FI914487A0 - 1,3-bensoxazinderivat, deras framstaellning och anvaendning. - Google Patents

1,3-bensoxazinderivat, deras framstaellning och anvaendning.

Info

Publication number
FI914487A0
FI914487A0 FI914487A FI914487A FI914487A0 FI 914487 A0 FI914487 A0 FI 914487A0 FI 914487 A FI914487 A FI 914487A FI 914487 A FI914487 A FI 914487A FI 914487 A0 FI914487 A0 FI 914487A0
Authority
FI
Finland
Prior art keywords
benzozazinderivat
deras framstaellning
framstaellning och
och anvaendning
anvaendning
Prior art date
Application number
FI914487A
Other languages
English (en)
Other versions
FI914487A (fi
Inventor
Mitsuru Shiraishi
Shohei Hashiguchi
Toshifumi Watanabe
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of FI914487A0 publication Critical patent/FI914487A0/fi
Publication of FI914487A publication Critical patent/FI914487A/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/041,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/121,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/141,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/161,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with only hydrogen or carbon atoms directly attached in positions 2 and 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
FI914487A 1990-09-25 1991-09-24 1,3-bensoxazinderivat, deras framstaellning och anvaendning. FI914487A (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP25647890 1990-09-25
JP41705090 1990-12-28
JP7674291 1991-03-15
JP20423591 1991-08-14

Publications (2)

Publication Number Publication Date
FI914487A0 true FI914487A0 (fi) 1991-09-24
FI914487A FI914487A (fi) 1992-03-26

Family

ID=27465972

Family Applications (1)

Application Number Title Priority Date Filing Date
FI914487A FI914487A (fi) 1990-09-25 1991-09-24 1,3-bensoxazinderivat, deras framstaellning och anvaendning.

Country Status (14)

Country Link
US (1) US5270308A (fi)
EP (1) EP0477789A1 (fi)
KR (1) KR920006336A (fi)
CN (1) CN1060467A (fi)
AU (1) AU640820B2 (fi)
CA (1) CA2052145A1 (fi)
CS (1) CS293291A3 (fi)
FI (1) FI914487A (fi)
HU (1) HUT62003A (fi)
IE (1) IE913186A1 (fi)
IL (1) IL99474A0 (fi)
NO (1) NO913745L (fi)
PL (1) PL291823A1 (fi)
PT (1) PT99030A (fi)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE152102T1 (de) * 1991-05-10 1997-05-15 Takeda Chemical Industries Ltd Pyridinderivate, deren herstellung und anwendung
KR100231634B1 (ko) * 1992-08-17 1999-11-15 나가야마 오사무 벤조피란 및 벤족사진 유도체
GB9309716D0 (en) * 1993-05-12 1993-06-23 Zeneca Ltd Heterocyclic derivatives
JP3814742B2 (ja) * 1996-10-18 2006-08-30 イハラケミカル工業株式会社 4−フルオロサリチル酸類
US6265417B1 (en) * 1997-12-18 2001-07-24 Abbott Laboratories Potassium channel openers
US6593335B1 (en) * 1997-12-18 2003-07-15 Abbott Laboratories Potassium channel openers
US6455554B1 (en) 1999-06-07 2002-09-24 Targacept, Inc. Oxopyridinyl pharmaceutical compositions and methods for use
US6538004B2 (en) * 2000-03-03 2003-03-25 Abbott Laboratories Tricyclic dihydropyrazolone and tricyclic dihydroisoxazolone potassium channel openers
JP2007504202A (ja) * 2003-09-04 2007-03-01 ポセイドン ファーマシュティカルズ アクティーゼルスカブ 心臓不整脈を治療するためのergチャネル開口薬
WO2006002470A1 (en) * 2004-06-30 2006-01-12 Monash University Chiral ligands for asymmetric catalysis
US8258131B2 (en) * 2007-08-01 2012-09-04 Mitsubishi Tanabe Pharma Corporation Fused bicyclic compound
US8389758B2 (en) * 2009-06-05 2013-03-05 3M Innovative Properties Company Benzoxazine-thiol adducts
US8383706B2 (en) 2009-06-05 2013-02-26 3M Innovative Properties Company Benzoxazine-thiol adducts
AU2010276537B2 (en) 2009-07-27 2015-04-16 Gilead Sciences, Inc. Fused heterocyclic compounds as ion channel modulators
EP2588197B1 (en) 2010-07-02 2014-11-05 Gilead Sciences, Inc. Fused heterocyclic compounds as ion channel modulators
TWI510480B (zh) 2011-05-10 2015-12-01 Gilead Sciences Inc 充當離子通道調節劑之稠合雜環化合物
TW201837023A (zh) 2011-07-01 2018-10-16 美商基利科學股份有限公司 作為離子通道調節劑之稠合雜環化合物
NO3175985T3 (fi) 2011-07-01 2018-04-28
ITMI20122221A1 (it) * 2012-12-21 2014-06-22 C4T S C A R L Nuovi composti del 2,3-diidro-4h-1,3-benzossazin-4-one, metodo per prepararli e forma farmaceutica che li comprende
CN109336781A (zh) * 2018-12-12 2019-02-15 湖南海利常德农药化工有限公司 一种水杨腈的纯化方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2321496A1 (de) 1973-04-27 1974-11-14 Nii Farmakol Akad Med 2-aminomethyl-4,4-dialkyl-4h-1,3-benzoxazine, deren salze und verfahren zu ihrer herstellung
JPS57130979A (en) 1981-02-09 1982-08-13 Sankyo Co Ltd 4-amino-1,3-benzoxazine derivative and its preparation
ZM7682A1 (en) 1981-09-25 1983-05-23 Beecham Group Plc Active compounds
EP0076075B1 (en) * 1981-09-25 1986-11-20 Beecham Group Plc Pharmaceutically active benzopyran compounds
US4971982A (en) 1987-07-06 1990-11-20 Hoffmann-La Roche Inc. Benzopyran derivatives
US5021432A (en) 1988-04-26 1991-06-04 Yoshitomi Pharmaceutical Industries, Ltd. Benzopyran compound and its pharmaceutical use
DE3840011A1 (de) * 1988-11-26 1990-05-31 Merck Patent Gmbh Benzoxazinderivate
TW224941B (fi) * 1989-11-08 1994-06-11 Yamanouchi Pharma Co Ltd

Also Published As

Publication number Publication date
CA2052145A1 (en) 1992-03-26
PT99030A (pt) 1992-09-30
EP0477789A1 (en) 1992-04-01
HU913050D0 (en) 1992-01-28
HUT62003A (en) 1993-03-29
FI914487A (fi) 1992-03-26
AU640820B2 (en) 1993-09-02
IE913186A1 (en) 1992-02-25
KR920006336A (ko) 1992-04-27
PL291823A1 (en) 1992-08-24
NO913745D0 (no) 1991-09-24
US5270308A (en) 1993-12-14
AU8474891A (en) 1992-04-02
NO913745L (no) 1992-03-26
CN1060467A (zh) 1992-04-22
CS293291A3 (en) 1992-08-12
IL99474A0 (en) 1992-08-18

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Legal Events

Date Code Title Description
FD Application lapsed