FI924354L - Imidazolylpropensyraderivat - Google Patents

Imidazolylpropensyraderivat Download PDF

Info

Publication number
FI924354L
FI924354L FI924354A FI924354A FI924354L FI 924354 L FI924354 L FI 924354L FI 924354 A FI924354 A FI 924354A FI 924354 A FI924354 A FI 924354A FI 924354 L FI924354 L FI 924354L
Authority
FI
Finland
Prior art keywords
imidazolylpropeneic
acid derivatives
derivatives
acid
imidazolylpropeneic acid
Prior art date
Application number
FI924354A
Other languages
English (en)
Finnish (fi)
Other versions
FI924354A0 (fi
FI924354A7 (fi
Inventor
Thomas Kraemer
Juergen Dressel
Rudolf Hanko
Walter Huebsch
Ulrich Mueller
Matthias Mueller-Gliemann
Martin Beuck
Stanislav Kazda
Johannes-Peter Stasch
Andreas Knorr
Stefan Wohlfeil
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of FI924354A0 publication Critical patent/FI924354A0/fi
Publication of FI924354A7 publication Critical patent/FI924354A7/fi
Publication of FI924354L publication Critical patent/FI924354L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI924354A 1991-10-01 1992-09-29 Imidazolylpropensyraderivat FI924354L (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4132631A DE4132631A1 (de) 1991-10-01 1991-10-01 Imidazolyl-propensaeurederivate

Publications (3)

Publication Number Publication Date
FI924354A0 FI924354A0 (fi) 1992-09-29
FI924354A7 FI924354A7 (fi) 1993-04-02
FI924354L true FI924354L (fi) 1993-04-02

Family

ID=6441873

Family Applications (1)

Application Number Title Priority Date Filing Date
FI924354A FI924354L (fi) 1991-10-01 1992-09-29 Imidazolylpropensyraderivat

Country Status (15)

Country Link
US (1) US5294633A (cs)
EP (1) EP0535463A1 (cs)
JP (1) JPH05213938A (cs)
KR (1) KR930007936A (cs)
AU (1) AU646977B2 (cs)
CA (1) CA2079281A1 (cs)
CZ (1) CZ298892A3 (cs)
DE (1) DE4132631A1 (cs)
FI (1) FI924354L (cs)
HU (1) HUT62577A (cs)
IL (1) IL103291A0 (cs)
MX (1) MX9205436A (cs)
NO (1) NO923579L (cs)
TW (1) TW208701B (cs)
ZA (1) ZA927501B (cs)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4132633A1 (de) * 1991-10-01 1993-04-08 Bayer Ag Cyclisch substituierte imidazolyl-propensaeurederivate
AT398202B (de) * 1991-10-04 1994-10-25 Chem Pharm Forsch Gmbh Neue imidazolderivate, verfahren zu ihrer herstellung und ihre verwendung
ATE266402T1 (de) * 1994-03-16 2004-05-15 Sankyo Co Okulares hypotonikum
CA2186606A1 (en) * 1994-03-29 1995-10-05 Edward B. Nelson Treatment of atherosclerosis with angiotensin ii receptor blocking imidazoles
CN103601792B (zh) 2007-06-04 2016-06-29 协同医药品公司 有效用于胃肠功能紊乱、炎症、癌症和其他疾病治疗的鸟苷酸环化酶激动剂
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
WO2009149279A2 (en) 2008-06-04 2009-12-10 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
WO2010009319A2 (en) 2008-07-16 2010-01-21 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal, inflammation, cancer and other disorders
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
US9486494B2 (en) 2013-03-15 2016-11-08 Synergy Pharmaceuticals, Inc. Compositions useful for the treatment of gastrointestinal disorders
WO2014151206A1 (en) 2013-03-15 2014-09-25 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase and their uses
CA2913737A1 (en) 2013-06-05 2014-12-11 Synergy Pharmaceuticals, Inc. Ultra-pure agonists of guanylate cyclase c, method of making and using same

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5138069A (en) * 1986-07-11 1992-08-11 E. I. Du Pont De Nemours And Company Angiotensin II receptor blocking imidazoles
CA2018443A1 (en) * 1989-06-14 1990-12-14 Joseph A. Finkelstein Imidazolyl-alkenoic acids
DK0955294T3 (da) * 1989-06-14 2004-02-02 Smithkline Beecham Corp Imidazolylalkensyre
WO1991000281A2 (en) * 1989-06-30 1991-01-10 E.I. Du Pont De Nemours And Company Fused-ring aryl substituted imidazoles
DK0479903T3 (da) * 1989-06-30 1996-03-18 Du Pont Substituerede imidazoler og deres anvendelse som angiotensin II hæmmere
AU640417B2 (en) * 1989-10-25 1993-08-26 Smithkline Beecham Corporation Substituted 5-((tetrazolyl)alkenyl)imidazoles
GB9017482D0 (en) * 1990-08-09 1990-09-26 Ici Plc Manufacturing process
DE4132632A1 (de) * 1991-10-01 1993-04-08 Bayer Ag Substituierte imidazolyl-propensaeurederivate

Also Published As

Publication number Publication date
CA2079281A1 (en) 1993-04-02
EP0535463A1 (de) 1993-04-07
FI924354A0 (fi) 1992-09-29
AU2602392A (en) 1993-04-08
ZA927501B (en) 1993-05-03
HU9203124D0 (en) 1992-12-28
IL103291A0 (en) 1993-02-21
TW208701B (cs) 1993-07-01
NO923579D0 (no) 1992-09-15
KR930007936A (ko) 1993-05-20
HUT62577A (en) 1993-05-28
JPH05213938A (ja) 1993-08-24
US5294633A (en) 1994-03-15
MX9205436A (es) 1993-04-01
FI924354A7 (fi) 1993-04-02
NO923579L (no) 1993-04-02
AU646977B2 (en) 1994-03-10
DE4132631A1 (de) 1993-04-08
CZ298892A3 (en) 1993-04-14

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