FI791562A - Foerfarande foer framstaellning av 4-amino-2-piperidinokinazolinderivat - Google Patents

Foerfarande foer framstaellning av 4-amino-2-piperidinokinazolinderivat

Info

Publication number
FI791562A
FI791562A FI791562A FI791562A FI791562A FI 791562 A FI791562 A FI 791562A FI 791562 A FI791562 A FI 791562A FI 791562 A FI791562 A FI 791562A FI 791562 A FI791562 A FI 791562A
Authority
FI
Finland
Prior art keywords
piperidinokinazoline
framstation
derivatives
amino
procedure
Prior art date
Application number
FI791562A
Other languages
English (en)
Other versions
FI64589C (fi
FI64589B (fi
Inventor
Simon Fraser Campbell
John Christopher Danilewicz
Colin William Greengrass
Rhona Plews
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI791562A publication Critical patent/FI791562A/fi
Application granted granted Critical
Publication of FI64589B publication Critical patent/FI64589B/fi
Publication of FI64589C publication Critical patent/FI64589C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D211/62Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/46Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
FI791562A 1978-05-18 1979-05-16 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 4-amino-2-piperidinokinazolinderivat FI64589C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB2035178 1978-05-18
GB2035178 1978-05-18

Publications (3)

Publication Number Publication Date
FI791562A true FI791562A (fi) 1979-11-19
FI64589B FI64589B (fi) 1983-08-31
FI64589C FI64589C (fi) 1983-12-12

Family

ID=10144517

Family Applications (1)

Application Number Title Priority Date Filing Date
FI791562A FI64589C (fi) 1978-05-18 1979-05-16 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 4-amino-2-piperidinokinazolinderivat

Country Status (30)

Country Link
US (1) US4243666A (fi)
JP (1) JPS554370A (fi)
AR (2) AR223487A1 (fi)
AT (1) ATA363379A (fi)
AU (1) AU512947B2 (fi)
BE (1) BE876297A (fi)
CA (1) CA1240325A (fi)
CH (1) CH643553A5 (fi)
CS (1) CS214796B2 (fi)
DD (1) DD143613A5 (fi)
DE (1) DE2919800A1 (fi)
DK (1) DK159079A (fi)
ES (2) ES480671A1 (fi)
FI (1) FI64589C (fi)
FR (1) FR2434162A1 (fi)
GR (1) GR72824B (fi)
HU (1) HU182562B (fi)
IL (1) IL57297A (fi)
IN (1) IN153045B (fi)
IT (1) IT1114222B (fi)
LU (1) LU81284A1 (fi)
NL (1) NL172157C (fi)
NO (1) NO791648L (fi)
NZ (1) NZ190465A (fi)
PH (1) PH14802A (fi)
PL (2) PL121158B1 (fi)
PT (1) PT69622A (fi)
SE (1) SE439306B (fi)
YU (2) YU115279A (fi)
ZA (1) ZA792390B (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4607034A (en) * 1979-10-29 1986-08-19 Mitsubishi Yuka Pharmaceutical Co., Ltd. Quinazoline derivatives and pharmaceutical composition thereof
JPS5962766U (ja) * 1982-06-30 1984-04-25 守田 智 小動物用給水器
GB8414518D0 (en) * 1984-06-07 1984-07-11 Pfizer Ltd Therapeutic agents
US5801195A (en) * 1994-12-30 1998-09-01 Celgene Corporation Immunotherapeutic aryl amides
US6248888B1 (en) 1997-11-14 2001-06-19 Teva Pharmaceutical Industries Ltd. Process for the preparation of terazosin hydrochloride dihydrate
WO2002057235A1 (fr) * 2001-01-18 2002-07-25 Takeda Chemical Industries, Ltd. Procede de preparation de composes de benzylpiperidine
US6746460B2 (en) * 2002-08-07 2004-06-08 Satiety, Inc. Intra-gastric fastening devices
JP2007510642A (ja) * 2003-11-03 2007-04-26 ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー 中枢神経系障害の治療のための新規ノルエピネフリン再取込み阻害薬
WO2008045564A2 (en) * 2006-10-12 2008-04-17 Epix Delaware, Inc. Carboxamide compounds and their use as antagonists of the chemokine ccr2 receptor
KR101441930B1 (ko) * 2007-04-04 2014-09-19 시플라 리미티드 에르로티닙 및 그의 약학적으로 허용가능한 염의 제조방법
EP2280766A1 (en) * 2007-12-11 2011-02-09 CytoPathfinder, Inc. Carboxamide compounds and their use as chemokine receptor agonists
BRPI0922010A2 (pt) * 2008-11-14 2015-12-15 Hoffmann La Roche dervivados de quinazolina como antagonistas receptores de nk3

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1156973A (en) * 1965-07-06 1969-07-02 Quinazoline Derivatives
US3511836A (en) * 1967-12-13 1970-05-12 Pfizer & Co C 2,4,6,7-tetra substituted quinazolines
FR2321890A1 (fr) * 1975-08-26 1977-03-25 Synthelabo Nouveaux derives de la quinazoline, leurs sels, leur preparation et les medicaments qui en renferment
DK140695C (da) * 1976-05-07 1980-05-12 Synthelabo Analogifremgangsmaade til fremstilling af 2,4-diamino-6,7-dimethoxyquinazolinderivater eller syreadditionssalte heraf

Also Published As

Publication number Publication date
NO791648L (no) 1979-11-20
ES488210A0 (es) 1980-12-16
CS214796B2 (en) 1982-05-28
PL215626A1 (fi) 1980-08-25
PL121158B1 (en) 1982-04-30
IN153045B (fi) 1984-05-26
YU256382A (en) 1983-04-30
SE439306B (sv) 1985-06-10
ZA792390B (en) 1980-07-30
LU81284A1 (fr) 1980-12-16
JPS5623992B2 (fi) 1981-06-03
AR224784A1 (es) 1982-01-15
FI64589C (fi) 1983-12-12
BE876297A (fr) 1979-11-16
IL57297A0 (en) 1979-09-30
SE7904358L (sv) 1979-11-19
NZ190465A (en) 1981-05-01
IT1114222B (it) 1986-01-27
JPS554370A (en) 1980-01-12
AR223487A1 (es) 1981-08-31
AU512947B2 (en) 1980-11-06
PL223844A1 (fi) 1981-01-02
IL57297A (en) 1983-02-23
PL120651B1 (en) 1982-03-31
PH14802A (en) 1981-12-14
NL7903853A (nl) 1979-11-20
IT7922720A0 (it) 1979-05-16
FI64589B (fi) 1983-08-31
HU182562B (en) 1984-02-28
DD143613A5 (de) 1980-09-03
AU4710179A (en) 1979-11-22
ES8101584A1 (es) 1980-12-16
FR2434162B1 (fi) 1983-04-22
FR2434162A1 (fr) 1980-03-21
YU115279A (en) 1983-04-30
DE2919800A1 (de) 1979-11-22
GR72824B (fi) 1983-12-06
US4243666A (en) 1981-01-06
ES480671A1 (es) 1980-08-16
DK159079A (da) 1979-11-19
CH643553A5 (de) 1984-06-15
ATA363379A (de) 1983-05-15
CA1240325A (en) 1988-08-09
PT69622A (en) 1979-06-01
NL172157C (nl) 1983-07-18
NL172157B (nl) 1983-02-16

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: PFIZER CORPORATION