ES8304798A1 - Un procedimiento para la preparacion de una composicion de 4-amino-n-(5-metil-3-isoxazowil)benzenosulfonamida-5(3,4,5- trimetoxifenil)metil(2,4-pirimidinodamina. - Google Patents
Un procedimiento para la preparacion de una composicion de 4-amino-n-(5-metil-3-isoxazowil)benzenosulfonamida-5(3,4,5- trimetoxifenil)metil(2,4-pirimidinodamina.Info
- Publication number
- ES8304798A1 ES8304798A1 ES508351A ES508351A ES8304798A1 ES 8304798 A1 ES8304798 A1 ES 8304798A1 ES 508351 A ES508351 A ES 508351A ES 508351 A ES508351 A ES 508351A ES 8304798 A1 ES8304798 A1 ES 8304798A1
- Authority
- ES
- Spain
- Prior art keywords
- composition
- coelomic
- administration
- trimethoprim
- ingredients
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/683—Diesters of a phosphorus acid with two hydroxy compounds, e.g. phosphatidylinositols
- A61K31/685—Diesters of a phosphorus acid with two hydroxy compounds, e.g. phosphatidylinositols one of the hydroxy compounds having nitrogen atoms, e.g. phosphatidylserine, lecithin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
- A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE COMPOSICIONES DE 4-AMINO-N-(5-METIL-3-ISOXAZOLIL)BENCENOSULFONAMIDA/ 5- (3,4,5-TRIMETOXIFENIL)METIL -2,4-PIRIMIDINDIAMINA, QUE TIENE APLICACIONES FARMACOLOGICAS PARA LA ADMINISTRACION CELOMICA DE AGENTES ANTIMICROBIANOS. CONSISTE EN MEZCLAR 4-AMINO-N-(5-METIL-3-ISOXAZOLIL)BENCENOSULFONAMIDA Y 5- (3,4,5-TRIMETOXIFENIL)METIL -2,4-PIRIMIDINDIAMINA EN PROPORCIONES ADECUADAS CON UN FOSFOLIPIDO, EN PROPORCION DE 0,5-5%, EN CALIENTE Y CON AGITACION HASTA CONSEGUIR UNA DISPERSION UNIFORME, Y A CONTINUACION MOLDEAR LA DISPERSION OBTENIDA.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP55185780A JPS57109713A (en) | 1980-12-26 | 1980-12-26 | Pharmaceutical preparation of combined agent of sulfamethoxazole and trimethoprim for medication through celom |
Publications (2)
Publication Number | Publication Date |
---|---|
ES508351A0 ES508351A0 (es) | 1983-03-16 |
ES8304798A1 true ES8304798A1 (es) | 1983-03-16 |
Family
ID=16176757
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES508351A Expired ES8304798A1 (es) | 1980-12-26 | 1981-12-24 | Un procedimiento para la preparacion de una composicion de 4-amino-n-(5-metil-3-isoxazowil)benzenosulfonamida-5(3,4,5- trimetoxifenil)metil(2,4-pirimidinodamina. |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP0055609A1 (es) |
JP (1) | JPS57109713A (es) |
AU (1) | AU546228B2 (es) |
ES (1) | ES8304798A1 (es) |
GB (1) | GB2090138A (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5946223A (ja) * | 1982-08-30 | 1984-03-15 | Daito Koeki Kk | 抗菌性組成物 |
US4699776A (en) * | 1985-06-28 | 1987-10-13 | R. P. Scherer Corporation | Suppositories containing analgesics, antipyretics or anti-inflammatory agents |
HU210693B (en) * | 1991-10-11 | 1995-06-28 | Egyt Gyogyszervegyeszeti Gyar | Process for producing pharmaceutical compositions for injections without tissue damages, containing sulfamethoxazol and trimetoprime |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE667500C (de) * | 1934-09-28 | 1938-11-14 | Chemisch Pharmazeutische A G B | Verfahren zur Herstellung von Grundmassen fuer Arzneistoffe zur Einfuehrung in Koerperhoehlen |
US3485840A (en) * | 1964-11-12 | 1969-12-23 | Hoffmann La Roche | 2,4-diamino - 5 - (2',4',5'-substituted benzyl) pyrimidines,intermediates and processes |
IT1043853B (it) * | 1973-04-19 | 1980-02-29 | Chiesi P | Supposte contenenti l associazione trimetoprim sulfametossazolo e metodo per ottenerle |
JPS55102517A (en) * | 1979-01-30 | 1980-08-05 | Shionogi & Co Ltd | Preparation of sulfamethoxazole-trimethoprim complex for administration via body cavity |
DE2951142C2 (de) * | 1979-12-19 | 1983-11-03 | A. Nattermann & Cie GmbH, 5000 Köln | Suppositorium-Zubereitung von Indometacin oder Acemetacin |
-
1980
- 1980-12-26 JP JP55185780A patent/JPS57109713A/ja active Granted
-
1981
- 1981-12-23 AU AU78801/81A patent/AU546228B2/en not_active Expired
- 1981-12-23 EP EP81306107A patent/EP0055609A1/en not_active Withdrawn
- 1981-12-23 GB GB8138860A patent/GB2090138A/en active Pending
- 1981-12-24 ES ES508351A patent/ES8304798A1/es not_active Expired
Also Published As
Publication number | Publication date |
---|---|
ES508351A0 (es) | 1983-03-16 |
GB2090138A (en) | 1982-07-07 |
AU7880181A (en) | 1982-07-01 |
EP0055609A1 (en) | 1982-07-07 |
AU546228B2 (en) | 1985-08-22 |
JPS57109713A (en) | 1982-07-08 |
JPS6348246B2 (es) | 1988-09-28 |
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