ES2693520T3 - Quinazolinas sustituidas con sulfoximina para composiciones farmacéuticas - Google Patents
Quinazolinas sustituidas con sulfoximina para composiciones farmacéuticas Download PDFInfo
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- ES2693520T3 ES2693520T3 ES14808895.8T ES14808895T ES2693520T3 ES 2693520 T3 ES2693520 T3 ES 2693520T3 ES 14808895 T ES14808895 T ES 14808895T ES 2693520 T3 ES2693520 T3 ES 2693520T3
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
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Landscapes
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| EP13195720 | 2013-12-04 | ||
| EP13195720 | 2013-12-04 | ||
| PCT/EP2014/075890 WO2015082324A1 (en) | 2013-12-04 | 2014-11-28 | Sulfoximine substituted quinazolines for pharmaceutical compositions |
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| ES2693520T3 true ES2693520T3 (es) | 2018-12-12 |
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| AR117788A1 (es) * | 2019-01-14 | 2021-08-25 | Pi Industries Ltd | Compuestos de fenilamidina 3-sustituida, preparación y uso |
| CN112812136B (zh) * | 2019-11-15 | 2022-04-12 | 武汉光谷亚太医药研究院有限公司 | 新型2,3-二氢化茚衍生化合物、制备方法和应用 |
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| CA2188772A1 (en) | 1994-06-08 | 1995-12-14 | Balreddy Kamireddy | Cyclic sulfonamide herbicides |
| SE0102147D0 (sv) | 2001-06-18 | 2001-06-18 | Pharmacia Ab | New methods |
| JP4518378B2 (ja) | 2001-10-29 | 2010-08-04 | ベーリンガー インゲルハイム インテルナツィオナール ゲゼルシャフト ミット ベシュレンクテル ハフツング | エネルギー恒常性および細胞小器官代謝の調節に関与するＭｎｋキナーゼ相同性タンパク質 |
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| GB0315587D0 (en) | 2003-07-03 | 2003-08-13 | Univ Dundee | Anti-inflammatory assay and compounds |
| US7678920B2 (en) | 2004-04-08 | 2010-03-16 | Dow Agrosciences Llc | Insecticidal N-substituted sulfoximines |
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| EP2004656B1 (en) * | 2006-04-07 | 2013-07-10 | Boehringer Ingelheim International GmbH | Thienopyrimidines having mnk1 /mnk2 inhibiting activity for pharmaceutical compositions |
| JP2009541268A (ja) | 2006-06-22 | 2009-11-26 | ビオヴィトルム・アクチボラゲット（プブリクト） | Ｍｎｋキナーゼ阻害剤としてのピリジンおよびピラジン誘導体 |
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| UY33241A (es) * | 2010-02-26 | 2011-09-30 | Boehringer Ingelheim Int | ?Tienopirimidinas que contienen heterocicloalquilo para composiciones farmacéuticas?. |
| UY33245A (es) | 2010-02-26 | 2011-09-30 | Boehringer Ingelheim Int | Tienopirimidinas que contienen un grupo alquilo sustituido para composiciones farmacéuticas |
| AR088082A1 (es) | 2011-10-13 | 2014-05-07 | Lilly Co Eli | Moduladores selectivos del receptor androgeno |
| ES2635262T3 (es) * | 2012-11-09 | 2017-10-03 | Evotec International Gmbh | Quinazolinas sustituidas con sulfoximina para composiciones farmacéuticas |
| WO2014206922A1 (en) * | 2013-06-28 | 2014-12-31 | Boehringer Ingelheim International Gmbh | Sulfoximine substituted quinazolines and their use as mnk1 and/or mnk2 kinase inhibitors |
-
2014
- 2014-11-28 WO PCT/EP2014/075890 patent/WO2015082324A1/en not_active Ceased
- 2014-11-28 JP JP2016536528A patent/JP6457523B2/ja not_active Expired - Fee Related
- 2014-11-28 EP EP14808895.8A patent/EP3077383B1/en active Active
- 2014-11-28 AU AU2014359456A patent/AU2014359456B2/en not_active Ceased
- 2014-11-28 US US15/101,620 patent/US10093660B2/en active Active
- 2014-11-28 ES ES14808895.8T patent/ES2693520T3/es active Active
- 2014-11-28 CA CA2929742A patent/CA2929742C/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| EP3077383B1 (en) | 2018-08-22 |
| US10093660B2 (en) | 2018-10-09 |
| JP6457523B2 (ja) | 2019-01-23 |
| AU2014359456A1 (en) | 2016-06-09 |
| EP3077383A1 (en) | 2016-10-12 |
| CA2929742C (en) | 2022-09-20 |
| AU2014359456B2 (en) | 2019-01-24 |
| US20170174668A1 (en) | 2017-06-22 |
| WO2015082324A1 (en) | 2015-06-11 |
| JP2016539148A (ja) | 2016-12-15 |
| CA2929742A1 (en) | 2015-06-11 |
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