ES541799A0 - Procedimiento de preparar derivados penam y sus sales - Google Patents

Procedimiento de preparar derivados penam y sus sales

Info

Publication number
ES541799A0
ES541799A0 ES541799A ES541799A ES541799A0 ES 541799 A0 ES541799 A0 ES 541799A0 ES 541799 A ES541799 A ES 541799A ES 541799 A ES541799 A ES 541799A ES 541799 A0 ES541799 A0 ES 541799A0
Authority
ES
Spain
Prior art keywords
salts
preparing
procedure
penam derivatives
penam
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES541799A
Other languages
English (en)
Other versions
ES8700669A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Taiho Pharmaceutical Co Ltd
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Publication of ES541799A0 publication Critical patent/ES541799A0/es
Publication of ES8700669A1 publication Critical patent/ES8700669A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/86Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with only atoms other than nitrogen atoms directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES541799A 1984-04-06 1985-04-01 Procedimiento de preparar derivados penam y sus sales Expired ES8700669A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP59069843A JPS60214792A (ja) 1984-04-06 1984-04-06 ペナム酸エステル誘導体

Publications (2)

Publication Number Publication Date
ES541799A0 true ES541799A0 (es) 1986-11-16
ES8700669A1 ES8700669A1 (es) 1986-11-16

Family

ID=13414488

Family Applications (2)

Application Number Title Priority Date Filing Date
ES541799A Expired ES8700669A1 (es) 1984-04-06 1985-04-01 Procedimiento de preparar derivados penam y sus sales
ES551250A Expired ES8703478A1 (es) 1984-04-06 1986-01-27 Procedimiento de preparar derivados penam y sus sales.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES551250A Expired ES8703478A1 (es) 1984-04-06 1986-01-27 Procedimiento de preparar derivados penam y sus sales.

Country Status (8)

Country Link
US (1) US4626384A (es)
EP (1) EP0158494B1 (es)
JP (1) JPS60214792A (es)
KR (1) KR900007199B1 (es)
AU (1) AU555768B2 (es)
CA (1) CA1240667A (es)
DE (1) DE3576342D1 (es)
ES (2) ES8700669A1 (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3306473B1 (ja) * 2001-05-01 2002-07-24 大塚化学株式会社 β−ラクタム化合物の無水結晶及びその製造法
US7417143B2 (en) * 2004-04-07 2008-08-26 Orchid Chemicals & Pharmaceuticals Limited Process for the preparation of Tazobactam in pure form
US20060173177A1 (en) * 2005-01-28 2006-08-03 Gego Csaba L Process for preparation of penam derivatives
CN102952148B (zh) * 2011-08-26 2014-11-05 秦引林 一种他唑巴坦钠的精制方法
WO2013036783A2 (en) 2011-09-09 2013-03-14 Cubist Pharmaceuticals, Inc. Methods for treating intrapulmonary infections
US8809314B1 (en) 2012-09-07 2014-08-19 Cubist Pharmacueticals, Inc. Cephalosporin compound
US8476425B1 (en) 2012-09-27 2013-07-02 Cubist Pharmaceuticals, Inc. Tazobactam arginine compositions
KR102329764B1 (ko) 2013-03-15 2021-11-23 머크 샤프 앤드 돔 코포레이션 세프톨로잔 항균성 조성물
US9872906B2 (en) 2013-03-15 2018-01-23 Merck Sharp & Dohme Corp. Ceftolozane antibiotic compositions
US20140274991A1 (en) 2013-03-15 2014-09-18 Cubist Pharmaceuticals, Inc. Ceftolozane pharmaceutical compositions
WO2015035376A2 (en) 2013-09-09 2015-03-12 Calixa Therapeutics, Inc. Treating infections with ceftolozane/tazobactam in subjects having impaired renal function
US8906898B1 (en) 2013-09-27 2014-12-09 Calixa Therapeutics, Inc. Solid forms of ceftolozane

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4364957A (en) * 1979-09-26 1982-12-21 Pfizer Inc. Bis-esters of alkanediols as antibacterial agents
US4540687A (en) * 1981-09-09 1985-09-10 Pfizer Inc. Antibacterial 6'-(2-amino-2-[4-acyloxyphenyl]acetamido)penicillanoyloxymethyl penicillanate 1,1-dioxide compounds
AU541028B2 (en) * 1982-06-21 1984-12-13 Taiho Pharmaceutical Co., Ltd. 6-unsubstituted penicillin derivatives
JPS5995291A (ja) * 1982-11-24 1984-06-01 Taiho Yakuhin Kogyo Kk ペニシリン誘導体
US4562073A (en) * 1982-12-24 1985-12-31 Taiho Pharmaceutical Company Limited Penicillin derivatives

Also Published As

Publication number Publication date
KR900007199B1 (ko) 1990-10-05
JPH041757B2 (es) 1992-01-14
CA1240667A (en) 1988-08-16
EP0158494A1 (en) 1985-10-16
ES551250A0 (es) 1987-03-01
DE3576342D1 (de) 1990-04-12
KR850007601A (ko) 1985-12-07
US4626384A (en) 1986-12-02
JPS60214792A (ja) 1985-10-28
AU555768B2 (en) 1986-10-09
EP0158494B1 (en) 1990-03-07
ES8703478A1 (es) 1987-03-01
ES8700669A1 (es) 1986-11-16
AU4048985A (en) 1985-10-10

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20000601