ES8406415A1 - Procedimiento analogo para preparar acido (r,s)-5-amino-hepta-5,6-dienoico,acido (s)-4-amino-hepta-5,6-dienoico o sus sales farmaceuticamente aceptables. - Google Patents
Procedimiento analogo para preparar acido (r,s)-5-amino-hepta-5,6-dienoico,acido (s)-4-amino-hepta-5,6-dienoico o sus sales farmaceuticamente aceptables.Info
- Publication number
- ES8406415A1 ES8406415A1 ES522436A ES522436A ES8406415A1 ES 8406415 A1 ES8406415 A1 ES 8406415A1 ES 522436 A ES522436 A ES 522436A ES 522436 A ES522436 A ES 522436A ES 8406415 A1 ES8406415 A1 ES 8406415A1
- Authority
- ES
- Spain
- Prior art keywords
- aminoalkadiene
- derivative
- hepta
- gaba
- gamma
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/30—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and unsaturated
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
- C07C227/16—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions not involving the amino or carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/30—Preparation of optical isomers
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Saccharide Compounds (AREA)
- Pyrrole Compounds (AREA)
Abstract
PROCEDIMIENTO ANALOGO PARA PREPARAR ACIDO (R,S)-5-AMINO-HEPTA-5,6-DIENOICO, ACIDO (S)-4-AMINO-HEPTA-5,6-DIENOICO O SUS SALES FARMACEUTICAMENTE ACEPTABLES.SE CONVIERTE EL GRUPO ETIXILO DE UN DERIVADO AMINO-PROTEGIDO DE UN COMPUESTO DE (S)-O (R,S)-AMINOALQUILO DE FORMULA I, EN UN GRUPO ALENILO. DICHA TRANSFORMACION TIENE LUGAR CALENTANDO EL DERIVADO CON FORMALDEIDO Y UNA AMINA SECUNDARIA TENIENDO UN ATOMO DE HIDROGENO SOBRE EL ATOMO BAB-CARBONO, EN UN DISOLVENTE ORGANICO Y EN PRESENCIA DE UNA SAL INORGANICA.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8214290 | 1982-05-17 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8406415A1 true ES8406415A1 (es) | 1984-08-16 |
| ES522436A0 ES522436A0 (es) | 1984-08-16 |
Family
ID=10530399
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES522436A Granted ES522436A0 (es) | 1982-05-17 | 1983-05-16 | Procedimiento analogo para preparar acido (r,s)-5-amino-hepta-5,6-dienoico,acido (s)-4-amino-hepta-5,6-dienoico o sus sales farmaceuticamente aceptables. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4454156A (es) |
| EP (1) | EP0094886B1 (es) |
| JP (1) | JPS58208255A (es) |
| KR (1) | KR900006127B1 (es) |
| AT (1) | ATE14216T1 (es) |
| AU (1) | AU555635B2 (es) |
| CA (1) | CA1196656A (es) |
| DE (1) | DE3360386D1 (es) |
| DK (1) | DK164661C (es) |
| ES (1) | ES522436A0 (es) |
| GB (1) | GB2120244B (es) |
| GR (1) | GR77487B (es) |
| IE (1) | IE54819B1 (es) |
| IL (1) | IL68525A (es) |
| NO (1) | NO164021C (es) |
| NZ (1) | NZ204017A (es) |
| PH (1) | PH22652A (es) |
| ZA (1) | ZA833012B (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8311804D0 (en) * | 1983-04-29 | 1983-06-02 | Merrell Toraude & Co | Treatment of seizure disorders and pharmaceutical compositions |
| NO842759L (no) * | 1983-07-07 | 1985-01-08 | Syntex Inc | Fremgangsmaate ved fremstilling av nye, terapeutisk virksomme gamma-allenyl-gamma-aminosmoersyrer |
| US4668703A (en) * | 1983-07-07 | 1987-05-26 | Syntex (U.S.A.) Inc. | γ-allenyl-γ-aminobutyric acids |
| ES535188A0 (es) * | 1983-08-17 | 1985-12-01 | Syntex Inc | Procedimiento para la preparacion de alfa-aminoacidos alfa-alenicos |
| JPS62148462A (ja) * | 1985-12-19 | 1987-07-02 | メレルダウフア−マス−テイカルズ インコ−ポレ−テツド | 原生動物の生長を抑制する新規な方法 |
| US5196450A (en) * | 1985-12-19 | 1993-03-23 | Merrell Dow Pharmaceuticals Inc. | Method of inhibiting protozoal growth |
