ES552284A0 - Procedimiento para preparar 1,2-dihidro-naftalenos y derivados 1-oxa,1-tia, 1-sulfinilo y 1-sulfonilo de los mismos - Google Patents

Procedimiento para preparar 1,2-dihidro-naftalenos y derivados 1-oxa,1-tia, 1-sulfinilo y 1-sulfonilo de los mismos

Info

Publication number
ES552284A0
ES552284A0 ES552284A ES552284A ES552284A0 ES 552284 A0 ES552284 A0 ES 552284A0 ES 552284 A ES552284 A ES 552284A ES 552284 A ES552284 A ES 552284A ES 552284 A0 ES552284 A0 ES 552284A0
Authority
ES
Spain
Prior art keywords
tia
sulfinyl
oxa
dihydro
naphthalene
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES552284A
Other languages
English (en)
Other versions
ES8708223A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GSK Consumer Healthcare SARL
Original Assignee
Zyma SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zyma SA filed Critical Zyma SA
Publication of ES8708223A1 publication Critical patent/ES8708223A1/es
Publication of ES552284A0 publication Critical patent/ES552284A0/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/74Naphthothiophenes
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/10Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pulmonology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ES552284A 1985-02-23 1986-02-21 Procedimiento para preparar 1,2-dihidro-naftalenos y derivados 1-oxa,1-tia, 1-sulfinilo y 1-sulfonilo de los mismos Expired ES8708223A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858504702A GB8504702D0 (en) 1985-02-23 1985-02-23 Tricyclic compounds

Publications (2)

Publication Number Publication Date
ES8708223A1 ES8708223A1 (es) 1987-10-01
ES552284A0 true ES552284A0 (es) 1987-10-01

Family

ID=10574972

Family Applications (2)

Application Number Title Priority Date Filing Date
ES552284A Expired ES8708223A1 (es) 1985-02-23 1986-02-21 Procedimiento para preparar 1,2-dihidro-naftalenos y derivados 1-oxa,1-tia, 1-sulfinilo y 1-sulfonilo de los mismos
ES557389A Expired ES8801834A1 (es) 1985-02-23 1987-02-13 Procedimiento para preparar 1,2-dihidronaftalenos y derivados 1-oxa, 1-tia 1-sulfinilo y 1-sulfonilo de los mismos

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES557389A Expired ES8801834A1 (es) 1985-02-23 1987-02-13 Procedimiento para preparar 1,2-dihidronaftalenos y derivados 1-oxa, 1-tia 1-sulfinilo y 1-sulfonilo de los mismos

Country Status (19)

Country Link
US (1) US4797414A (es)
EP (1) EP0193493A3 (es)
JP (1) JPS61194081A (es)
KR (1) KR860006470A (es)
AU (1) AU593238B2 (es)
CA (1) CA1284326C (es)
DD (1) DD249019A5 (es)
DK (1) DK81586A (es)
ES (2) ES8708223A1 (es)
FI (1) FI860738A (es)
GB (1) GB8504702D0 (es)
GR (1) GR860500B (es)
HU (1) HU196075B (es)
IL (1) IL77919A0 (es)
NO (1) NO164172C (es)
NZ (1) NZ215253A (es)
PH (1) PH24908A (es)
PT (1) PT82061B (es)
ZA (1) ZA861304B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005536518A (ja) * 2002-07-19 2005-12-02 ファルマシア コーポレイション 炎症治療のための置換チオフェンカルボキサミド化合物
JP2006151810A (ja) * 2002-12-26 2006-06-15 Daiichi Asubio Pharma Co Ltd ジヒドロチエノキノリン誘導体及びそれを含む細胞接着阻害剤
US7384974B2 (en) * 2003-07-31 2008-06-10 Taisha Pharmaceutical Co., Ltd. 4,5-dihydronaphtho[1,2-b]thiophene derivative
WO2006080439A1 (ja) * 2005-01-28 2006-08-03 Taisho Pharmaceutical Co., Ltd. 三環性化合物
WO2006080406A1 (ja) * 2005-01-28 2006-08-03 Taisho Pharmaceutical Co., Ltd. 三環性化合物
PL2276767T3 (pl) 2008-03-31 2014-09-30 Genentech Inc Związki benzopiranowe i benzoksepinowe będące inhibitorami pi3k oraz metody ich stosowania
SG10201407781SA (en) 2009-09-28 2015-01-29 Hoffmann La Roche Benzoxepin PI3K Inhibitor Compounds And Methods Of Use
RS53164B (en) 2009-09-28 2014-06-30 F. Hoffmann-La Roche Ag BENZOXAZEPINE PI3K INHIBITOR COMPOUNDS AND THEIR USE IN CANCER TREATMENT
CA2825966A1 (en) 2011-03-21 2012-09-27 F. Hoffmann-La Roche Ag Benzoxazepin compounds selective for pi3k p110 delta and methods of use
ES2715832T3 (es) * 2011-05-27 2019-06-06 Lexicon Pharmaceuticals Inc Inhibidores a base de 4H-tieno[3,2-c]-cromeno de pectina acetilesterasa de notum y métodos de utilización de los mismos

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1917601C3 (de) * 1969-04-05 1980-09-25 Bayer Ag, 5090 Leverkusen Benzoxazolyl-(2)-dihydronaphtho [4,5-b] thiophene und deren Verwendung als optische Aufheller
US3656906A (en) * 1970-04-13 1972-04-18 Little Inc A Method for detecting and quantitating the presence of cannabinoids and analogs thereof in biological materials and resulting products
DK44278A (da) * 1977-02-08 1978-08-09 Sandoz Ag Fremgangsmaade til fremstilling af thiophenderivater
US4268516A (en) * 1978-10-11 1981-05-19 Pfizer Inc. [1]Benzothiopyrano[4,3-c]pyrazoles as immunoregulatory agents
DE3023301A1 (de) * 1980-06-21 1982-01-14 Bayer Ag, 5090 Leverkusen Benzoxazolyldihydronaphthothiophenverbindungen sowie verwendung als optische aufheller

Also Published As

Publication number Publication date
PT82061A (en) 1986-03-01
IL77919A0 (en) 1986-09-30
FI860738A (fi) 1986-08-24
DK81586D0 (da) 1986-02-21
JPS61194081A (ja) 1986-08-28
CA1284326C (en) 1991-05-21
NO860654L (no) 1986-08-25
HUT41762A (en) 1987-05-28
AU5387586A (en) 1986-08-28
ES8801834A1 (es) 1988-02-16
AU593238B2 (en) 1990-02-08
ES557389A0 (es) 1988-02-16
NO164172B (no) 1990-05-28
FI860738A0 (fi) 1986-02-19
DD249019A5 (de) 1987-08-26
PH24908A (en) 1990-12-26
KR860006470A (ko) 1986-09-11
NO164172C (no) 1990-09-05
ES8708223A1 (es) 1987-10-01
GR860500B (en) 1986-06-18
HU196075B (en) 1988-09-28
EP0193493A2 (en) 1986-09-03
DK81586A (da) 1986-08-24
GB8504702D0 (en) 1985-03-27
NZ215253A (en) 1989-10-27
ZA861304B (en) 1986-10-29
US4797414A (en) 1989-01-10
PT82061B (pt) 1988-07-01
EP0193493A3 (en) 1988-01-13

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