NO955215L - Nye tricykliske oximetere, fremgangsmåter ved deres fremstilling og farmasöytiske sammensetninger inneholdende dem - Google Patents
Nye tricykliske oximetere, fremgangsmåter ved deres fremstilling og farmasöytiske sammensetninger inneholdende demInfo
- Publication number
- NO955215L NO955215L NO955215A NO955215A NO955215L NO 955215 L NO955215 L NO 955215L NO 955215 A NO955215 A NO 955215A NO 955215 A NO955215 A NO 955215A NO 955215 L NO955215 L NO 955215L
- Authority
- NO
- Norway
- Prior art keywords
- substd
- opt
- alkyl
- phenyl
- cycloalkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Otolaryngology (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Indole Compounds (AREA)
Abstract
Forbindelser med formel (I) hvor R, er H, alkyl, alkenyl, cykloalkyl, cykloalkylalkyl, hydroksy, alkoksy, fenyl, fenylalkyl, fenoksy og fenylalkoksy, eller R, sammen med R, og kjeden -CH-(CH2)y-N(R3)- som bærer dem, danner et N- holdig ringsystem med fra 5 til 8 ringelementer; R2 og R3 er uavhengig H, alkyl, alkenyl, cykloalkyl, indanyl, cykloalkylalkyl, fenyl og fenylalkyl, eller Rj og R3 med N-atomet som bærer dem, danner et heterocyklisk system: r\)m /-s?i .¿N og _N Y ' \_J \___/ hvor m er O, i, 2, 3 eller 4, n er O, l eller 2, Y' er O, S eller >N-R4 hvor R< er H, alkyl(CH2).-fenyl, hvor a er O, l, 2, 3 eller 4, xogyerO, l, 2, 3 eller 4, A er en gruppe med formel (a), og danner med det heterocykliske system som bærer den, tieno[2,3-d]pyrrolo- [l,2-a]pyrrol med formel (!¿) , og R5 og Rj er H, alkyl, hydroksy, alkoksy, halo, trifluormetyl, alkoksykarbonyl, -(CH2)p-fenyl, hvor p er O, l, 2, 3 eller 4 og -0-(CH2)p.- fenyl, hvor p' er O, l, 2, 3 eller 4, en gruppe med formel (6), og danner med det heterocykliske system som bærer den, tieno[3,2-d]pyrrolo[l,2-a]pyrrol med formel (IB), en gruppe med formel (7), og danner med det heter- ocykliske system som bærer den, danner pyrrolo[l,2-a]- indol med formel (IT), deres ds- eller trans-isomerer, deres enantiomerer eller diastereoisomerer og deres hydrater og/eller farmasøytisk akseptable addisjonssalt- er. Legemidler.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9415431A FR2728571B1 (fr) | 1994-12-22 | 1994-12-22 | Nouveaux ethers d'oximes tricycliques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO955215D0 NO955215D0 (no) | 1995-12-21 |
| NO955215L true NO955215L (no) | 1996-06-24 |
Family
ID=9470078
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO955215A NO955215L (no) | 1994-12-22 | 1995-12-21 | Nye tricykliske oximetere, fremgangsmåter ved deres fremstilling og farmasöytiske sammensetninger inneholdende dem |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US5627203A (no) |
| EP (1) | EP0718299B1 (no) |
| JP (1) | JP2937837B2 (no) |
| CN (2) | CN1066449C (no) |
| AT (1) | ATE191483T1 (no) |
| AU (1) | AU693615B2 (no) |
| CA (1) | CA2165618C (no) |
| DE (1) | DE69516100T2 (no) |
| DK (1) | DK0718299T3 (no) |
| ES (1) | ES2147271T3 (no) |
| FI (1) | FI956136A (no) |
| FR (1) | FR2728571B1 (no) |
| GR (1) | GR3033507T3 (no) |
| NO (1) | NO955215L (no) |
| NZ (1) | NZ280734A (no) |
| PT (1) | PT718299E (no) |
| ZA (1) | ZA9510901B (no) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2781482B1 (fr) * | 1998-07-27 | 2001-08-31 | Adir | Nouveaux derives de 8h-thieno-[2,3-b]pyrrolizine-8-one, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| WO2004047730A2 (en) * | 2002-11-21 | 2004-06-10 | New York Blood Center | Compounds for inhibition of hiv infection by blocking hiv entry |