| IL100360A (en) * | 1990-12-17 | 1998-08-16 | Merrell Dow Pharma | HISTORY OF PYROLIDINONE USED AS SUBSTANCE (S) -Vinyl and Alanyl GABA |
| US5208345A (en) * | 1990-12-17 | 1993-05-04 | Merrell Dow Pharmaceuticals Inc. | Process for the production of (S)-vinyl and allenyl gaba |
| US5316944A (en) * | 1992-07-17 | 1994-05-31 | Merrell Dow Pharmaceuticals | Enzymatic resolution of a racemic mixture of gamma-amino acids using penicillin acylase |
| WO1995000470A1 (en) * | 1993-06-23 | 1995-01-05 | Merrell Pharmaceuticals Inc. | Novel processes for preparing (s)-4-amino-hepta-5,6-dienoic acid and intermediates thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3960927A (en) * | 1975-03-18 | 1976-06-01 | Richardson-Merrell Inc. | Olefinic derivatives of amino acids |
| US4326071A (en) * | 1977-09-28 | 1982-04-20 | Merrell Toraude Et Compagnie | Halomethyl derivatives of gamma-aminobutyric acid and related compounds |
| US4178463A (en) * | 1978-01-30 | 1979-12-11 | Merrell Toraude Et Compagnie | Process for making 4-aminohex-5-enoic acid |
-
1983
- 1983-04-25 GB GB08311234A patent/GB2120244B/en not_active Expired
- 1983-04-26 IE IE960/83A patent/IE54819B1/en not_active IP Right Cessation
- 1983-04-27 NZ NZ204017A patent/NZ204017A/en unknown
- 1983-04-28 ZA ZA833012A patent/ZA833012B/xx unknown
- 1983-04-28 CA CA000426934A patent/CA1196656A/en not_active Expired
- 1983-04-29 IL IL68525A patent/IL68525A/xx not_active IP Right Cessation
- 1983-04-29 PH PH28830A patent/PH22652A/en unknown
- 1983-05-04 AU AU14230/83A patent/AU555635B2/en not_active Expired
- 1983-05-09 US US06/492,986 patent/US4454156A/en not_active Expired - Lifetime
- 1983-05-13 EP EP83400973A patent/EP0094886B1/en not_active Expired
- 1983-05-13 AT AT83400973T patent/ATE14216T1/de not_active IP Right Cessation
- 1983-05-13 DE DE8383400973T patent/DE3360386D1/de not_active Expired
- 1983-05-16 NO NO831743A patent/NO164021C/no not_active IP Right Cessation
- 1983-05-16 KR KR1019830002131A patent/KR900006127B1/ko not_active IP Right Cessation
- 1983-05-16 ES ES522436A patent/ES522436A0/es active Granted
- 1983-05-16 DK DK218083A patent/DK164661C/da not_active IP Right Cessation
- 1983-05-16 JP JP58084290A patent/JPS58208255A/ja active Granted
- 1983-05-17 GR GR71366A patent/GR77487B/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL68525A0 (en) | 1983-07-31 |
| PH22652A (en) | 1988-10-28 |
| CA1196656A (en) | 1985-11-12 |
| IL68525A (en) | 1986-07-31 |
| GB2120244B (en) | 1985-05-01 |
| DE3360386D1 (de) | 1985-08-14 |
| DK164661C (da) | 1992-12-14 |
| EP0094886B1 (en) | 1985-07-10 |
| DK218083A (da) | 1983-11-18 |
| KR900006127B1 (ko) | 1990-08-24 |
| DK218083D0 (da) | 1983-05-16 |
| NZ204017A (en) | 1985-03-20 |
| IE54819B1 (en) | 1990-02-14 |
| AU555635B2 (en) | 1986-10-02 |
| IE830960L (en) | 1983-11-17 |
| JPH0465056B2 (es) | 1992-10-16 |
| GB2120244A (en) | 1983-11-30 |
| DK164661B (da) | 1992-07-27 |
| EP0094886A1 (en) | 1983-11-23 |
| JPS58208255A (ja) | 1983-12-03 |
| GB8311234D0 (en) | 1983-06-02 |
| GR77487B (es) | 1984-09-24 |
| NO831743L (no) | 1983-11-18 |
| AU1423083A (en) | 1983-11-24 |
| NO164021C (no) | 1990-08-22 |
| ZA833012B (en) | 1984-01-25 |
| US4454156A (en) | 1984-06-12 |
| KR840005070A (ko) | 1984-11-03 |
| ES522436A0 (es) | 1984-08-16 |
| ATE14216T1 (de) | 1985-07-15 |
| NO164021B (no) | 1990-05-14 |
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