-thiophenemethanamines
GB8525716D0 (en) * 1985-10-18 1985-11-20 Roussel Lab Ltd Chemical compounds
FR2655043B1 (fr) * 1989-11-24 1992-02-07 Adir Nouveaux derives du thiophene, leur procede de preparation et les compositions pharmaceutiques les renfermant.
US5571810A (en) * 1990-06-11 1996-11-05 Fujisawa Pharmaceutical Co., Ltd. Thiophene derivatives
GB9012936D0 (en) * 1990-06-11 1990-08-01 Fujisawa Pharmaceutical Co Thiophene derivatives,processes for preparation thereof and pharmaceutical composition comprising the same

Also Published As

Publication number Publication date
JPH08253470A (ja) 1996-10-01
CN1058965C (zh) 2000-11-29
GR3036192T3 (en) 2001-10-31
FR2730996B1 (fr) 1997-06-20
DE69612416D1 (de) 2001-05-17
NO314997B1 (no) 2003-06-23
CA2170097A1 (fr) 1996-08-24
DE69612416T2 (de) 2001-11-22
FI960795A0 (fi) 1996-02-21
NO960706L (no) 1996-08-26
NZ286045A (en) 1996-10-28
ZA961472B (en) 1996-08-28
CN1142496A (zh) 1997-02-12
FR2730996A1 (fr) 1996-08-30
EP0728755B1 (fr) 2001-04-11
ES2158255T3 (es) 2001-09-01
US5705525A (en) 1998-01-06
DK0728755T3 (da) 2001-07-30
PT728755E (pt) 2001-09-28
CY2262B1 (en) 2003-07-04
ATE200488T1 (de) 2001-04-15
USRE37078E1 (en) 2001-02-27
CA2170097C (fr) 2002-02-26
EP0728755A1 (fr) 1996-08-28
AU697832B2 (en) 1998-10-15
NO960706D0 (no) 1996-02-22
AU4567596A (en) 1996-08-29

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Legal Events

Date Code Title Description
MA Patent expired