ES556370A0 - Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8-puenteados - Google Patents
Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8-puenteadosInfo
- Publication number
- ES556370A0 ES556370A0 ES556370A ES556370A ES556370A0 ES 556370 A0 ES556370 A0 ES 556370A0 ES 556370 A ES556370 A ES 556370A ES 556370 A ES556370 A ES 556370A ES 556370 A0 ES556370 A0 ES 556370A0
- Authority
- ES
- Spain
- Prior art keywords
- quinolon
- bridged
- procedure
- obtaining
- carboxylic acids
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Quinoline Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19853522406 DE3522406A1 (de) | 1985-06-22 | 1985-06-22 | Verfahren zur herstellung von 1,8-verbrueckten 4-chinolon-3-carbonsaeuren |
Publications (2)
Publication Number | Publication Date |
---|---|
ES556370A0 true ES556370A0 (es) | 1987-12-16 |
ES8801210A1 ES8801210A1 (es) | 1987-12-16 |
Family
ID=6273930
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES556370A Expired ES8801210A1 (es) | 1985-06-22 | 1986-06-20 | Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8-puenteados |
ES557698A Expired ES8801920A1 (es) | 1985-06-22 | 1987-08-28 | Procedimiento para la obtencio de enaminas |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES557698A Expired ES8801920A1 (es) | 1985-06-22 | 1987-08-28 | Procedimiento para la obtencio de enaminas |
Country Status (6)
Country | Link |
---|---|
US (3) | US4762831A (es) |
EP (1) | EP0206101A1 (es) |
JP (1) | JPS62452A (es) |
KR (1) | KR880000439A (es) |
DE (1) | DE3522406A1 (es) |
ES (2) | ES8801210A1 (es) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3522405A1 (de) * | 1985-06-22 | 1987-01-02 | Bayer Ag | 1,8-verbrueckte 4-chinolon-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende arzneimittel und ihre verwendung zur herstellung von arzneimitteln |
US5237060A (en) * | 1985-12-10 | 1993-08-17 | Bayer Aktiengesellschaft | Process of preparing enantiomerically pure 1,8-bridged 4-quinolone-3-carboxylic acids |
US5147871A (en) * | 1986-07-03 | 1992-09-15 | Hoffmann La-Roche, Inc. | Anti-bacterial cephalosporin compounds |
DE3881939T2 (de) * | 1987-02-26 | 1993-09-30 | Rohto Pharma | Verwendung von Ofloxacin zur lokalen Behandlung oder Prophylaxe von Beschwerden der Wurzelhaut der Zähne. |
US5591744A (en) * | 1987-04-16 | 1997-01-07 | Otsuka Pharmaceutical Company, Limited | Benzoheterocyclic compounds |
US5290934A (en) * | 1987-04-16 | 1994-03-01 | Otsuka Pharmaceutical Company, Limited | Benzoheterocyclic compounds |
JPH0826029B2 (ja) * | 1987-12-22 | 1996-03-13 | 第一製薬株式会社 | 魚類感染症の予防・治療剤 |
US4920120A (en) | 1988-01-25 | 1990-04-24 | Warner-Lambert Company | Antibacterial agents |
US5585491A (en) * | 1988-01-25 | 1996-12-17 | Otsuka Pharmaceutical Co., Ltd. | Antibacterial agents |
JPH0228178A (ja) * | 1988-04-23 | 1990-01-30 | Toyama Chem Co Ltd | 新規なピリドンカルボン酸誘導体およびその塩並びにそれらの製造法 |
CS273349B2 (en) * | 1988-03-31 | 1991-03-12 | Hoffmann La Roche | Method of cephalosporin's new derivatives production |
US5336768A (en) * | 1988-05-24 | 1994-08-09 | Hoffmann-La Roche Inc. | Antibacterial cephalosporin compounds |
DE3902079A1 (de) * | 1988-04-15 | 1989-10-26 | Bayer Ag | I.m. injektionsformen von gyrase-inhibitoren |
US4996355A (en) * | 1989-04-14 | 1991-02-26 | Mallinckrodt, Inc. | Novel intermediates for the production of 2,4,5-trifluorobenzoyl fluoride |
US5162523A (en) * | 1989-07-21 | 1992-11-10 | Hoffmann-La Roche Inc. | Cephalosporin antibacterial compounds |
US5159077A (en) * | 1989-07-21 | 1992-10-27 | Hoffmann-La Roche Inc. | Penam antibacterial compounds |
CA2081548A1 (en) * | 1991-02-28 | 1992-08-29 | Hideo Tsutsumi | Process for producing tricyclic compounds or salts thereof |
WO1994007873A1 (es) * | 1992-10-07 | 1994-04-14 | Derivados Del Etilo, S.A. | Prodedimiento para la obtencion de benzoxazinas utiles para la sintesis de ofloxacina, levofloxacina y derivados |
