FI884595A - Menetelmä terapeuttisesti käyttökelpoisten imidatso/1,5-a/tieno/3,2-d/- ja -/3,2-e/pyrimidiinien valmistamiseksi - Google Patents

Menetelmä terapeuttisesti käyttökelpoisten imidatso/1,5-a/tieno/3,2-d/- ja -/3,2-e/pyrimidiinien valmistamiseksi Download PDF

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Publication number
FI884595A
FI884595A FI884595A FI884595A FI884595A FI 884595 A FI884595 A FI 884595A FI 884595 A FI884595 A FI 884595A FI 884595 A FI884595 A FI 884595A FI 884595 A FI884595 A FI 884595A
Authority
FI
Finland
Prior art keywords
thieno
pyrimidines
preparation
therapeutically useful
chem
Prior art date
Application number
FI884595A
Other languages
English (en)
Swedish (sv)
Other versions
FI91759B (fi
FI91759C (fi
FI884595A0 (fi
Inventor
Frank Waetjen
Holger Claus Hansen
Original Assignee
Ferrosan As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferrosan As filed Critical Ferrosan As
Publication of FI884595A0 publication Critical patent/FI884595A0/fi
Publication of FI884595A publication Critical patent/FI884595A/fi
Publication of FI91759B publication Critical patent/FI91759B/fi
Application granted granted Critical
Publication of FI91759C publication Critical patent/FI91759C/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
FI884595A 1987-10-06 1988-10-06 Menetelmä terapeuttisesti käyttökelpoisten imidatso/1,5-a/tieno/3,2-d/- ja -/3,2-e/pyrimidiinien valmistamiseksi FI91759C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK522187A DK522187D0 (da) 1987-10-06 1987-10-06 Imidozothienopyrimidiner, deres fremstilling og anvendelse
DK522187 1987-10-06

Publications (4)

Publication Number Publication Date
FI884595A0 FI884595A0 (fi) 1988-10-06
FI884595A true FI884595A (fi) 1989-04-07
FI91759B FI91759B (fi) 1994-04-29
FI91759C FI91759C (fi) 1994-08-10

Family

ID=8140567

Family Applications (1)

Application Number Title Priority Date Filing Date
FI884595A FI91759C (fi) 1987-10-06 1988-10-06 Menetelmä terapeuttisesti käyttökelpoisten imidatso/1,5-a/tieno/3,2-d/- ja -/3,2-e/pyrimidiinien valmistamiseksi

Country Status (18)

Country Link
US (1) US4866065A (fi)
EP (1) EP0311321B1 (fi)
JP (1) JP2662426B2 (fi)
KR (1) KR0130978B1 (fi)
AT (1) ATE100107T1 (fi)
AU (1) AU611718B2 (fi)
CA (1) CA1323365C (fi)
DE (1) DE3887064T2 (fi)
DK (1) DK522187D0 (fi)
ES (1) ES2061675T3 (fi)
FI (1) FI91759C (fi)
IE (1) IE64931B1 (fi)
IL (1) IL87780A (fi)
NO (1) NO168646C (fi)
NZ (1) NZ226461A (fi)
PH (1) PH25297A (fi)
PT (1) PT88673B (fi)
ZA (1) ZA887313B (fi)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5185446A (en) * 1990-09-04 1993-02-09 Neurogen Corporation Certain cycloalkyl imidazopyrimidines; a new class of gaba brainreceptor ligands
FR2872165B1 (fr) * 2004-06-24 2006-09-22 Sod Conseils Rech Applic Nouveaux derives de pyrimido-benzimidazole
CA2644996A1 (en) * 2006-03-02 2007-09-13 Cv Therapeutics, Inc. A2a adenosine receptor antagonists

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2411274A1 (de) * 1974-03-06 1975-09-18 Schering Ag Neue 2-nitrothieno eckige klammer auf 2,3-d eckige klammer zu pyrimidinon-derivate und verfahren zu ihrer herstellung
CA1142924A (en) * 1980-06-27 1983-03-15 Hoffmann-La Roche Limited Pyrimidine derivatives
GB8432073D0 (en) * 1984-12-19 1985-01-30 Roussel Lab Ltd Chemical compounds
AU587802B2 (en) * 1985-03-08 1989-08-31 Ferrosan A/S Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds
US4622320A (en) * 1985-05-17 1986-11-11 As Ferrosan Oxadiazolylimidazobenzodiazepine, compositions, and method
US4771051A (en) * 1985-05-17 1988-09-13 A/S Ferrosan 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
EP0226282B1 (en) * 1985-10-17 1989-07-05 A/S Ferrosan Heterocyclic compounds and their preparation and use

Also Published As

Publication number Publication date
CA1323365C (en) 1993-10-19
KR0130978B1 (ko) 1998-04-16
FI91759B (fi) 1994-04-29
JP2662426B2 (ja) 1997-10-15
IE882794L (en) 1989-04-06
NO168646C (no) 1992-03-18
IL87780A (en) 1992-02-16
NO884431D0 (no) 1988-10-05
EP0311321B1 (en) 1994-01-12
DE3887064D1 (de) 1994-02-24
FI91759C (fi) 1994-08-10
KR890006653A (ko) 1989-06-15
AU611718B2 (en) 1991-06-20
EP0311321A2 (en) 1989-04-12
ES2061675T3 (es) 1994-12-16
PH25297A (en) 1991-04-30
ZA887313B (en) 1989-06-28
AU2334188A (en) 1989-04-06
NO884431L (no) 1989-04-07
NO168646B (no) 1991-12-09
EP0311321A3 (en) 1990-08-01
ATE100107T1 (de) 1994-01-15
PT88673B (pt) 1992-12-31
NZ226461A (en) 1990-05-28
DE3887064T2 (de) 1994-05-05
IE64931B1 (en) 1995-09-20
US4866065A (en) 1989-09-12
DK522187D0 (da) 1987-10-06
JPH01121291A (ja) 1989-05-12
FI884595A0 (fi) 1988-10-06

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MM Patent lapsed

Owner name: NOVO NORDISK A/S