FI913369A - Tioxoheterocykler. - Google Patents

Tioxoheterocykler. Download PDF

Info

Publication number
FI913369A
FI913369A FI913369A FI913369A FI913369A FI 913369 A FI913369 A FI 913369A FI 913369 A FI913369 A FI 913369A FI 913369 A FI913369 A FI 913369A FI 913369 A FI913369 A FI 913369A
Authority
FI
Finland
Prior art keywords
sulphinyl
sulphonyl
thio
oxy
alkylene
Prior art date
Application number
FI913369A
Other languages
English (en)
Finnish (fi)
Other versions
FI913369A0 (fi
Inventor
Pierre Andre Raymond Bruneau
Original Assignee
Ici Pharma
Ici Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ici Pharma, Ici Plc filed Critical Ici Pharma
Publication of FI913369A0 publication Critical patent/FI913369A0/fi
Publication of FI913369A publication Critical patent/FI913369A/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D245/00—Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Detergent Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Quinoline Compounds (AREA)
FI913369A 1990-07-13 1991-07-11 Tioxoheterocykler. FI913369A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP90402034 1990-07-13
EP91400079 1991-01-15

Publications (2)

Publication Number Publication Date
FI913369A0 FI913369A0 (fi) 1991-07-11
FI913369A true FI913369A (fi) 1992-01-14

Family

ID=26127361

Family Applications (1)

Application Number Title Priority Date Filing Date
FI913369A FI913369A (fi) 1990-07-13 1991-07-11 Tioxoheterocykler.

Country Status (22)

Country Link
US (1) US5240941A (es)
EP (1) EP0466452B1 (es)
JP (1) JPH04243877A (es)
KR (1) KR920002561A (es)
AT (1) ATE128133T1 (es)
AU (1) AU638579B2 (es)
CA (1) CA2046006A1 (es)
CS (1) CS214891A3 (es)
DE (1) DE69113148T2 (es)
DK (1) DK0466452T3 (es)
ES (1) ES2076472T3 (es)
FI (1) FI913369A (es)
GB (1) GB9113137D0 (es)
GR (1) GR3017453T3 (es)
HU (1) HUT61999A (es)
IE (1) IE912138A1 (es)
IL (1) IL98603A0 (es)
MX (1) MX174406B (es)
NO (1) NO912750L (es)
NZ (1) NZ238703A (es)
PT (1) PT98292A (es)
TW (1) TW235918B (es)

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US5643933A (en) * 1995-06-02 1997-07-01 G. D. Searle & Co. Substituted sulfonylphenylheterocycles as cyclooxygenase-2 and 5-lipoxygenase inhibitors
US6677364B2 (en) * 1998-04-20 2004-01-13 G.D. Searle & Co. Substituted sulfonylphenylheterocycles as cyclooxygenase-2 and 5-lipoxygenase inhibitors
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US8158362B2 (en) 2005-03-30 2012-04-17 Decode Genetics Ehf. Methods of diagnosing susceptibility to myocardial infarction and screening for an LTA4H haplotype
WO2006068760A2 (en) 2004-11-19 2006-06-29 The Regents Of The University Of California Anti-inflammatory pyrazolopyrimidines
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US8193182B2 (en) 2008-01-04 2012-06-05 Intellikine, Inc. Substituted isoquinolin-1(2H)-ones, and methods of use thereof
ES2647163T3 (es) 2008-01-04 2017-12-19 Intellikine, Inc. Derivados de isoquinolinona sustituidos con una purina útiles como inhibidores de la PI3K
EP2252293B1 (en) 2008-03-14 2018-06-27 Intellikine, LLC Kinase inhibitors and methods of use
US8993580B2 (en) 2008-03-14 2015-03-31 Intellikine Llc Benzothiazole kinase inhibitors and methods of use
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WO2010006072A2 (en) 2008-07-08 2010-01-14 The Regents Of The University Of California Mtor modulators and uses thereof
CA2738429C (en) 2008-09-26 2016-10-25 Intellikine, Inc. Heterocyclic kinase inhibitors
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US8476431B2 (en) 2008-11-03 2013-07-02 Itellikine LLC Benzoxazole kinase inhibitors and methods of use
EP2427195B1 (en) 2009-05-07 2019-05-01 Intellikine, LLC Heterocyclic compounds and uses thereof
US8980899B2 (en) 2009-10-16 2015-03-17 The Regents Of The University Of California Methods of inhibiting Ire1
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WO2012088266A2 (en) 2010-12-22 2012-06-28 Incyte Corporation Substituted imidazopyridazines and benzimidazoles as inhibitors of fgfr3
CA2824197C (en) 2011-01-10 2020-02-25 Michael Martin Processes for preparing isoquinolinones and solid forms of isoquinolinones
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US8828998B2 (en) 2012-06-25 2014-09-09 Infinity Pharmaceuticals, Inc. Treatment of lupus, fibrotic conditions, and inflammatory myopathies and other disorders using PI3 kinase inhibitors
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US9266892B2 (en) 2012-12-19 2016-02-23 Incyte Holdings Corporation Fused pyrazoles as FGFR inhibitors
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US9751888B2 (en) 2013-10-04 2017-09-05 Infinity Pharmaceuticals, Inc. Heterocyclic compounds and uses thereof
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US11628162B2 (en) 2019-03-08 2023-04-18 Incyte Corporation Methods of treating cancer with an FGFR inhibitor
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Also Published As

Publication number Publication date
TW235918B (es) 1994-12-11
CS214891A3 (en) 1992-02-19
DK0466452T3 (da) 1996-01-02
ES2076472T3 (es) 1995-11-01
MX174406B (es) 1994-05-13
DE69113148D1 (de) 1995-10-26
IE912138A1 (en) 1992-01-15
NO912750D0 (no) 1991-07-12
GR3017453T3 (en) 1995-12-31
AU638579B2 (en) 1993-07-01
GB9113137D0 (en) 1991-08-07
DE69113148T2 (de) 1996-03-28
AU7933791A (en) 1992-01-16
EP0466452A2 (en) 1992-01-15
CA2046006A1 (en) 1992-01-14
US5240941A (en) 1993-08-31
JPH04243877A (ja) 1992-08-31
FI913369A0 (fi) 1991-07-11
HU912295D0 (en) 1991-12-30
KR920002561A (ko) 1992-02-28
EP0466452B1 (en) 1995-09-20
PT98292A (pt) 1992-05-29
ATE128133T1 (de) 1995-10-15
NO912750L (no) 1992-01-14
NZ238703A (en) 1994-01-26
HUT61999A (en) 1993-03-29
EP0466452A3 (en) 1992-08-19
IL98603A0 (en) 1992-07-15

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