ES2531149T3 - Derivados de 2-piridiniletilcarboxamida y su uso como fungicidas - Google Patents

Derivados de 2-piridiniletilcarboxamida y su uso como fungicidas Download PDF

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Publication number
ES2531149T3
ES2531149T3 ES05716432T ES05716432T ES2531149T3 ES 2531149 T3 ES2531149 T3 ES 2531149T3 ES 05716432 T ES05716432 T ES 05716432T ES 05716432 T ES05716432 T ES 05716432T ES 2531149 T3 ES2531149 T3 ES 2531149T3
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Spain
Prior art keywords
alkyl
halogen atoms
group
hydrogen atom
haloalkyl
Prior art date
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ES05716432T
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English (en)
Inventor
Darren James Mansfield
Heiko Rieck
Pierre-Yves Coqueron
Philippe Desbordes
Marie-Claire Grosjean-Cournoyer
Pierre Genix
Alain Villier
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Bayer Intellectual Property GmbH
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Bayer Intellectual Property GmbH
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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/561,2-Diazoles; Hydrogenated 1,2-diazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/781,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Un compuesto de fórmula general (I)**Fórmula** en la que: - n es 1, 2, 3 o 4; - X es igual o diferente, y es un átomo de halógeno, un alquilo C1-C8, un alcoxiimino C1-C6, un (alcoxiimino C1- C6)-alquilo C1-C6 o un alcoxi C1-C6-alquilcarbonilo-C1-C6; - R1 y R2 son iguales o diferentes, y son seleccionados, de manera independiente entre sí, entre un átomo de hidrógeno, un átomo de halógeno, un grupo ciano, un grupo hidroxi, un alquilo C1-C6, un halogenoalquilo C1-C6 que tiene de 1 a 5 átomos de halógeno, un alquenilo C2-C6, un alcoxi C1-C6, un alquilsulfanilo C1-C6, un alquilsulfenilo C1-C6, un alquilsulfinilo C1-C6, un alcoxicarbonilo C1-C6, un alquilcarbonilamino C1-C6, un alcoxicarboniloxi C1-C6, un alcoxicarbonilamino C1-C6 o un grupo fenilo; o R1 y R2 pueden formar juntos un ciclopropilo, un ciclobutilo, un ciclopentilo o un ciclohexilo; - R3 y R4 son iguales o diferentes, y son seleccionados, de manera independiente entre sí, entre un átomo de hidrógeno, un átomo de halógeno, un grupo ciano, un alquilo C1-C6, un halogenoalquilo C1-C6 que tiene de 1 a 5 átomos de halógeno o un grupo fenilo; con la condición de que cuando tres de los cuatro sustituyentes R1, R2, R3 y R4 sean un átomo de hidrógeno, entonces el cuarto sustituyente no sea un átomo de hidrógeno; - R5 es un átomo de hidrógeno, un grupo ciano, un grupo formilo, un grupo hidroxi, un alquilo C1-C6, un halogenoalquilo C1-C6 que tiene de 1 a 5 átomos de halógeno, un alcoxi C1-C6, un halogenoalcoxi C1-C6 que tiene de 1 a 5 átomos de halógeno, un cicloalquilo C3-C6, un halogenocicloalquilo C3-C6 que tiene de 1 a 5 átomos de halógeno, un alquenilo C2-C6, un alquinilo C2-C6, un alcoxi C1-C6-alquilo C1-C6, un cianoalquilo C1-C6, un aminoalquilo C1-C6, un alquilamino C1-C6-alquilo C1-C6, un di-alquilamino-C1-C6-alquilo C1-C6, un alquilcarbonilo C1-C6, un halogenalquilcarbonilo C1-C6 que tiene de 1 a 5 átomos de halógeno, un alquiloxicarbonilo C1-C6, un benciloxicarbonilo C1-C6, un alcoxi C1-C6-alquilcarbonilo C1-C6, un alquilsulfonilo C1- C6 o un halogenoalquilsulfonilo C1-C6 que tiene de 1 a 5 átomos de halógeno; - Het representa:**Fórmula** en la que: - R6 y R7 pueden ser iguales o diferentes, y pueden ser un átomo de hidrógeno, un átomo de halógeno, un grupo amino, un grupo nitro, un alquilo C1-C4 o un halogenoalquilo C1-C4 que tiene de 1 a 5 átomos de halógeno; y - R8 puede ser un átomo de halógeno, un grupo nitro, un alquilo C1-C4 o un halogenoalquilo C1-C4 que tiene de 1 a 5 átomos de halógeno.**Fórmula**
ES05716432T 2004-03-03 2005-03-01 Derivados de 2-piridiniletilcarboxamida y su uso como fungicidas Active ES2531149T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04356029A EP1574511A1 (en) 2004-03-03 2004-03-03 2-Pyridinylethylcarboxamide derivatives and their use as fungicides
PCT/EP2005/003282 WO2005085238A1 (en) 2004-03-03 2005-03-01 2-pyridinylethylcarboxamide derivatives and their use as fungicides

Publications (1)

Publication Number Publication Date
ES2531149T3 true ES2531149T3 (es) 2015-03-11

Family

ID=34814434

Family Applications (1)

Application Number Title Priority Date Filing Date
ES05716432T Active ES2531149T3 (es) 2004-03-03 2005-03-01 Derivados de 2-piridiniletilcarboxamida y su uso como fungicidas

Country Status (12)

