ES2147271T3 - Eteres de oximas triciclicas, sus procedimentos de preparacion y las composiciones farmaceuticas que los contienen. - Google Patents
Eteres de oximas triciclicas, sus procedimentos de preparacion y las composiciones farmaceuticas que los contienen.Info
- Publication number
- ES2147271T3 ES2147271T3 ES95402865T ES95402865T ES2147271T3 ES 2147271 T3 ES2147271 T3 ES 2147271T3 ES 95402865 T ES95402865 T ES 95402865T ES 95402865 T ES95402865 T ES 95402865T ES 2147271 T3 ES2147271 T3 ES 2147271T3
- Authority
- ES
- Spain
- Prior art keywords
- triciclicas
- oximas
- eteres
- contain
- pharmaceutical compositions
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Otolaryngology (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Indole Compounds (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A LOS COMPUESTOS DE FORMULA (I): EN LA QUE A, X, Y, R{SUB,1}, R{SUB,2} Y R{SUB,3} SON TALES COMO SE DEFINEN EN LA DESCRIPCION. MEDICAMENTOS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9415431A FR2728571B1 (fr) | 1994-12-22 | 1994-12-22 | Nouveaux ethers d'oximes tricycliques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2147271T3 true ES2147271T3 (es) | 2000-09-01 |
Family
ID=9470078
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES95402865T Expired - Lifetime ES2147271T3 (es) | 1994-12-22 | 1995-12-19 | Eteres de oximas triciclicas, sus procedimentos de preparacion y las composiciones farmaceuticas que los contienen. |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US5627203A (es) |
| EP (1) | EP0718299B1 (es) |
| JP (1) | JP2937837B2 (es) |
| CN (2) | CN1066449C (es) |
| AT (1) | ATE191483T1 (es) |
| AU (1) | AU693615B2 (es) |
| CA (1) | CA2165618C (es) |
| DE (1) | DE69516100T2 (es) |
| DK (1) | DK0718299T3 (es) |
| ES (1) | ES2147271T3 (es) |
| FI (1) | FI956136L (es) |
| FR (1) | FR2728571B1 (es) |
| GR (1) | GR3033507T3 (es) |
| NO (1) | NO955215L (es) |
| NZ (1) | NZ280734A (es) |
| PT (1) | PT718299E (es) |
| ZA (1) | ZA9510901B (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2781482B1 (fr) * | 1998-07-27 | 2001-08-31 | Adir | Nouveaux derives de 8h-thieno-[2,3-b]pyrrolizine-8-one, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| EP1567491A4 (en) * | 2002-11-21 | 2007-09-19 | New York Blood Ct Inc | COMPOUNDS FOR INHIBITING HIV INFECTION BY BLOCKING HIV INJECTION |
| DE102008015032A1 (de) * | 2008-03-17 | 2009-09-24 | Aicuris Gmbh & Co. Kg | Substituierte Pyrazolamide und ihre Verwendung |
| DE102008015033A1 (de) * | 2008-03-17 | 2009-09-24 | Aicuris Gmbh & Co. Kg | Substituierte (Pyrazolyl-carbonyl)imidazolidinone und ihre Verwendung |
| DE102008062863A1 (de) | 2008-12-17 | 2010-06-24 | Aicuris Gmbh & Co. Kg | Substituierte (Thiophenyl-carbonyl)imidazolidinone und ihre Verwendung |
| DE102008062878A1 (de) | 2008-12-17 | 2010-06-24 | Aicuris Gmbh & Co. Kg | Substituierte Furancarboxamide und ihre Verwendung |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE371193B (es) * | 1972-03-24 | 1974-11-11 | Kabi Ab | |
| US4308399A (en) * | 1977-08-30 | 1981-12-29 | Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. | O-(3-Amino-2-hydroxy-propyl)-amidoxime derivatives, process for the preparation thereof and pharmaceutical compositions containing same |
| US4134894A (en) * | 1978-05-04 | 1979-01-16 | Warner-Lambert Company | Pyrrolo[1,2-a]indole compounds |
| HU180739B (en) * | 1979-07-03 | 1983-04-29 | Egyt Gyogyszervegyeszeti Gyar | Process for producing basic oxime-ethers |
| US5128364A (en) * | 1991-03-28 | 1992-07-07 | Merck Frosst Canada, Inc. | Pyrrolo[1,2-a]indole hydroxylamine derivatives as inhibitors of leukotriene biosynthesis |
-
1994
- 1994-12-22 FR FR9415431A patent/FR2728571B1/fr not_active Expired - Fee Related
-
1995
- 1995-12-19 ES ES95402865T patent/ES2147271T3/es not_active Expired - Lifetime
- 1995-12-19 CA CA002165618A patent/CA2165618C/fr not_active Expired - Fee Related
- 1995-12-19 EP EP95402865A patent/EP0718299B1/fr not_active Expired - Lifetime
- 1995-12-19 DK DK95402865T patent/DK0718299T3/da active
- 1995-12-19 DE DE69516100T patent/DE69516100T2/de not_active Expired - Fee Related
- 1995-12-19 PT PT95402865T patent/PT718299E/pt unknown
- 1995-12-19 AT AT95402865T patent/ATE191483T1/de not_active IP Right Cessation
- 1995-12-20 AU AU40593/95A patent/AU693615B2/en not_active Ceased
- 1995-12-20 FI FI956136A patent/FI956136L/fi unknown
- 1995-12-21 NZ NZ280734A patent/NZ280734A/en unknown
- 1995-12-21 US US08/576,678 patent/US5627203A/en not_active Expired - Fee Related
- 1995-12-21 JP JP7333347A patent/JP2937837B2/ja not_active Expired - Lifetime
- 1995-12-21 ZA ZA9510901A patent/ZA9510901B/xx unknown
- 1995-12-21 NO NO955215A patent/NO955215L/no not_active Application Discontinuation
- 1995-12-22 CN CN95120144A patent/CN1066449C/zh not_active Expired - Fee Related
-
1999
- 1999-12-03 CN CN99120993A patent/CN1261073A/zh active Pending
-
2000
- 2000-05-25 GR GR20000401198T patent/GR3033507T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| NO955215L (no) | 1996-06-24 |
| ZA9510901B (en) | 1996-06-24 |
| NZ280734A (en) | 1997-09-22 |
| ATE191483T1 (de) | 2000-04-15 |
| CN1261073A (zh) | 2000-07-26 |
| FR2728571A1 (fr) | 1996-06-28 |
| CA2165618A1 (fr) | 1996-06-23 |
| FI956136A7 (fi) | 1996-06-23 |
| CA2165618C (fr) | 2001-04-10 |
| CN1066449C (zh) | 2001-05-30 |
| GR3033507T3 (en) | 2000-09-29 |
| US5627203A (en) | 1997-05-06 |
| EP0718299A1 (fr) | 1996-06-26 |
| DK0718299T3 (da) | 2000-09-04 |
| CN1131155A (zh) | 1996-09-18 |
| NO955215D0 (no) | 1995-12-21 |
| DE69516100T2 (de) | 2000-12-14 |
| AU693615B2 (en) | 1998-07-02 |
| FI956136A0 (fi) | 1995-12-20 |
| AU4059395A (en) | 1996-06-27 |
| DE69516100D1 (de) | 2000-05-11 |
| JP2937837B2 (ja) | 1999-08-23 |
| EP0718299B1 (fr) | 2000-04-05 |
| FI956136L (fi) | 1996-06-23 |
| JPH08231554A (ja) | 1996-09-10 |
| FR2728571B1 (fr) | 1997-01-31 |
| PT718299E (pt) | 2000-07-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
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