FI3539540T3 - Sglt2:n estäjä 1-kloori-4-(beta-d-glukopyranos-1-yyli)-2-[4-((s)-tetrahydrofuran-3-yylioksi)bentsyyli]bentseeni yhdessä insuliinin kanssa käytettäväksi menetelmässä hypoglykemiariskin vähentämiseksi - Google Patents

Sglt2:n estäjä 1-kloori-4-(beta-d-glukopyranos-1-yyli)-2-[4-((s)-tetrahydrofuran-3-yylioksi)bentsyyli]bentseeni yhdessä insuliinin kanssa käytettäväksi menetelmässä hypoglykemiariskin vähentämiseksi Download PDF

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Publication number
FI3539540T3
FI3539540T3 FIEP19163940.0T FI19163940T FI3539540T3 FI 3539540 T3 FI3539540 T3 FI 3539540T3 FI 19163940 T FI19163940 T FI 19163940T FI 3539540 T3 FI3539540 T3 FI 3539540T3
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Finland
Prior art keywords
insulin
sglt2 inhibitor
use according
patient
group
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FIEP19163940.0T
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English (en)
Finnish (fi)
Inventor
Rolf Grempler
Odd-Erik Johansen
Thomas Klein
Gerd Luippold
Michael Mark
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Boehringer Ingelheim Int
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44906182&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI3539540(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
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Publication of FI3539540T3 publication Critical patent/FI3539540T3/fi

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    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
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FIEP19163940.0T 2010-11-08 2011-11-07 Sglt2:n estäjä 1-kloori-4-(beta-d-glukopyranos-1-yyli)-2-[4-((s)-tetrahydrofuran-3-yylioksi)bentsyyli]bentseeni yhdessä insuliinin kanssa käytettäväksi menetelmässä hypoglykemiariskin vähentämiseksi FI3539540T3 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP10190303 2010-11-08
EP11151059 2011-01-17

Publications (1)

Publication Number Publication Date
FI3539540T3 true FI3539540T3 (fi) 2025-01-21

Family

ID=44906182

Family Applications (1)

Application Number Title Priority Date Filing Date
FIEP19163940.0T FI3539540T3 (fi) 2010-11-08 2011-11-07 Sglt2:n estäjä 1-kloori-4-(beta-d-glukopyranos-1-yyli)-2-[4-((s)-tetrahydrofuran-3-yylioksi)bentsyyli]bentseeni yhdessä insuliinin kanssa käytettäväksi menetelmässä hypoglykemiariskin vähentämiseksi

Country Status (31)

Country Link
US (6) US20120283169A1 (enExample)
EP (2) EP3539540B1 (enExample)
JP (3) JP2013541576A (enExample)
KR (3) KR20130125365A (enExample)
CN (2) CN106177957A (enExample)
AP (1) AP2013006813A0 (enExample)
AR (1) AR083787A1 (enExample)
AU (1) AU2011328231B2 (enExample)
BR (1) BR112013011968A2 (enExample)
CA (1) CA2813661C (enExample)
CL (1) CL2013001104A1 (enExample)
CO (1) CO6781465A2 (enExample)
DK (1) DK3539540T3 (enExample)
EA (1) EA026712B1 (enExample)
EC (1) ECSP13012661A (enExample)
ES (1) ES3012504T3 (enExample)
FI (1) FI3539540T3 (enExample)
HR (1) HRP20250096T1 (enExample)
HU (1) HUE070541T2 (enExample)
IL (1) IL225597A0 (enExample)
LT (1) LT3539540T (enExample)
MA (1) MA34640B1 (enExample)
MX (2) MX374694B (enExample)
NZ (1) NZ608829A (enExample)
PE (1) PE20140244A1 (enExample)
PH (2) PH12013500809A1 (enExample)
PL (1) PL3539540T3 (enExample)
RS (1) RS66479B1 (enExample)
SG (1) SG189249A1 (enExample)
SI (1) SI3539540T1 (enExample)
WO (1) WO2012062698A1 (enExample)

