ES8304798A1 - Un procedimiento para la preparacion de una composicion de 4-amino-n-(5-metil-3-isoxazowil)benzenosulfonamida-5(3,4,5- trimetoxifenil)metil(2,4-pirimidinodamina. - Google Patents

Un procedimiento para la preparacion de una composicion de 4-amino-n-(5-metil-3-isoxazowil)benzenosulfonamida-5(3,4,5- trimetoxifenil)metil(2,4-pirimidinodamina.

Info

Publication number
ES8304798A1
ES8304798A1 ES508351A ES508351A ES8304798A1 ES 8304798 A1 ES8304798 A1 ES 8304798A1 ES 508351 A ES508351 A ES 508351A ES 508351 A ES508351 A ES 508351A ES 8304798 A1 ES8304798 A1 ES 8304798A1
Authority
ES
Spain
Prior art keywords
composition
coelomic
administration
trimethoprim
ingredients
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES508351A
Other languages
English (en)
Other versions
ES508351A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Shionogi and Co Ltd
Original Assignee
Shionogi and Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi and Co Ltd filed Critical Shionogi and Co Ltd
Publication of ES508351A0 publication Critical patent/ES508351A0/es
Publication of ES8304798A1 publication Critical patent/ES8304798A1/es
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/683Diesters of a phosphorus acid with two hydroxy compounds, e.g. phosphatidylinositols
    • A61K31/685Diesters of a phosphorus acid with two hydroxy compounds, e.g. phosphatidylinositols one of the hydroxy compounds having nitrogen atoms, e.g. phosphatidylserine, lecithin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/63Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/02Suppositories; Bougies; Bases therefor; Ovules
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE COMPOSICIONES DE 4-AMINO-N-(5-METIL-3-ISOXAZOLIL)BENCENOSULFONAMIDA/ 5- (3,4,5-TRIMETOXIFENIL)METIL -2,4-PIRIMIDINDIAMINA, QUE TIENE APLICACIONES FARMACOLOGICAS PARA LA ADMINISTRACION CELOMICA DE AGENTES ANTIMICROBIANOS. CONSISTE EN MEZCLAR 4-AMINO-N-(5-METIL-3-ISOXAZOLIL)BENCENOSULFONAMIDA Y 5- (3,4,5-TRIMETOXIFENIL)METIL -2,4-PIRIMIDINDIAMINA EN PROPORCIONES ADECUADAS CON UN FOSFOLIPIDO, EN PROPORCION DE 0,5-5%, EN CALIENTE Y CON AGITACION HASTA CONSEGUIR UNA DISPERSION UNIFORME, Y A CONTINUACION MOLDEAR LA DISPERSION OBTENIDA.
ES508351A 1980-12-26 1981-12-24 Un procedimiento para la preparacion de una composicion de 4-amino-n-(5-metil-3-isoxazowil)benzenosulfonamida-5(3,4,5- trimetoxifenil)metil(2,4-pirimidinodamina. Expired ES8304798A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP55185780A JPS57109713A (en) 1980-12-26 1980-12-26 Pharmaceutical preparation of combined agent of sulfamethoxazole and trimethoprim for medication through celom

Publications (2)

Publication Number Publication Date
ES508351A0 ES508351A0 (es) 1983-03-16
ES8304798A1 true ES8304798A1 (es) 1983-03-16

Family

ID=16176757

Family Applications (1)

Application Number Title Priority Date Filing Date
ES508351A Expired ES8304798A1 (es) 1980-12-26 1981-12-24 Un procedimiento para la preparacion de una composicion de 4-amino-n-(5-metil-3-isoxazowil)benzenosulfonamida-5(3,4,5- trimetoxifenil)metil(2,4-pirimidinodamina.

Country Status (5)

Country Link
EP (1) EP0055609A1 (es)
JP (1) JPS57109713A (es)
AU (1) AU546228B2 (es)
ES (1) ES8304798A1 (es)
GB (1) GB2090138A (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5946223A (ja) * 1982-08-30 1984-03-15 Daito Koeki Kk 抗菌性組成物
US4699776A (en) * 1985-06-28 1987-10-13 R. P. Scherer Corporation Suppositories containing analgesics, antipyretics or anti-inflammatory agents
HU210693B (en) * 1991-10-11 1995-06-28 Egyt Gyogyszervegyeszeti Gyar Process for producing pharmaceutical compositions for injections without tissue damages, containing sulfamethoxazol and trimetoprime

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE667500C (de) * 1934-09-28 1938-11-14 Chemisch Pharmazeutische A G B Verfahren zur Herstellung von Grundmassen fuer Arzneistoffe zur Einfuehrung in Koerperhoehlen
US3485840A (en) * 1964-11-12 1969-12-23 Hoffmann La Roche 2,4-diamino - 5 - (2',4',5'-substituted benzyl) pyrimidines,intermediates and processes
IT1043853B (it) * 1973-04-19 1980-02-29 Chiesi P Supposte contenenti l associazione trimetoprim sulfametossazolo e metodo per ottenerle
JPS55102517A (en) * 1979-01-30 1980-08-05 Shionogi & Co Ltd Preparation of sulfamethoxazole-trimethoprim complex for administration via body cavity
DE2951142C2 (de) * 1979-12-19 1983-11-03 A. Nattermann & Cie GmbH, 5000 Köln Suppositorium-Zubereitung von Indometacin oder Acemetacin

Also Published As

Publication number Publication date
ES508351A0 (es) 1983-03-16
GB2090138A (en) 1982-07-07
AU7880181A (en) 1982-07-01
EP0055609A1 (en) 1982-07-07
AU546228B2 (en) 1985-08-22
JPS57109713A (en) 1982-07-08
JPS6348246B2 (es) 1988-09-28

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