Country Link
US (1) US7723363B2 (es)
EP (2) EP1574511A1 (es)
JP (1) JP4769789B2 (es)
KR (1) KR101234362B1 (es)
CN (1) CN1926134B (es)
BR (1) BRPI0506565A (es)
CA (1) CA2553252C (es)
DK (1) DK1720865T3 (es)
ES (1) ES2531149T3 (es)
IL (1) IL177263A (es)
WO (1) WO2005085238A1 (es)
ZA (1) ZA200606678B (es)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2866886B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives d'aryl-et d'heteroaryl-akylcarbamates, leur preparation et leur application en therapeutique
JP4869251B2 (ja) * 2004-12-21 2012-02-08 バイエル・クロップサイエンス・アーゲー 2−ピリジルエチルカルボキサミド誘導体の調製方法
TWI435863B (zh) * 2006-03-20 2014-05-01 Nihon Nohyaku Co Ltd N-2-(雜)芳基乙基甲醯胺衍生物及含該衍生物之蟲害防治劑
JP5065384B2 (ja) 2006-06-16 2012-10-31 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト 殺微生物剤として有用なエテニルカルボキサミド誘導体
WO2008003741A1 (en) * 2006-07-06 2008-01-10 Bayer Cropscience Sa N- [ (pyridin- 2 -yl) methoxy]heterocyclyl carboxamide derivatives and related compounds as fungicides
JP2010506880A (ja) * 2006-10-18 2010-03-04 バイエル・クロツプサイエンス・エス・アー 殺菌剤としてのn−(3−ピリジン−2−イルプロピル)ベンズアミド誘導体
EP1992617A1 (en) * 2007-05-15 2008-11-19 Syngeta Participations AG Optically active ethyl amides
RU2010103102A (ru) * 2007-07-02 2011-08-10 Зингента Партисипейшнс Аг (Ch) Новые микробиоциды
EP2218717A1 (en) * 2009-02-17 2010-08-18 Bayer CropScience AG Fungicidal N-((HET)Arylethyl)thiocarboxamide derivatives
ES2533026T3 (es) 2010-06-03 2015-04-07 Bayer Intellectual Property Gmbh N-[(het)arilalquil)]pirazol (tio)carboxamidas y sus análogos heterosustituidos
WO2012129491A1 (en) * 2011-03-24 2012-09-27 Abbott Laboratories Trpv3 modulators
EP2606727A1 (en) 2011-12-21 2013-06-26 Bayer CropScience AG Compounds with nematicidal activity
EP2589292A1 (en) 2011-11-02 2013-05-08 Bayer CropScience AG Compounds with nematicidal activity
CA2853876A1 (en) 2011-11-02 2013-05-10 Bayer Intellectual Property Gmbh Compounds with nematicidal activity
MX2014004849A (es) 2011-11-02 2014-08-27 Bayer Ip Gmbh Compuesto con actividad nematicida.
EP2606728A1 (en) 2011-12-21 2013-06-26 Bayer CropScience AG Compounds with nematicidal activity
EP2589294A1 (en) 2011-11-02 2013-05-08 Bayer CropScience AG Compounds with nematicidal activity
PT2782565T (pt) 2011-11-25 2020-01-07 Bayer Ip Gmbh Utilização de aril- e hetaril-carboxamidas como endoparasiticidas
US8815772B2 (en) 2012-06-29 2014-08-26 E I Du Pont De Nemours And Company Fungicidal heterocyclic carboxamides
TWI654180B (zh) * 2012-06-29 2019-03-21 美商艾佛艾姆希公司 殺真菌之雜環羧醯胺
EP2730570A1 (de) * 2012-11-13 2014-05-14 Bayer CropScience AG Pyridyloxyalkylcarboxamide und deren Verwendung als Endoparasitizide und Nematizide
WO2014177514A1 (en) * 2013-04-30 2014-11-06 Bayer Cropscience Ag Nematicidal n-substituted phenethylcarboxamides
UY35772A (es) 2013-10-14 2015-05-29 Bayer Cropscience Ag Nuevos compuestos plaguicidas
JPWO2015125824A1 (ja) * 2014-02-18 2017-03-30 日産化学工業株式会社 アルキニルピリジン置換アミド化合物及び有害生物防除剤

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GB8332704D0 (en) 1983-12-07 1984-01-11 Pfizer Ltd Growth promotants for animals
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WO2001005769A2 (en) * 1999-07-20 2001-01-25 Dow Agrosciences Llc Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
KR100718863B1 (ko) * 1999-08-18 2007-05-16 바이엘 크롭사이언스 게엠베하 살진균제
GB9930750D0 (en) * 1999-12-29 2000-02-16 Novartis Ag Organic compounds
GB0001447D0 (en) * 2000-01-21 2000-03-08 Novartis Ag Organic compounds
DK1531673T3 (da) * 2002-08-12 2006-03-06 Bayer Cropscience Sa Hidtil ukendt 2-pyridylethylbenzamidderivat
EP1449841A1 (en) * 2003-02-19 2004-08-25 Bayer CropScience SA New fungicidal compounds

Also Published As

Publication number Publication date
US7723363B2 (en) 2010-05-25
IL177263A0 (en) 2006-12-10
EP1720865A1 (en) 2006-11-15
KR101234362B1 (ko) 2013-02-18
EP1720865B1 (en) 2014-12-31
CA2553252A1 (en) 2005-09-15
CN1926134B (zh) 2011-09-21
CN1926134A (zh) 2007-03-07
JP2007526279A (ja) 2007-09-13
US20070167491A1 (en) 2007-07-19
IL177263A (en) 2011-10-31
DK1720865T3 (en) 2015-03-02
EP1574511A1 (en) 2005-09-14
CA2553252C (en) 2014-05-13
JP4769789B2 (ja) 2011-09-07
BRPI0506565A (pt) 2007-04-17
KR20060130144A (ko) 2006-12-18
ZA200606678B (en) 2008-02-27
WO2005085238A1 (en) 2005-09-15

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