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US7772191B2 (en) 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
PE20080697A1 (es) 2006-05-03 2008-08-05 Boehringer Ingelheim Int Derivados de benzonitrilo sustituidos con glucopiranosilo, composiciones farmaceuticas que contienen compuestos de este tipo, su uso y procedimiento para su fabricacion
PE20090938A1 (es) 2007-08-16 2009-08-08 Boehringer Ingelheim Int Composicion farmaceutica que comprende un derivado de benceno sustituido con glucopiranosilo
LT2395983T (lt) 2009-02-13 2020-07-10 Boehringer Ingelheim International Gmbh Farmacinė kompozicija, apimanti sglt2 inhibitorių, dpp-iv inhibitorių ir, pasirinktinai, papildomą priešdiabetinį agentą, bei jos panaudojimas
PH12012500633B1 (en) 2009-09-30 2017-12-13 Boehringer Ingelheim Int Method for the preparation of a crystalline form of 1-chloro -4- (beta -d- glucopyranos -1-yl) -2- (4-((s)- tetrahydrofuran -3- yloxy) benzyl) benzene
WO2011039108A2 (en) 2009-09-30 2011-04-07 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives
UY32919A (es) 2009-10-02 2011-04-29 Boehringer Ingelheim Int Composición farmacéutica, forma de dosificación farmacéutica, procedimiento para su preparación, mé todos para su tratamiento y sus usos
US20120283169A1 (en) 2010-11-08 2012-11-08 Boehringer Ingelheim International Gmbh Pharmaceutical composition, methods for treating and uses thereof
UY33937A (es) 2011-03-07 2012-09-28 Boehringer Ingelheim Int Composiciones farmacéuticas que contienen inhibidores de dpp-4 y/o sglt-2 y metformina
US9555001B2 (en) 2012-03-07 2017-01-31 Boehringer Ingelheim International Gmbh Pharmaceutical composition and uses thereof
US9192617B2 (en) 2012-03-20 2015-11-24 Boehringer Ingelheim International Gmbh Pharmaceutical composition, methods for treating and uses thereof
WO2014161836A1 (en) 2013-04-04 2014-10-09 Boehringer Ingelheim Vetmedica Gmbh Treatment of metabolic disorders in equine animals
PT2981271T (pt) 2013-04-05 2019-02-19 Boehringer Ingelheim Int Utilizações terapêuticas de empagliflozina
HK1213818A1 (zh) 2013-04-05 2016-07-15 勃林格殷格翰国际有限公司 依帕列净的治疗用途
CA2812519A1 (en) 2013-04-05 2014-10-05 Boehringer Ingelheim International Gmbh Pharmaceutical composition, methods for treating and uses thereof
CA2812016A1 (en) * 2013-04-05 2014-10-05 Boehringer Ingelheim International Gmbh Pharmaceutical composition, methods for treating and uses thereof
US11813275B2 (en) 2013-04-05 2023-11-14 Boehringer Ingelheim International Gmbh Pharmaceutical composition, methods for treating and uses thereof
EA033286B1 (ru) 2013-04-18 2019-09-30 Бёрингер Ингельхайм Интернациональ Гмбх Способ лечения или отсрочки развития хронической болезни почек
CN105828815B (zh) * 2013-12-17 2020-03-27 勃林格殷格翰动物保健有限公司 猫科动物中代谢紊乱的治疗
ES2951127T3 (es) 2014-01-23 2023-10-18 Boehringer Ingelheim Vetmedica Gmbh Inhibidores de SGLT2 para el tratamiento de trastornos metabólicos en animales caninos
AU2015239655B2 (en) 2014-04-01 2019-10-24 Boehringer Ingelheim Vetmedica Gmbh Treatment of metabolic disorders in equine animals
NZ728804A (en) 2014-09-25 2022-10-28 Boehringer Ingelheim Vetmedica Gmbh Combination treatment of sglt2 inhibitors and dopamine agonists for preventing metabolic disorders in equine animals
CN104473920A (zh) * 2014-12-20 2015-04-01 长沙佰顺生物科技有限公司 一种用于治疗2型糖尿病的复方制剂及其制备方法
RS66325B1 (sr) 2015-08-27 2025-01-31 Boehringer Ingelheim Vetmedica Gmbh Tečne farmaceutske kompozicije koje obuhvataju inhibitore sglt 2
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