FI870672A7 - Substituerade tienoimidazolderivat, foerfarande foer deras framstaellning, dessa innehaollande farmaceutiska produkter och deras anvaendning som magsyrasekretionshaemmande aemne. - Google Patents

Substituerade tienoimidazolderivat, foerfarande foer deras framstaellning, dessa innehaollande farmaceutiska produkter och deras anvaendning som magsyrasekretionshaemmande aemne. Download PDF

Info

Publication number
FI870672A7
FI870672A7 FI870672A FI870672A FI870672A7 FI 870672 A7 FI870672 A7 FI 870672A7 FI 870672 A FI870672 A FI 870672A FI 870672 A FI870672 A FI 870672A FI 870672 A7 FI870672 A7 FI 870672A7
Authority
FI
Finland
Prior art keywords
deras
tienoimidazolderivat
magsyrasekretionshaemmande
farmaceutiska
aemne
Prior art date
Application number
FI870672A
Other languages
English (en)
Finnish (fi)
Other versions
FI870672A0 (fi
Inventor
Hans-Jochen Lang
Robert Rippel
Andreas W Herling
Klaus Weidmann
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19863605395 external-priority patent/DE3605395A1/de
Priority claimed from DE19863623683 external-priority patent/DE3623683A1/de
Priority claimed from DE19873700436 external-priority patent/DE3700436A1/de
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of FI870672A0 publication Critical patent/FI870672A0/fi
Publication of FI870672A7 publication Critical patent/FI870672A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI870672A 1986-02-20 1987-02-18 Substituerade tienoimidazolderivat, foerfarande foer deras framstaellning, dessa innehaollande farmaceutiska produkter och deras anvaendning som magsyrasekretionshaemmande aemne. FI870672A7 (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19863605395 DE3605395A1 (de) 1986-02-20 1986-02-20 Substituierte thienoimidazol-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung als magensaeuresekretionshemmer
DE19863623683 DE3623683A1 (de) 1986-07-12 1986-07-12 Substituierte thienoimidazol-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung als magensaeuresekretionshemmer
DE19873700436 DE3700436A1 (de) 1987-01-09 1987-01-09 Substituierte thienoimidazol-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung als magensaeuresekretionshemmer

Publications (2)

Publication Number Publication Date
FI870672A0 FI870672A0 (fi) 1987-02-18
FI870672A7 true FI870672A7 (fi) 1987-08-21

Family

ID=27194035

Family Applications (1)

Application Number Title Priority Date Filing Date
FI870672A FI870672A7 (fi) 1986-02-20 1987-02-18 Substituerade tienoimidazolderivat, foerfarande foer deras framstaellning, dessa innehaollande farmaceutiska produkter och deras anvaendning som magsyrasekretionshaemmande aemne.

Country Status (22)

Country Link
US (1) US4845118A (enrdf_load_stackoverflow)
EP (1) EP0234485B1 (enrdf_load_stackoverflow)
JP (1) JPH0633275B2 (enrdf_load_stackoverflow)
KR (2) KR950001025B1 (enrdf_load_stackoverflow)
CN (1) CN1021911C (enrdf_load_stackoverflow)
AR (1) AR246739A1 (enrdf_load_stackoverflow)
AU (1) AU590390B2 (enrdf_load_stackoverflow)
CA (1) CA1337197C (enrdf_load_stackoverflow)
DE (1) DE3777855D1 (enrdf_load_stackoverflow)
DK (1) DK85087A (enrdf_load_stackoverflow)
EG (1) EG18128A (enrdf_load_stackoverflow)
ES (1) ES2032394T3 (enrdf_load_stackoverflow)
FI (1) FI870672A7 (enrdf_load_stackoverflow)
GR (1) GR3004765T3 (enrdf_load_stackoverflow)
HU (1) HU197330B (enrdf_load_stackoverflow)
IE (1) IE60572B1 (enrdf_load_stackoverflow)
IL (1) IL81609A (enrdf_load_stackoverflow)
MA (1) MA20880A1 (enrdf_load_stackoverflow)
NO (1) NO170155C (enrdf_load_stackoverflow)
NZ (1) NZ219320A (enrdf_load_stackoverflow)
PT (1) PT84319B (enrdf_load_stackoverflow)
TN (1) TNSN87024A1 (enrdf_load_stackoverflow)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI861772A7 (fi) * 1985-05-07 1986-11-08 Chemie Linz Ag Uudet tieno(2,3)imidatsolijohdokset ja menetelmä niiden valmistamiseksi.
CA1256109A (en) * 1986-09-10 1989-06-20 Franz Rovenszky Process for the preparation of derivatives of 4, 5-dihydrooxazoles
US4912101A (en) * 1987-03-13 1990-03-27 Fujirebio Kabushiki Kaisha 4-aminomethyl-pyridyl-2-oxy derivatives having anti-ulcer activity
DE3723327A1 (de) * 1987-07-15 1989-02-02 Hoechst Ag Substituierte thienoimidazol-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung als magensaeuresekretionshemmer, magenschutzmittel sowie als medikament gegen intestinale entzuendungen
AU622866B2 (en) * 1987-07-21 1992-04-30 Hoechst Aktiengesellschaft Substituted thienoimidazole derivatives, processes for their preparation, pharmaceutical formulations containing them and their use as gastric acid secretion inhibitors
IT1222412B (it) * 1987-07-31 1990-09-05 Chiesi Farma Spa Tiometil e sulfinil metil derivati ad azione antisecretiva acida gastrica,loro procedimento di preparazione e composizioni farmaceutiche che li contengono
EP0304732A3 (de) * 1987-08-15 1990-06-13 Hoechst Aktiengesellschaft Substituierte Thienoimidazol-Derivate, Verfahren zu ihrer Herstellung, sie enthaltende pharmazeutische Zubereitungen und ihre Verwendung als Magensäuresekretionshemmer
ATE110078T1 (de) * 1987-11-13 1994-09-15 Hoechst Ag Substituierte thienoimidazol-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung als magensäuresekretionshemmer.
FI885878L (fi) * 1987-12-22 1989-06-23 Hoechst Ag Substituerade tienoimidazolderivat, foerfarande foer deras framstaellning, dessa innehaollande farmaceutiska kompositioner och deras anvaendning som inhibitorer vid avsoendring av magsyra.
US6852739B1 (en) 1999-02-26 2005-02-08 Nitromed Inc. Methods using proton pump inhibitors and nitric oxide donors
SI1187601T1 (sl) 1999-06-07 2005-12-31 Altana Pharma Ag Novi pripravek in dajalna oblika, ki obsega kislinsko labilen inhibitor protonske crpalke
US8048917B2 (en) 2005-04-06 2011-11-01 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
US7232924B2 (en) 2001-06-11 2007-06-19 Xenoport, Inc. Methods for synthesis of acyloxyalkyl derivatives of GABA analogs
US7186855B2 (en) 2001-06-11 2007-03-06 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
US6818787B2 (en) 2001-06-11 2004-11-16 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
US7211590B2 (en) * 2002-08-01 2007-05-01 Nitromed, Inc. Nitrosated proton pump inhibitors, compositions and methods of use
WO2004112756A1 (en) 2003-06-26 2004-12-29 Isa Odidi Proton pump-inhibitor-containing capsules which comprise subunits differently structured for a delayed release of the active ingredient
ATE531361T1 (de) * 2004-05-07 2011-11-15 Nycomed Gmbh Neue pharmazeutische dosierform und herstellungsverfahren
US8394409B2 (en) 2004-07-01 2013-03-12 Intellipharmaceutics Corp. Controlled extended drug release technology
US10624858B2 (en) 2004-08-23 2020-04-21 Intellipharmaceutics Corp Controlled release composition using transition coating, and method of preparing same
US10064828B1 (en) 2005-12-23 2018-09-04 Intellipharmaceutics Corp. Pulsed extended-pulsed and extended-pulsed pulsed drug delivery systems
JP5457830B2 (ja) 2006-04-03 2014-04-02 オディディ,イサ オルガノゾル被膜を含む制御放出送達デバイス
US10960077B2 (en) 2006-05-12 2021-03-30 Intellipharmaceutics Corp. Abuse and alcohol resistant drug composition
EP2486910A3 (en) 2006-10-27 2012-08-22 The Curators Of The University Of Missouri Multi-chambered apparatus comprising a dispenser head
US20080194307A1 (en) * 2007-02-13 2008-08-14 Jeff Sanger Sports-based game of chance
CN101980700A (zh) 2008-02-20 2011-02-23 密苏里大学董事会 包含奥美拉唑和兰索拉唑以及缓冲剂的组合的组合物及其使用方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3132167A1 (de) 1981-08-14 1983-03-03 Hoechst Ag, 6000 Frankfurt "5(6)-phenylsulfonyloxy-benzimidazolderivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung gegen leberegel"
SE416649B (sv) 1974-05-16 1981-01-26 Haessle Ab Forfarande for framstellning av foreningar som paverkar magsyrasekretionen
SE7804231L (sv) 1978-04-14 1979-10-15 Haessle Ab Magsyrasekretionsmedel
US4472409A (en) 1981-11-05 1984-09-18 Byk Gulden Lomberg Chemische Fabrik Gesellschaft Mit Beschrankter Haftung 2-Pyridylmethyl thio(sulfinyl)benzimidazoles with gastric acid secretion inhibiting effects
SE8300736D0 (sv) * 1983-02-11 1983-02-11 Haessle Ab Novel pharmacologically active compounds
US4575554A (en) * 1983-12-05 1986-03-11 The Upjohn Company Substituted 2-pyridylmethylthio- and sulfinyl-benzimidazoles as gastric antisecretory agents
GB8417171D0 (en) * 1984-07-05 1984-08-08 Beecham Group Plc Compounds
AU568441B2 (en) 1984-09-24 1987-12-24 Upjohn Company, The 2-(pyridylalkenesulfinyl) benzimidazole derivatives
FI861772A7 (fi) * 1985-05-07 1986-11-08 Chemie Linz Ag Uudet tieno(2,3)imidatsolijohdokset ja menetelmä niiden valmistamiseksi.
WO1987005296A1 (en) * 1986-03-07 1987-09-11 Pfizer Inc. 2-[(2-pyridyl)methylsulfinyl]thienoimidazoles and related compounds as antiulcer agents

