FI61885C - Foerfarande foer framstaellning av terapeutiskt aktiva 5-fluoropyrimidin-4-onderivat - Google Patents

Foerfarande foer framstaellning av terapeutiskt aktiva 5-fluoropyrimidin-4-onderivat Download PDF

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Publication number
FI61885C
FI61885C FI762166A FI762166A FI61885C FI 61885 C FI61885 C FI 61885C FI 762166 A FI762166 A FI 762166A FI 762166 A FI762166 A FI 762166A FI 61885 C FI61885 C FI 61885C
Authority
FI
Finland
Prior art keywords
fluoropyrimidin
formula
fluorouracil
fluoropyrimidine
mixture
Prior art date
Application number
FI762166A
Other languages
English (en)
Finnish (fi)
Other versions
FI61885B (fi
FI762166A (da
Inventor
Mitugi Yasumoto
Junichi Yamashita
Ichiro Yamawaki
Norio Unemi
Kenji Kitazato
Sadao Hashimoto
Setsuro Fujii
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP15093775A external-priority patent/JPS6011033B2/ja
Priority claimed from JP50150936A external-priority patent/JPS6011032B2/ja
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Publication of FI762166A publication Critical patent/FI762166A/fi
Publication of FI61885B publication Critical patent/FI61885B/fi
Application granted granted Critical
Publication of FI61885C publication Critical patent/FI61885C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI762166A 1975-12-16 1976-07-28 Foerfarande foer framstaellning av terapeutiskt aktiva 5-fluoropyrimidin-4-onderivat FI61885C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP15093675 1975-12-16
JP15093775A JPS6011033B2 (ja) 1975-12-16 1975-12-16 ５‐フルオルピリミジン―４―オン誘導体の製造法
JP15093775 1975-12-16
JP50150936A JPS6011032B2 (ja) 1975-12-16 1975-12-16 ２―置換―５―フルオルピリミジン―４―オン誘導体の製造法

Publications (3)

Publication Number Publication Date
FI762166A FI762166A (da) 1977-06-17
FI61885B FI61885B (fi) 1982-06-30
FI61885C true FI61885C (fi) 1982-10-11

Family

ID=26480366

Family Applications (1)

Application Number Title Priority Date Filing Date
FI762166A FI61885C (fi) 1975-12-16 1976-07-28 Foerfarande foer framstaellning av terapeutiskt aktiva 5-fluoropyrimidin-4-onderivat

Country Status (12)

Country Link
US (1) US4080455A (da)
AU (1) AU505440B2 (da)
CA (1) CA1063606A (da)
CH (2) CH621544A5 (da)
DE (1) DE2633359C3 (da)
DK (1) DK137957B (da)
FI (1) FI61885C (da)
FR (1) FR2335228A1 (da)
GB (1) GB1501537A (da)
NL (1) NL162643C (da)
NO (1) NO143903C (da)
SE (1) SE439159B (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GR68935B (da) * 1976-03-31 1982-03-29 Takeda Chemical Industries Ltd
JPS5446791A (en) * 1977-09-22 1979-04-12 Takeda Chem Ind Ltd Fluorouracil derivative
US4343940A (en) * 1979-02-13 1982-08-10 Mead Johnson & Company Anti-tumor quinazoline compounds
WO2008033466A2 (en) * 2006-09-14 2008-03-20 Combinatorx (Singapore) Pre. Ltd. Compositions and methods for treatment of viral diseases
CN102532039B (zh) * 2010-09-29 2014-03-26 浙江工业大学 一种5-氟嘧啶-4(3h)-酮类化合物在制备抗肿瘤药物中的应用
CN101955465B (zh) * 2010-09-29 2012-07-04 浙江工业大学 一种5-氟嘧啶-4(3h)-酮类化合物及其制备方法和应用
CN102659689B (zh) * 2012-05-16 2014-12-17 浙江工业大学 4-取代-2-丁氧基-5-氟嘧啶类化合物及其制备方法和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2802005A (en) * 1957-08-06 S-eluorourace
US3784693A (en) * 1972-10-18 1974-01-08 Sandoz Ag 3-substituted phenyl-quinazoline-4(3h)-ones as sedative hypnotics
CH579057A5 (da) * 1973-09-07 1976-08-31 Hoffmann La Roche

Also Published As

Publication number Publication date
FI61885B (fi) 1982-06-30
DE2633359B2 (de) 1980-12-04
NL162643C (nl) 1980-06-16
CH621544A5 (da) 1981-02-13
NO143903C (no) 1981-05-06
NO143903B (no) 1981-01-26
DK137957B (da) 1978-06-12
GB1501537A (en) 1978-02-15
FI762166A (da) 1977-06-17
SE439159B (sv) 1985-06-03
DK137957C (da) 1978-11-06
CA1063606A (en) 1979-10-02
NL7608537A (nl) 1977-06-20
NL162643B (nl) 1980-01-15
DK346176A (da) 1977-06-17
FR2335228A1 (fr) 1977-07-15
FR2335228B1 (da) 1978-11-17
DE2633359A1 (de) 1977-06-30
CH625230A5 (da) 1981-09-15
NO762664L (da) 1977-06-17
AU505440B2 (en) 1979-11-22
SE7608306L (sv) 1977-06-17
AU1547576A (en) 1978-01-05
DE2633359C3 (de) 1981-12-17
US4080455A (en) 1978-03-21

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Owner name: TAIHO PHARMACEUTICAL COMPANY, LIMITED