ES2055656B1 (es) * | 1992-10-07 | 1995-11-16 | Etilo Derivados | Procedimiento para la obtencion de benzoxazinas utiles para sintesis de ofloxacina, levofloxacina y derivados. |
US5644056A (en) * | 1995-06-07 | 1997-07-01 | Hoechst Celanese Corporation | Method of preparing 7,8-difluoro-2,3-dihydro-3-methyl-4H-1, 4-benzoxazine |
KR100309871B1 (ko) | 1999-02-24 | 2001-10-29 | 윤종용 | (-)피리도벤즈옥사진 카르복실산 유도체의 제조방법 |
WO2006009143A1 (ja) * | 2004-07-21 | 2006-01-26 | Kyorin Pharmaceutical Co., Ltd. | (3s)-3-ヒドロキシメチル-7-オキソピリドベンゾオキサジン-6-カルボン酸エステルの製造方法 |
CA2629077C (en) * | 2005-11-16 | 2014-03-18 | F. Hoffmann-La Roche Ag | Novel process for the preparation of thoc |
ES2427247T3 (es) | 2006-03-13 | 2013-10-30 | Kyorin Pharmaceutical Co., Ltd. | Aminoquinolonas como inhibidores de GSK-3 |
BRPI0816814B1 (pt) | 2007-09-12 | 2021-08-31 | Kyorin Pharmaceutical Co. Ltd | Composto, composição farmacêutica e uso de um composto |
WO2010104205A1 (en) | 2009-03-11 | 2010-09-16 | Kyorin Pharmaceutical Co., Ltd. | 7-cycloalkylaminoquinolones as gsk-3 inhibitors |
CN103183684B (zh) * | 2011-12-29 | 2015-11-18 | 杭州师范大学 | 一种喹喏酮内酯化合物及其制备方法和应用 |
CN105037388A (zh) * | 2015-08-28 | 2015-11-11 | 安徽环球药业股份有限公司 | 一种安妥沙星的制备方法 |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE62321C (de) * | O. MEURER in Köln a. Rh., Mühlenbach 54—58 | Neuerung an einem Bodenbelag für Malztennen u. dergl | ||
DD62321A (es) * | ||||
CA947301A (en) * | 1970-01-28 | 1974-05-14 | Sumitomo Chemical Company | Process for the preparation of compound having antibacterial action |
US3883522A (en) * | 1974-02-11 | 1975-05-13 | Riker Laboratories Inc | Substituted pyrido(1,2,3-de)-1,4-benzoxazines |
DE2808070A1 (de) * | 1978-02-24 | 1979-08-30 | Bayer Ag | Verfahren zur herstellung von 4-pyridon-3-carbonsaeuren und/oder deren derivaten |
JPS5746986A (en) * | 1980-09-02 | 1982-03-17 | Dai Ichi Seiyaku Co Ltd | Pyrido(1,2,3-de)(1,4)benzoxazine derivative |
SE440354B (sv) * | 1981-02-19 | 1985-07-29 | Kyorin Seiyaku Kk | Kinolinkarboxylsyraderivat |
US4499270A (en) * | 1981-04-16 | 1985-02-12 | Riker Laboratories, Inc. | Substituted pyridoquinoxaline-6-carboxylic acids and derivatives thereof |
US4571396A (en) * | 1984-04-16 | 1986-02-18 | Warner-Lambert Company | Antibacterial agents |
DE3416120A1 (de) * | 1984-04-30 | 1985-10-31 | Henkel KGaA, 4000 Düsseldorf | Benzoylalanine und ihre verwendung als korrosionsinhibitoren fuer waessrige systeme |
US4571346A (en) * | 1984-08-01 | 1986-02-18 | General Foods Corporation | Method for producing cold-water soluble gelatin dessert mixes and products therefrom |
US4777253A (en) * | 1986-04-25 | 1988-10-11 | Abbott Laboratories | Process for preparation of racemate and optically active ofloxacin and related derivatives |
-
1985
- 1985-06-22 DE DE19853522406 patent/DE3522406A1/de not_active Withdrawn
-
1986
- 1986-06-10 EP EP86107908A patent/EP0206101A1/de not_active Withdrawn
- 1986-06-13 US US06/874,182 patent/US4762831A/en not_active Expired - Fee Related
- 1986-06-20 ES ES556370A patent/ES8801210A1/es not_active Expired
- 1986-06-20 JP JP61143150A patent/JPS62452A/ja active Pending
- 1986-06-21 KR KR1019860004972A patent/KR880000439A/ko not_active Application Discontinuation
-
1987
- 1987-08-28 ES ES557698A patent/ES8801920A1/es not_active Expired
-
1988
- 1988-03-24 US US07/172,612 patent/US4859773A/en not_active Expired - Fee Related
-
1989
- 1989-03-30 US US07/331,339 patent/US4958045A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EP0206101A1 (de) | 1986-12-30 |
US4762831A (en) | 1988-08-09 |
ES557698A0 (es) | 1988-03-01 |
ES8801920A1 (es) | 1988-03-01 |
US4859773A (en) | 1989-08-22 |
US4958045A (en) | 1990-09-18 |
DE3522406A1 (de) | 1987-01-02 |
KR880000439A (ko) | 1988-03-25 |
JPS62452A (ja) | 1987-01-06 |
ES8801210A1 (es) | 1987-12-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD1A | Patent lapsed |
Effective date: 19970401 |