| DE102008015032A1 (de) * | 2008-03-17 | 2009-09-24 | Aicuris Gmbh & Co. Kg | Substituierte Pyrazolamide und ihre Verwendung |
| DE102008015033A1 (de) * | 2008-03-17 | 2009-09-24 | Aicuris Gmbh & Co. Kg | Substituierte (Pyrazolyl-carbonyl)imidazolidinone und ihre Verwendung |
| DE102008062878A1 (de) | 2008-12-17 | 2010-06-24 | Aicuris Gmbh & Co. Kg | Substituierte Furancarboxamide und ihre Verwendung |
| DE102008062863A1 (de) | 2008-12-17 | 2010-06-24 | Aicuris Gmbh & Co. Kg | Substituierte (Thiophenyl-carbonyl)imidazolidinone und ihre Verwendung |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE371193B (no) * | 1972-03-24 | 1974-11-11 | Kabi Ab | |
| US4308399A (en) * | 1977-08-30 | 1981-12-29 | Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. | O-(3-Amino-2-hydroxy-propyl)-amidoxime derivatives, process for the preparation thereof and pharmaceutical compositions containing same |
| US4134894A (en) * | 1978-05-04 | 1979-01-16 | Warner-Lambert Company | Pyrrolo[1,2-a]indole compounds |
| HU180739B (en) * | 1979-07-03 | 1983-04-29 | Egyt Gyogyszervegyeszeti Gyar | Process for producing basic oxime-ethers |
| US5128364A (en) * | 1991-03-28 | 1992-07-07 | Merck Frosst Canada, Inc. | Pyrrolo[1,2-a]indole hydroxylamine derivatives as inhibitors of leukotriene biosynthesis |
-
1994
- 1994-12-22 FR FR9415431A patent/FR2728571B1/fr not_active Expired - Fee Related
-
1995
- 1995-12-19 DK DK95402865T patent/DK0718299T3/da active
- 1995-12-19 CA CA002165618A patent/CA2165618C/fr not_active Expired - Fee Related
- 1995-12-19 AT AT95402865T patent/ATE191483T1/de not_active IP Right Cessation
- 1995-12-19 EP EP95402865A patent/EP0718299B1/fr not_active Expired - Lifetime
- 1995-12-19 DE DE69516100T patent/DE69516100T2/de not_active Expired - Fee Related
- 1995-12-19 ES ES95402865T patent/ES2147271T3/es not_active Expired - Lifetime
- 1995-12-19 PT PT95402865T patent/PT718299E/pt unknown
- 1995-12-20 FI FI956136A patent/FI956136A/fi unknown
- 1995-12-20 AU AU40593/95A patent/AU693615B2/en not_active Ceased
- 1995-12-21 NO NO955215A patent/NO955215L/no not_active Application Discontinuation
- 1995-12-21 JP JP7333347A patent/JP2937837B2/ja not_active Expired - Lifetime
- 1995-12-21 US US08/576,678 patent/US5627203A/en not_active Expired - Fee Related
- 1995-12-21 ZA ZA9510901A patent/ZA9510901B/xx unknown
- 1995-12-21 NZ NZ280734A patent/NZ280734A/en unknown
- 1995-12-22 CN CN95120144A patent/CN1066449C/zh not_active Expired - Fee Related
-
1999
- 1999-12-03 CN CN99120993A patent/CN1261073A/zh active Pending
-
2000
- 2000-05-25 GR GR20000401198T patent/GR3033507T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| US5627203A (en) | 1997-05-06 |
| JPH08231554A (ja) | 1996-09-10 |
| JP2937837B2 (ja) | 1999-08-23 |
| CA2165618C (fr) | 2001-04-10 |
| ZA9510901B (en) | 1996-06-24 |
| EP0718299A1 (fr) | 1996-06-26 |
| FI956136A0 (fi) | 1995-12-20 |
| NO955215D0 (no) | 1995-12-21 |
| CN1066449C (zh) | 2001-05-30 |
| GR3033507T3 (en) | 2000-09-29 |
| AU4059395A (en) | 1996-06-27 |
| CN1131155A (zh) | 1996-09-18 |
| CN1261073A (zh) | 2000-07-26 |
| ATE191483T1 (de) | 2000-04-15 |
| FI956136A (fi) | 1996-06-23 |
| NZ280734A (en) | 1997-09-22 |
| EP0718299B1 (fr) | 2000-04-05 |
| DE69516100D1 (de) | 2000-05-11 |
| DK0718299T3 (da) | 2000-09-04 |
| PT718299E (pt) | 2000-07-31 |
| FR2728571A1 (fr) | 1996-06-28 |
| CA2165618A1 (fr) | 1996-06-23 |
| FR2728571B1 (fr) | 1997-01-31 |
| DE69516100T2 (de) | 2000-12-14 |
| AU693615B2 (en) | 1998-07-02 |
| ES2147271T3 (es) | 2000-09-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |