FI810255L - Nya 17-amino-16-hydroxisteroider ur androstan- och estranserier och deras derivat foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska kompositioner - Google Patents
Nya 17-amino-16-hydroxisteroider ur androstan- och estranserier och deras derivat foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska kompositionerInfo
- Publication number
- FI810255L FI810255L FI810255A FI810255A FI810255L FI 810255 L FI810255 L FI 810255L FI 810255 A FI810255 A FI 810255A FI 810255 A FI810255 A FI 810255A FI 810255 L FI810255 L FI 810255L
- Authority
- FI
- Finland
- Prior art keywords
- och
- deras
- amino
- hydroxisteroider
- estranserier
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 3
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 3
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000001183 hydrocarbyl group Chemical group 0.000 abstract 2
- QZLYKIGBANMMBK-UGCZWRCOSA-N 5α-Androstane Chemical compound C([C@@H]1CC2)CCC[C@]1(C)[C@@H]1[C@@H]2[C@@H]2CCC[C@@]2(C)CC1 QZLYKIGBANMMBK-UGCZWRCOSA-N 0.000 abstract 1
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 230000003288 anthiarrhythmic effect Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- GRXPVLPQNMUNNX-MHJRRCNVSA-N estrane Chemical class C1CC2CCCC[C@@H]2[C@@H]2[C@@H]1[C@@H]1CCC[C@@]1(C)CC2 GRXPVLPQNMUNNX-MHJRRCNVSA-N 0.000 abstract 1
- 231100000252 nontoxic Toxicity 0.000 abstract 1
- 230000003000 nontoxic effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 150000003431 steroids Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0059—Estrane derivatives substituted in position 17 by a keto group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0062—Estrane derivatives substituted in position 17 alfa not substituted in position 17 beta
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C07J41/0011—Unsubstituted amino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C07J41/0027—Azides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0036—Nitrogen-containing hetero ring
- C07J71/0042—Nitrogen only
- C07J71/0052—Nitrogen only at position 16(17)
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0036—Nitrogen-containing hetero ring
- C07J71/0057—Nitrogen and oxygen
- C07J71/0068—Nitrogen and oxygen at position 16(17)
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Cardiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Heart & Thoracic Surgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8003053 | 1980-01-30 | ||
| GB8003053 | 1980-01-30 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI810255L true FI810255L (fi) | 1981-07-31 |
| FI69631B FI69631B (fi) | 1985-11-29 |
| FI69631C FI69631C (fi) | 1986-03-10 |
Family
ID=10510984
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI810255A FI69631C (fi) | 1980-01-30 | 1981-01-29 | Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 17beta-amino-16alfa-hydroxisteroider av androstan- och estranserier samt av enantiomerer och racemat och farmaceutisktgodtagbara syraadditionssalter av dessa |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP0033561B1 (fi) |
| JP (1) | JPS56120699A (fi) |
| AT (1) | ATE3298T1 (fi) |
| AU (1) | AU542419B2 (fi) |
| CA (1) | CA1167837A (fi) |
| DE (1) | DE3160232D1 (fi) |
| DK (1) | DK163997C (fi) |
| ES (1) | ES498942A0 (fi) |
| FI (1) | FI69631C (fi) |
| GR (1) | GR73137B (fi) |
| HU (1) | HU185441B (fi) |
| IE (1) | IE51100B1 (fi) |
| ZA (1) | ZA81348B (fi) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19917930A1 (de) * | 1999-04-15 | 2000-10-19 | Schering Ag | Ent-Steroide als selektiv wirksame Estrogene |
| WO2002036605A2 (en) | 2000-11-03 | 2002-05-10 | Washington University | Estrone-derivatives having cytoprotective activity |
| JPWO2005026190A1 (ja) * | 2003-09-10 | 2010-02-25 | 学校法人日本大学 | アミノ化環状化合物の製造方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL104598C (fi) * | 1959-07-23 | |||
| GB1439605A (en) * | 1972-07-14 | 1976-06-16 | Akzo Nv | 2beta-hydroxy-3-alpha-amino-steroids and derivatives thereof and the processes for their preparation |
| GB2030569A (en) * | 1978-10-03 | 1980-04-10 | Akzo Nv | Amino hydroxy steroids and derivatives thereof |
-
1981
- 1981-01-19 ZA ZA00810348A patent/ZA81348B/xx unknown
- 1981-01-20 DE DE8181200066T patent/DE3160232D1/de not_active Expired
- 1981-01-20 AT AT81200066T patent/ATE3298T1/de active
- 1981-01-20 EP EP81200066A patent/EP0033561B1/en not_active Expired
- 1981-01-21 IE IE107/81A patent/IE51100B1/en not_active IP Right Cessation
- 1981-01-28 GR GR63992A patent/GR73137B/el unknown
- 1981-01-28 AU AU66649/81A patent/AU542419B2/en not_active Ceased
- 1981-01-29 ES ES498942A patent/ES498942A0/es active Granted
- 1981-01-29 FI FI810255A patent/FI69631C/fi not_active IP Right Cessation
- 1981-01-29 HU HU81201A patent/HU185441B/hu not_active IP Right Cessation
- 1981-01-29 CA CA000369677A patent/CA1167837A/en not_active Expired
- 1981-01-29 JP JP1218781A patent/JPS56120699A/ja active Granted
- 1981-01-29 DK DK039981A patent/DK163997C/da not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| EP0033561A1 (en) | 1981-08-12 |
| FI69631C (fi) | 1986-03-10 |
| ES8300788A1 (es) | 1982-11-16 |
| ZA81348B (en) | 1982-02-24 |
| DK163997C (da) | 1992-09-21 |
| DE3160232D1 (en) | 1983-06-16 |
| EP0033561B1 (en) | 1983-05-11 |
| ATE3298T1 (de) | 1983-05-15 |
| HU185441B (en) | 1985-02-28 |
| AU542419B2 (en) | 1985-02-21 |
| JPH0115518B2 (fi) | 1989-03-17 |
| IE51100B1 (en) | 1986-10-01 |
| DK163997B (da) | 1992-04-27 |
| CA1167837A (en) | 1984-05-22 |
| JPS56120699A (en) | 1981-09-22 |
| AU6664981A (en) | 1981-08-06 |
| DK39981A (da) | 1981-07-31 |
| GR73137B (fi) | 1984-02-07 |
| ES498942A0 (es) | 1982-11-16 |
| IE810107L (en) | 1981-07-30 |
| FI69631B (fi) | 1985-11-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM | Patent lapsed | ||
| MM | Patent lapsed |
Owner name: AKZO N.V. |