ES464555A1 - Procedimiento para preparar derivados de acidos tiazolidin- ,tiazano-carboxilicos y afines. - Google Patents

Procedimiento para preparar derivados de acidos tiazolidin- ,tiazano-carboxilicos y afines.

Info

Publication number
ES464555A1
ES464555A1 ES464555A ES464555A ES464555A1 ES 464555 A1 ES464555 A1 ES 464555A1 ES 464555 A ES464555 A ES 464555A ES 464555 A ES464555 A ES 464555A ES 464555 A1 ES464555 A1 ES 464555A1
Authority
ES
Spain
Prior art keywords
thiazane
thiazolidine
esters
carboxylic acids
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES464555A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of ES464555A1 publication Critical patent/ES464555A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D277/06Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/041,3-Thiazines; Hydrogenated 1,3-thiazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/121,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
ES464555A 1976-12-03 1977-11-29 Procedimiento para preparar derivados de acidos tiazolidin- ,tiazano-carboxilicos y afines. Expired ES464555A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74728176A 1976-12-03 1976-12-03
US83610777A 1977-09-23 1977-09-23

Publications (1)

Publication Number Publication Date
ES464555A1 true ES464555A1 (es) 1978-09-01

Family

ID=27114718

Family Applications (1)

Application Number Title Priority Date Filing Date
ES464555A Expired ES464555A1 (es) 1976-12-03 1977-11-29 Procedimiento para preparar derivados de acidos tiazolidin- ,tiazano-carboxilicos y afines.

Country Status (28)

Country Link
JP (1) JPS5382778A (ro)
AR (1) AR220689A1 (ro)
AT (1) AT363467B (ro)
AU (1) AU518147B2 (ro)
BG (1) BG32269A3 (ro)
CA (1) CA1146940A (ro)
CH (1) CH634062A5 (ro)
DD (1) DD133798A5 (ro)
DE (1) DE2752719C2 (ro)
DK (1) DK152494C (ro)
EG (1) EG13037A (ro)
ES (1) ES464555A1 (ro)
FI (1) FI67378C (ro)
FR (1) FR2372817A1 (ro)
GB (1) GB1578940A (ro)
GR (1) GR72453B (ro)
HK (1) HK55881A (ro)
IE (1) IE46169B1 (ro)
IL (1) IL53352A0 (ro)
IN (1) IN146945B (ro)
IT (1) IT1092179B (ro)
NL (3) NL171055C (ro)
NO (1) NO148416C (ro)
NZ (1) NZ185800A (ro)
PT (1) PT67352B (ro)
RO (2) RO78013A (ro)
SE (1) SE441267B (ro)
YU (1) YU41823B (ro)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1105731B (it) * 1977-06-29 1985-11-04 Yoshitomi Pharmaceutical Composti di tiazolidina
JPS5455565A (en) * 1977-10-06 1979-05-02 Santen Pharmaceut Co Ltd Novel thiazolidine derivative
US4430344A (en) * 1978-04-08 1984-02-07 Santen Pharmaceutical Co., Ltd. Antihypertensive 4-thiazolidinecarboxylic acids
JPS557255A (en) * 1978-07-03 1980-01-19 Santen Pharmaceut Co Ltd Thiazolidine derivative
JPS5531022A (en) * 1978-08-24 1980-03-05 Yoshitomi Pharmaceut Ind Ltd Hydroxamic acid derivative and its preparation
GR73585B (ro) * 1978-09-11 1984-03-26 Univ Miami
JPS5540622A (en) * 1978-09-14 1980-03-22 Santen Pharmaceut Co Ltd Hypotensive agent
JPS5829950B2 (ja) * 1978-10-05 1983-06-25 ウェルファイド株式会社 環状イミノカルボン酸誘導体およびその塩類
US4483861A (en) * 1978-10-31 1984-11-20 Santen Pharmaceutical Co., Ltd. Antihypertensive sulfur-containing compounds
JPS5562060A (en) * 1978-10-31 1980-05-10 Santen Pharmaceut Co Ltd Sulfur-containing compound
JPS565415A (en) * 1979-06-26 1981-01-20 Santen Pharmaceut Co Ltd Ester-type hypotensor
US4347371A (en) * 1978-12-30 1982-08-31 Santen Pharmaceutical Co., Ltd. Disulfide compounds
JPS55124757A (en) * 1979-03-17 1980-09-26 Santen Pharmaceut Co Ltd Sulfur-containing compound
JPS5683483A (en) * 1979-12-13 1981-07-08 Santen Pharmaceut Co Ltd Thiazolidine compound
JPS56139455A (en) * 1980-04-02 1981-10-30 Santen Pharmaceut Co Ltd Sulfur-containing acylaminoacid
DE3152643A1 (de) * 1980-12-29 1982-12-16 Santen Pharmaceutical Co Ltd Heterocyclic 5-membered ring compounds
JPH0662529B2 (ja) * 1984-07-13 1994-08-17 三共株式会社 アミノ酸誘導体
DE3685829T2 (de) * 1985-02-04 1992-12-17 Searle & Co Heterocyclische amide.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2446100C3 (de) * 1974-09-26 1982-01-14 Ludwig Merckle Kg Chem. Pharm. Fabrik, 7902 Blaubeuren Phenoxyalkancarbonsäureamide von Thiazolidincarbonsäuren, Verfahren zu ihrer Herstellung und Arzneimittel
AU509899B2 (en) * 1976-02-13 1980-05-29 E.R. Squibb & Sons, Inc. Proline derivatives and related compounds

Also Published As

Publication number Publication date
ATA857677A (de) 1981-01-15
JPS618834B2 (ro) 1986-03-18
CH634062A5 (en) 1983-01-14
DD133798A5 (de) 1979-01-24
NL7713274A (nl) 1978-06-06
HK55881A (en) 1981-11-20
RO72596A (ro) 1983-08-03
PT67352B (fr) 1979-05-15
FR2372817A1 (fr) 1978-06-30
FR2372817B1 (ro) 1981-06-19
EG13037A (en) 1980-12-31
IN146945B (ro) 1979-10-20
IE46169B1 (en) 1983-03-09
FI773640A (fi) 1978-06-04
FI67378B (fi) 1984-11-30
FI67378C (fi) 1985-03-11
IE46169L (en) 1978-06-03
DE2752719A1 (de) 1978-06-08
NO148416C (no) 1983-10-12
NO148416B (no) 1983-06-27
DK152494C (da) 1988-07-25
NL8201145A (nl) 1982-07-01
DE2752719C2 (de) 1982-03-25
IL53352A0 (en) 1978-01-31
RO72596B (ro) 1983-07-30
GR72453B (ro) 1983-11-09
NL171055C (nl) 1983-02-01
DK152494B (da) 1988-03-07
RO78013A (ro) 1981-12-25
NL8201146A (nl) 1982-07-01
DK538277A (da) 1978-06-04
AU518147B2 (en) 1981-09-17
NZ185800A (en) 1980-04-28
SE441267B (sv) 1985-09-23
JPS5382778A (en) 1978-07-21
SE7713722L (sv) 1978-06-04
IT1092179B (it) 1985-07-06
AT363467B (de) 1981-08-10
CA1146940A (en) 1983-05-24
BG32269A3 (en) 1982-06-15
AU3037977A (en) 1979-05-17
PT67352A (fr) 1978-01-01
YU41823B (en) 1988-02-29
GB1578940A (en) 1980-11-12
NO774126L (no) 1978-06-06
YU283777A (en) 1983-01-21
AR220689A1 (es) 1980-11-28

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19991213