ES2837484T3 - Rapadocinas, inhibidores del transportador de nucleósidos equilibrativo 1 y usos de los mismos - Google Patents
Rapadocinas, inhibidores del transportador de nucleósidos equilibrativo 1 y usos de los mismosInfo
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- ES2837484T3 ES2837484T3 ES17748270T ES17748270T ES2837484T3 ES 2837484 T3 ES2837484 T3 ES 2837484T3 ES 17748270 T ES17748270 T ES 17748270T ES 17748270 T ES17748270 T ES 17748270T ES 2837484 T3 ES2837484 T3 ES 2837484T3
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| US201662291428P | 2016-02-04 | 2016-02-04 | |
| PCT/US2017/016494 WO2017136717A1 (en) | 2016-02-04 | 2017-02-03 | Rapadocins, inhibitors of equilibrative nucleoside transporter 1 and uses thereof |
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| ES2837484T3 true ES2837484T3 (es) | 2021-06-30 |
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| ES17748270T Active ES2837484T3 (es) | 2016-02-04 | 2017-02-03 | Rapadocinas, inhibidores del transportador de nucleósidos equilibrativo 1 y usos de los mismos |
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| EP (2) | EP3411032B1 (https=) |
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| US10774110B2 (en) * | 2016-02-04 | 2020-09-15 | The Johns Hopkins University | Rapadocins, inhibitors of equilibrative nucleoside transporter 1 and uses thereof |
| CA3013783A1 (en) * | 2016-02-04 | 2017-08-10 | The Johns Hopkins University | Rapaglutins, novel inhibitors of glut and use thereof |
| US11066416B2 (en) | 2016-02-04 | 2021-07-20 | The Johns Hopkins University | Rapafucin derivative compounds and methods of use thereof |
| TW202126323A (zh) * | 2019-10-01 | 2021-07-16 | 約翰斯赫普金斯大學 | 雷帕弗辛（Ｒａｐａｆｕｃｉｎ）衍生化合物及其使用方法 |
| AR121777A1 (es) * | 2020-04-07 | 2022-07-06 | iTeos Belgium SA | Derivados de diamina macrocíclica como inhibidores de ent para el tratamiento de cánceres, y combinación de estos con antagonistas del receptor de adenosina |
| JP2024537110A (ja) * | 2021-10-06 | 2024-10-10 | アイテオ ベルギウム エスエー | Ｅｎｔ１阻害活性を有する大環状化合物 |
| WO2023056910A1 (en) * | 2021-10-06 | 2023-04-13 | iTeos Belgium SA | Processes for preparing a macrocyclic compound having ent1 inhibiting activity |
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| US10774110B2 (en) | 2016-02-04 | 2020-09-15 | The Johns Hopkins University | Rapadocins, inhibitors of equilibrative nucleoside transporter 1 and uses thereof |
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| WO2018045250A1 (en) | 2016-09-02 | 2018-03-08 | The Johns Hopkins University | Mif inhibitors and methods of use thereof |
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| CN108697701A (zh) | 2018-10-23 |
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