ES2878001T3 - Composiciones del activador de la glucocinasa para el tratamiento de la diabetes - Google Patents
Composiciones del activador de la glucocinasa para el tratamiento de la diabetes Download PDFInfo
- Publication number
- ES2878001T3 ES2878001T3 ES13726933T ES13726933T ES2878001T3 ES 2878001 T3 ES2878001 T3 ES 2878001T3 ES 13726933 T ES13726933 T ES 13726933T ES 13726933 T ES13726933 T ES 13726933T ES 2878001 T3 ES2878001 T3 ES 2878001T3
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- Prior art keywords
- pharmaceutically acceptable
- acceptable salt
- diabetes
- pharmaceutical composition
- cyclohexyl
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| US201261648110P | 2012-05-17 | 2012-05-17 | |
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| PT2576524T (pt) | 2010-05-26 | 2017-11-17 | Vtv Therapeutics Llc | Resumo |
| IN2014DN09554A (enExample) * | 2012-05-17 | 2015-07-17 | Transtech Pharma Llc | |
| KR102408480B1 (ko) | 2018-05-30 | 2022-06-10 | 이삼구 | 당뇨질환의 치료용 조성물 |
| BR112020024269A2 (pt) * | 2018-05-31 | 2021-02-23 | Hua Medicine (Shanghai) Ltd. | combinação farmacêutica, composição e formulação de combinação contendo ativador de glucoquinase e ativador de receptor ppar e métodos de preparação e usos dos mesmos |
| CA3093025A1 (en) | 2018-06-12 | 2019-12-19 | Vtv Therapeutics Llc | Therapeutic uses of glucokinase activators in combination with insulin or insulin analogs |
| AU2020426356A1 (en) * | 2020-01-31 | 2022-08-25 | Hua Medicine (Shanghai) Ltd. | Treating treatment-resistant diabetes with glucokinase activator |
| US11872221B2 (en) | 2020-01-31 | 2024-01-16 | Hua Medicine (Shanghai) Ltd. | Treating untreated or treatment-resistant diabetes with glucokinase activator |
| US12391658B2 (en) | 2020-02-18 | 2025-08-19 | Vtv Therapeutics Llc | Sulfoxide and sulfone glucokinase activators and methods of use thereof |
| WO2021243646A1 (en) * | 2020-06-04 | 2021-12-09 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with hepatic impairment |
| CA3185831A1 (en) * | 2020-06-04 | 2021-12-09 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with renal impairment |
| US11857536B2 (en) | 2020-06-04 | 2024-01-02 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with renal impairment |
| US12479808B2 (en) | 2020-06-08 | 2025-11-25 | Vtv Therapeutics Llc | Salts or co-crystals of {2-[3-cyclohexyl-3-(trans-4-propoxy-cyclohexyl)-ureido]-thiazol-5-ylsulfanyl}-acetic acid and uses thereof |
| CA3181665A1 (en) * | 2020-06-08 | 2021-12-16 | Jing TENG | Crystalline forms of {2-[3-cyclohexyl-3-(trans-4-propoxy- cyclohexyl)-ureido]-thiazol-5-ylsulfanyl} -acetic acid and and uses thereof |
| CN115350268B (zh) * | 2022-08-24 | 2025-02-11 | 深圳青澜生物技术有限公司 | 一种用于治疗糖尿病的制剂、微针及其制备工艺 |
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| AU2013262895A1 (en) | 2014-11-13 |
| BR112014028622A2 (pt) | 2017-06-27 |
| US10980861B2 (en) | 2021-04-20 |
| US10588943B2 (en) | 2020-03-17 |
| KR102371364B1 (ko) | 2022-03-07 |
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| HK1202458A1 (en) | 2015-10-02 |
| EP2849776A2 (en) | 2015-03-25 |
| MX360304B (es) | 2018-10-29 |
| IL235484A0 (en) | 2014-12-31 |
| EA201492109A1 (ru) | 2015-07-30 |
| US20140066372A1 (en) | 2014-03-06 |
| US20180311314A1 (en) | 2018-11-01 |
| CN104349790A (zh) | 2015-02-11 |
| KR20150013838A (ko) | 2015-02-05 |
| US20200138909A1 (en) | 2020-05-07 |
| WO2013173417A2 (en) | 2013-11-21 |
| CA2872021C (en) | 2022-08-16 |
| SG11201406987UA (en) | 2014-12-30 |
| KR20210027547A (ko) | 2021-03-10 |
| CA2872021A1 (en) | 2013-11-21 |
| AU2017203835B2 (en) | 2018-11-22 |
| IN2014DN09554A (enExample) | 2015-07-17 |
| WO2013173417A3 (en) | 2014-02-20 |
| SG10201609644UA (en) | 2017-01-27 |
| CN118453592A (zh) | 2024-08-09 |
| US10004782B2 (en) | 2018-06-26 |
| AU2017203835A1 (en) | 2017-06-22 |
| MX2014013105A (es) | 2015-04-08 |
| EP2849776B1 (en) | 2021-04-21 |
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