FI91257B - Förfarande för framställning av terapeutiskt användbara 4-oxo-4H-pyrido/1,2-a/pyrimidin-3-karboxamidderivat - Google Patents

Förfarande för framställning av terapeutiskt användbara 4-oxo-4H-pyrido/1,2-a/pyrimidin-3-karboxamidderivat Download PDF

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Publication number
FI91257B
FI91257B FI890478A FI890478A FI91257B FI 91257 B FI91257 B FI 91257B FI 890478 A FI890478 A FI 890478A FI 890478 A FI890478 A FI 890478A FI 91257 B FI91257 B FI 91257B
Authority
FI
Finland
Prior art keywords
oxo
pyrido
mol
pyrimidine
chloroform
Prior art date
Application number
FI890478A
Other languages
English (en)
Finnish (fi)
Other versions
FI91257C (sv
FI890478A (sv
FI890478A0 (sv
Inventor
Judit Sipos
Jozsef Knoll
Istven Hermecz
Nee Debreczy Lelle Vasveri
Klera Gyires
Agnes Horveth
Leszlo Tardos
Meria Balogh
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of FI890478A0 publication Critical patent/FI890478A0/sv
Publication of FI890478A publication Critical patent/FI890478A/sv
Application granted granted Critical
Publication of FI91257B publication Critical patent/FI91257B/sv
Publication of FI91257C publication Critical patent/FI91257C/sv

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI890478A 1988-02-03 1989-02-01 Förfarande för framställning av terapeutiskt användbara 4-oxo-4H-pyrido/1,2-a/pyrimidin-3-karboxamidderivat FI91257C (sv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU50188 1988-02-03
HU88501A HU201551B (en) 1988-02-03 1988-02-03 Process for producing 4-oxo-4h-pyrido(1,2-a)pyrimidine-3-carboxylic acid amide derivatives and pharmaceutical compositions comprising same

Publications (4)

Publication Number Publication Date
FI890478A0 FI890478A0 (sv) 1989-02-01
FI890478A FI890478A (sv) 1989-08-04
FI91257B true FI91257B (sv) 1994-02-28
FI91257C FI91257C (sv) 1994-06-10

Family

ID=10949869

Family Applications (1)

Application Number Title Priority Date Filing Date
FI890478A FI91257C (sv) 1988-02-03 1989-02-01 Förfarande för framställning av terapeutiskt användbara 4-oxo-4H-pyrido/1,2-a/pyrimidin-3-karboxamidderivat

Country Status (18)

Country Link
US (1) US5158951A (sv)
EP (1) EP0326981B1 (sv)
JP (1) JPH01265090A (sv)
CN (1) CN1027263C (sv)
AT (1) ATE113948T1 (sv)
AU (1) AU611526B2 (sv)
CZ (1) CZ72689A3 (sv)
DD (1) DD283392A5 (sv)
DE (1) DE58908613D1 (sv)
DK (1) DK48389A (sv)
ES (1) ES2063771T3 (sv)
FI (1) FI91257C (sv)
HU (1) HU201551B (sv)
IL (1) IL89140A (sv)
NO (1) NO170281C (sv)
NZ (1) NZ227822A (sv)
RU (2) RU1820909C (sv)
YU (1) YU47205B (sv)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5580872A (en) * 1990-05-02 1996-12-03 Abbott Laboratories Quinolizinone type compounds
CA2727651C (en) * 2008-06-17 2016-04-05 Priscille Brodin Anti-infective compounds
AU2013347383B2 (en) * 2012-11-19 2017-04-06 Jiangsu Hansoh Pharmaceutical Co., Ltd. Pyrrole sulfonamide derivative, preparation method for same, and medical application thereof
CN104447491B (zh) * 2014-11-19 2017-06-23 连云港恒运医药有限公司 含吡咯环质子泵抑制剂的半富马酸盐及其中间体和医药用途
EP3344625A4 (en) * 2015-09-04 2019-03-27 Lysosomal Therapeutics Inc. THIAZOLO (3,2-A) PYRIMIDINONE AND OTHER HETEROBICYCLIC COMPOUNDS OF PYRIMIDINONE FOR THERAPEUTIC USE
WO2023102639A1 (en) * 2021-12-07 2023-06-15 Inca Renewable Technologies Inc. Methods for increasing absorption capacity of plant hurd material and products therefrom

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT302311B (de) * 1966-11-02 1972-09-15 Chinoin Gyogyszer Es Vegyeszet Verfahren zur herstellung von homopyrimidazol-derivaten und deren saeureadditionssalzen und quaternaeren ammoniumsalzen
HU168014B (sv) * 1973-03-30 1976-02-28
US4209622A (en) * 1973-03-30 1980-06-24 Chinoin Gygyszer es Vegyeszeti Termekek Gyara Rt. 3-(Ethoxycarbonyl-methyl)-6-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine
US4495189A (en) * 1975-11-27 1985-01-22 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara R.T. Condensed pyrimidines
HU173438B (hu) * 1975-11-27 1979-05-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh 4-okso-1,6,7,8-/tetragidro-4h-pirido/1,2/pirimidina s zaderzhivajuhhejj vozgoranie aktivnot'ju i protivosvertivajuhhem effektom
HU180439B (en) * 1977-12-29 1983-03-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-amino-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives
US4192944A (en) * 1978-04-03 1980-03-11 Bristol-Myers Company Optionally substituted 4-oxo-4H-pyrido[1,2-a]pyrimidine-3-N-(1H-tetrazol-4-yl)carboxamides and their use as antiallergy agents
US4666912A (en) * 1984-11-12 1987-05-19 Chinoin Gyogyszer Es Vegyeszeti Termeker Gyara Rt Treating process

Also Published As

Publication number Publication date
ES2063771T3 (es) 1995-01-16
US5158951A (en) 1992-10-27
JPH01265090A (ja) 1989-10-23
RU2051917C1 (ru) 1996-01-10
DK48389A (da) 1989-08-04
DK48389D0 (da) 1989-02-02
FI91257C (sv) 1994-06-10
AU2959489A (en) 1989-08-03
CN1036762A (zh) 1989-11-01
YU47205B (sh) 1995-01-31
IL89140A (en) 1993-01-14
CZ72689A3 (en) 1997-08-13
CN1027263C (zh) 1995-01-04
RU1820909C (ru) 1993-06-07
DD283392A5 (de) 1990-10-10
NO170281B (no) 1992-06-22
HUT49608A (en) 1989-10-30
NO890431L (no) 1989-08-04
FI890478A (sv) 1989-08-04
IL89140A0 (en) 1989-09-10
NO170281C (no) 1992-09-30
DE58908613D1 (de) 1994-12-15
EP0326981B1 (de) 1994-11-09
FI890478A0 (sv) 1989-02-01
AU611526B2 (en) 1991-06-13
NO890431D0 (no) 1989-02-02
ATE113948T1 (de) 1994-11-15
YU26089A (en) 1990-06-30
EP0326981A2 (de) 1989-08-09
EP0326981A3 (de) 1991-03-13
HU201551B (en) 1990-11-28
NZ227822A (en) 1990-08-28

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Legal Events

Date Code Title Description
BB Publication of examined application
MM Patent lapsed
MM Patent lapsed

Owner name: CHINOIN GYOGUSZER ES VEGYESZETI TERMEKEK