FI953777A0 - Heteroaromaattisia yhdisteitä, joilla on antipsykoottinen aktiivisuus - Google Patents

Heteroaromaattisia yhdisteitä, joilla on antipsykoottinen aktiivisuus

Info

Publication number
FI953777A0
FI953777A0 FI953777A FI953777A FI953777A0 FI 953777 A0 FI953777 A0 FI 953777A0 FI 953777 A FI953777 A FI 953777A FI 953777 A FI953777 A FI 953777A FI 953777 A0 FI953777 A0 FI 953777A0
Authority
FI
Finland
Prior art keywords
heteroaromatic compounds
antipsychotic activity
antipsychotic
activity
heteroaromatic
Prior art date
Application number
FI953777A
Other languages
English (en)
Swedish (sv)
Other versions
FI953777A (fi
Inventor
Mark Henry Norman
Iii Frank Navas
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of FI953777A publication Critical patent/FI953777A/fi
Publication of FI953777A0 publication Critical patent/FI953777A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D275/00Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI953777A 1993-02-10 1995-08-09 Heteroaromaattisia yhdisteitä, joilla on antipsykoottinen aktiivisuus FI953777A0 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB939302622A GB9302622D0 (en) 1993-02-10 1993-02-10 Heteroaromatic compounds
PCT/GB1994/000265 WO1994018196A1 (en) 1993-02-10 1994-02-10 Heteroaromatic compounds with antipsychotic activity

Publications (2)

Publication Number Publication Date
FI953777A FI953777A (fi) 1995-08-09
FI953777A0 true FI953777A0 (fi) 1995-08-09

Family

ID=10730183

Family Applications (1)

Application Number Title Priority Date Filing Date
FI953777A FI953777A0 (fi) 1993-02-10 1995-08-09 Heteroaromaattisia yhdisteitä, joilla on antipsykoottinen aktiivisuus

Country Status (15)

Country Link
EP (1) EP0683778A1 (fi)
JP (1) JPH08506337A (fi)
CN (1) CN1117731A (fi)
AU (1) AU6005194A (fi)
BG (1) BG99839A (fi)
CA (1) CA2155758A1 (fi)
CZ (1) CZ204495A3 (fi)
FI (1) FI953777A0 (fi)
GB (1) GB9302622D0 (fi)
HU (1) HUT73654A (fi)
IL (1) IL108601A0 (fi)
MX (1) MX9401080A (fi)
SK (1) SK99195A3 (fi)
WO (1) WO1994018196A1 (fi)
ZA (1) ZA94891B (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5364866A (en) 1989-05-19 1994-11-15 Hoechst-Roussel Pharmaceuticals, Inc. Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analetics
US5776963A (en) 1989-05-19 1998-07-07 Hoechst Marion Roussel, Inc. 3-(heteroaryl)-1- (2,3-dihydro-1h-isoindol-2-yl)alkyl!pyrrolidines and 3-(heteroaryl)-1- (2,3-dihydro-1h-indol-1-yl)alkyl!pyrrolidines and related compounds and their therapeutic untility
GB9420521D0 (en) * 1994-10-12 1994-11-30 Smithkline Beecham Plc Novel compounds
JP3274579B2 (ja) * 1995-01-12 2002-04-15 住友製薬株式会社 脳血管障害に伴う精神症候治療剤
DK0732332T3 (da) * 1995-03-17 2002-04-15 Aventis Pharma Inc Substituerede benzothienylpiperaziner, deres anvendelse som lægemidler og fremgangsmåder til fremstilling deraf
UA73981C2 (en) 2000-03-10 2005-10-17 Merck Patent Gmbh (r)-(-)-2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]-chromane for treatment of extrapyramidal movement disorders (variants), pharmaceutical composition and kit
RU2283648C2 (ru) * 2000-11-14 2006-09-20 Мерк Патент Гмбх Новое применение комбинированных селективных антагонистов допаминового рецептора d2 и агонистов рецептора 5-нт 1a
JP4497815B2 (ja) * 2001-02-16 2010-07-07 アベンティス・ファーマスーティカルズ・インコーポレイテツド 新規な複素環式アミド誘導体およびドーパミンd3受容体リガンドとしてのその使用
SI1408964T1 (sl) 2001-07-26 2007-06-30 Merck Patent Gmbh Uporaba 2- 5-(4-fluorofenil)-3-piridilmetil-aminometil -kromana in njegovih fizioloĺ ko sprejemljivih soli
GB0222912D0 (en) 2002-10-03 2002-11-13 Astrazeneca Ab Novel process and intermediates
GB0222909D0 (en) * 2002-10-03 2002-11-13 Astrazeneca Ab Novel process and intermediates
ZA200700527B (en) * 2004-07-20 2008-08-27 Siena Biotech Spa Modulators of alpha7 nicotinic acetylcholine receptors and therapeutic uses thereof
CL2008000119A1 (es) 2007-01-16 2008-05-16 Wyeth Corp Compuestos derivados de pirazol, antagonistas del receptor nicotinico de acetilcolina; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como demencia senil, alzheimer y esquizofrenia.
EP2736905A4 (en) * 2011-07-28 2015-07-29 Mapi Pharma Ltd INTERMEDIATE COMPOUNDS AND PROCESS FOR THE PREPARATION OF LURASIDONE AND SALTS THEREOF

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0625181B2 (ja) * 1985-03-27 1994-04-06 住友製薬株式会社 新規なイミド誘導体
AU593194B2 (en) * 1986-09-26 1990-02-01 Sumitomo Pharmaceuticals Company, Limited Imide derivatives ,and their production and use
US5143923B1 (en) * 1991-04-29 1993-11-02 Hoechst-Roussel Pharmaceuticals Incorporated Benzoisothiazole-and benzisoxazole-3-carboxamides
IL101722A (en) * 1991-05-02 1996-05-14 Wyeth John & Brother Ltd History of piperazine, their preparation and pharmaceutical preparations containing them

Also Published As

Publication number Publication date
AU6005194A (en) 1994-08-29
CA2155758A1 (en) 1994-08-18
HU9501881D0 (en) 1995-08-28
EP0683778A1 (en) 1995-11-29
MX9401080A (es) 1994-08-31
IL108601A0 (en) 1994-05-30
CZ204495A3 (en) 1996-03-13
WO1994018196A1 (en) 1994-08-18
JPH08506337A (ja) 1996-07-09
HUT73654A (en) 1996-09-30
GB9302622D0 (en) 1993-03-24
CN1117731A (zh) 1996-02-28
FI953777A (fi) 1995-08-09
SK99195A3 (en) 1995-12-06
ZA94891B (en) 1995-08-10
BG99839A (bg) 1996-02-28

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Legal Events

Date Code Title Description
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