Also Published As

Publication number Publication date
AR246739A1 (es) 1994-09-30
JPH0633275B2 (ja) 1994-05-02
NO870666L (no) 1987-08-21
EP0234485A1 (de) 1987-09-02
IE870421L (en) 1987-08-20
CN87100719A (zh) 1987-09-09
AU6906687A (en) 1987-08-27
CA1337197C (en) 1995-10-03
CN1021911C (zh) 1993-08-25
JPS62198683A (ja) 1987-09-02
GR3004765T3 (enrdf_load_stackoverflow) 1993-04-28
ES2032394T3 (es) 1993-02-16
KR870007934A (ko) 1987-09-23
PT84319B (pt) 1989-09-14
NZ219320A (en) 1990-06-26
TNSN87024A1 (fr) 1990-01-01
AU590390B2 (en) 1989-11-02
HU197330B (en) 1989-03-28
NO870666D0 (no) 1987-02-19
KR950001025B1 (ko) 1995-02-07
DK85087D0 (da) 1987-02-19
FI870672A0 (fi) 1987-02-18
HUT44255A (en) 1988-02-29
IL81609A0 (en) 1987-09-16
EG18128A (en) 1992-08-30
MA20880A1 (fr) 1987-10-01
IE60572B1 (en) 1994-07-27
DK85087A (da) 1987-08-21
NO170155C (no) 1992-09-16
DE3777855D1 (de) 1992-05-07
KR890009937A (ko) 1989-08-05
EP0234485B1 (de) 1992-04-01
IL81609A (en) 1994-10-21
NO170155B (no) 1992-06-09
US4845118A (en) 1989-07-04
PT84319A (de) 1987-03-01

