FI930621A7 - Bifenylsubstituerade kinolinderivat - Google Patents

Bifenylsubstituerade kinolinderivat Download PDF

Info

Publication number
FI930621A7
FI930621A7 FI930621A FI930621A FI930621A7 FI 930621 A7 FI930621 A7 FI 930621A7 FI 930621 A FI930621 A FI 930621A FI 930621 A FI930621 A FI 930621A FI 930621 A7 FI930621 A7 FI 930621A7
Authority
FI
Finland
Prior art keywords
biphenylsubstituerade
differents
quinoline
quinoline differents
biphenylsubstituerade quinoline
Prior art date
Application number
FI930621A
Other languages
English (en)
Finnish (fi)
Other versions
FI930621A0 (fi
Inventor
Denis Evan Ryono
John Lloyd
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of FI930621A0 publication Critical patent/FI930621A0/fi
Publication of FI930621A7 publication Critical patent/FI930621A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI930621A 1992-02-14 1993-02-12 Bifenylsubstituerade kinolinderivat FI930621A7 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US83778292A 1992-02-14 1992-02-14

Publications (2)

Publication Number Publication Date
FI930621A0 FI930621A0 (fi) 1993-02-12
FI930621A7 true FI930621A7 (fi) 1993-08-15

Family

ID=25275409

Family Applications (1)

Application Number Title Priority Date Filing Date
FI930621A FI930621A7 (fi) 1992-02-14 1993-02-12 Bifenylsubstituerade kinolinderivat

Country Status (16)

Country Link
EP (1) EP0556060A1 (OSRAM)
JP (1) JPH05286939A (OSRAM)
KR (1) KR930017891A (OSRAM)
CN (1) CN1044243C (OSRAM)
AU (1) AU656454B2 (OSRAM)
CA (1) CA2089185A1 (OSRAM)
FI (1) FI930621A7 (OSRAM)
HU (1) HU217627B (OSRAM)
IL (1) IL104623A (OSRAM)
MX (1) MX9300742A (OSRAM)
NO (1) NO930520L (OSRAM)
NZ (1) NZ245757A (OSRAM)
PL (1) PL172241B1 (OSRAM)
RU (1) RU2122540C1 (OSRAM)
TW (1) TW297025B (OSRAM)
ZA (1) ZA93531B (OSRAM)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5767129A (en) * 1995-08-24 1998-06-16 Warner-Lambert Company Substituted quinolines and isoquinolines as calcium channel blockers, their preparation and the use thereof
US6455554B1 (en) 1999-06-07 2002-09-24 Targacept, Inc. Oxopyridinyl pharmaceutical compositions and methods for use
ES2274005T3 (es) 2001-01-26 2007-05-16 Chugai Seiyaku Kabushiki Kaisha Inhibidores de malonyl-coa decarboxilasa usados como moduladores metabolicos.
JP4503232B2 (ja) 2001-01-26 2010-07-14 中外製薬株式会社 マロニル−CoA脱炭酸酵素阻害剤を用いた疾患の治療法
CA2735267C (en) 2001-01-26 2013-05-07 Chugai Seiyaku Kabushiki Kaisha Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
ES2330417T3 (es) 2001-02-20 2009-12-10 Chugai Seiyaku Kabushiki Kaisha Procedimientos para tratar enfermedades metabolicas usando inhibidores de malonil coa descarboxilasa.
US7709510B2 (en) 2001-02-20 2010-05-04 Chugai Seiyaku Kabushiki Kaisha Azoles as malonyl-CoA decarboxylase inhibitors useful as metabolic modulators
RU2201753C1 (ru) * 2002-03-12 2003-04-10 Нестерук Владимир Викторович Фармацевтическая композиция, обладающая диуретическим, дегидратирующим и гипотензивным действием
PE20040950A1 (es) * 2003-02-14 2005-01-01 Theravance Inc DERIVADOS DE BIFENILO COMO AGONISTAS DE LOS RECEPTORES ADRENERGICOS ß2 Y COMO ANTAGONISTAS DE LOS RECEPTORES MUSCARINICOS
WO2005011670A1 (en) 2003-08-01 2005-02-10 Chugai Seiyaku Kabushiki Kaisha Heterocyclic compounds useful as malonyl-coa decarboxylase inhibitors
CA2533749C (en) 2003-08-01 2012-07-10 Chugai Seiyaku Kabushiki Kaisha Piperidine compounds useful as malonyl-coa decarboxylase inhibitors
EP2208495B1 (en) 2003-08-01 2011-12-14 Chugai Seiyaku Kabushiki Kaisha Cyanoguanidine-based azole compounds useful as malonyl-CoA decarboxylase inhibitors
EP1648564B1 (en) 2003-08-01 2007-10-17 Chugai Seiyaku Kabushiki Kaisha Cyanoamide compounds useful as malonyl-coa decarboxylase inhibitors
TWI374883B (en) * 2004-08-16 2012-10-21 Theravance Inc Crystalline form of a biphenyl compound
PT1928457E (pt) 2005-09-30 2013-02-19 Pulmagen Therapeutics Asthma Ltd Quinolinas e sua utilização terapêutica
GB0519969D0 (en) * 2005-09-30 2005-11-09 Argenta Discovery Ltd Quinoline compounds
EA017093B1 (ru) * 2007-04-04 2012-09-28 Пульмаджен Терапьютикс (Эсме) Лимитед Хинолины и их терапевтическое применение

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4880804A (en) * 1988-01-07 1989-11-14 E. I. Du Pont De Nemours And Company Angiotensin II receptor blocking benzimidazoles
IE903911A1 (en) * 1989-11-20 1991-05-22 Ici Plc Diazine derivatives
US5049565A (en) * 1990-12-07 1991-09-17 Merck & Co., Inc. Microbial transformation process for preparing anti-hypertensive products
GB9102727D0 (en) * 1991-02-08 1991-03-27 Ici Plc Pharmaceutical agent
US5157040A (en) * 1991-04-05 1992-10-20 Merck & Co., Inc. Substituted quinolines as angiotensin ii antagonists

Also Published As

Publication number Publication date
JPH05286939A (ja) 1993-11-02
FI930621A0 (fi) 1993-02-12
RU2122540C1 (ru) 1998-11-27
PL297713A1 (en) 1993-08-23
CN1075720A (zh) 1993-09-01
EP0556060A1 (en) 1993-08-18
PL172241B1 (pl) 1997-08-29
HU217627B (hu) 2000-03-28
AU3299193A (en) 1993-08-19
CA2089185A1 (en) 1993-08-15
CN1044243C (zh) 1999-07-21
NO930520L (no) 1993-08-16
KR930017891A (ko) 1993-09-20
IL104623A0 (en) 1993-06-10
TW297025B (OSRAM) 1997-02-01
MX9300742A (es) 1993-09-01
ZA93531B (en) 1993-08-26
IL104623A (en) 1996-12-05
NO930520D0 (no) 1993-02-12
HU9300386D0 (en) 1993-04-28
HUT69694A (en) 1995-09-28
AU656454B2 (en) 1995-02-02
NZ245757A (en) 1995-09-26

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