Similar Documents

Publication Publication Date Title
FI870631A7 (fi) Polysackaridderivat, som innehaoller aldehydgrupper, deras framstaellning ur motsvarande acetaler och deras anvaendning som papperstillsatsmedel.
FI891078L (fi) Peptider och antikroppar, som inhiberar plateletadhesion.
FI881560A7 (fi) Vattenhaltiga, biocida, katjoniska plastdispersioner och deras anvaendning som fungicida bakteriocida och algicida slutbehandlingsmedel.
FI870614A7 (fi) Haerdbara blandningar, vilka innehaoller n-sulfonylaminosulfoniumsalter som kationiskt verksamma katalysatorer.
FI870672A7 (fi) Substituerade tienoimidazolderivat, foerfarande foer deras framstaellning, dessa innehaollande farmaceutiska produkter och deras anvaendning som magsyrasekretionshaemmande aemne.
FI874125A0 (fi) Tvaettmedelskompositioner, vilka innehaoller polyalkylenglykol-iminodiaettiksyra som stoedsubstans.
FI883175A7 (fi) Displayfoersett elektroniskt maolspel, som sjaelv raeknar poaeng.
FI872178L (fi) Herbicidtoleranta vaexter, som innehaoller glutation-s-transferasgen.
FI870788L (fi) Vattenhaltiga limaemnesdispersioner som innehaoller polyisocyanat, deras framstaellning och anvaendning.
FI873002A7 (fi) Substituerade hydrazoner, foerfaranden foer deras framstaellning och deras anvaendning som bekaempningsmedel foer skadedjur.
FI871452A0 (fi) Faergloesa ketiminer, deras framstaellning och anvaendning som foernaetningsmedel.
FI863660L (fi) Fosfatloesningar och deras anvaendning som bindemedel.
FI870973A7 (fi) Heteroaryl-oxi- -karbolinderivat, deras framstaellning och deras anvaendning som laekemedel.
FI873999L (fi) Keramiska produkter som innehaoller en polymerkomponent och foerfaranden foer framstaellning av dessa.
FI883699A0 (fi) Foerfarande foer foerbaettring av kvaliteten av vaxhaltiga oljor, med detta foerfarande framstaellda produkter och deras anvaendning som substitut foer laetta braennoljor och dieselbraensle.
FI875359L (fi) Vaermehaerdbara sammansaettningar anvaendbara som b-steg, foerfarande foer deras framstaellning och anvaendning av dessa sammansaettningar.
FI875145A7 (fi) Kondenserade heterocykliska tetrahydroaminokinoliner och beslaektade foereningar, en metod foer deras framstaellning och deras anvaendning som mediciner.
FI875055A7 (fi) Optiskt aktiva gyras-inhibitorer, deras framstaellning och deras anvaendning som antibiotika.
FI875643L (fi) Kemiska foereningar och deras anvaendning som braensletillsatser.
FI863470A7 (fi) 6-fenoximetyl-4 -hydroxitetrahydropyran-2-oner, foerfarande foer deras framstaellning, deras anvaendning som laekemedel farmaceutiska produkter och mellanprodukter.
FI882443A7 (fi) Substituerade vinylkefalosporiner, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.
FI872774A0 (fi) Bensimidazoler, deras framstaellning, formulering och anvaendning som inhibitorer foer magsyraavsoendring.
FI875707A0 (fi) Mycket fyllaemne innehaollande fenolhartsskumplaster och deras anvaendning som isolerformkroppar.
FI875361L (fi) Perestrar, deras framstaellning och anvaendning som polymerisationsinitiatorer.
FI882444A7 (fi) Substituerade vinylkefalosporiner, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.

Legal Events

Date Code Title Description
FA Application withdrawn [patent]

Owner name: HOECHST AKTIENGESELLSCHAFT