ES2471872T3 - Procedimiento para la preparación de compuestos de aminoarilalquilo - Google Patents

Procedimiento para la preparación de compuestos de aminoarilalquilo Download PDF

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Publication number
ES2471872T3
ES2471872T3 ES11175821.5T ES11175821T ES2471872T3 ES 2471872 T3 ES2471872 T3 ES 2471872T3 ES 11175821 T ES11175821 T ES 11175821T ES 2471872 T3 ES2471872 T3 ES 2471872T3
Authority
ES
Spain
Prior art keywords
aryl
alkyl
arylalkyl
compounds
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
ES11175821.5T
Other languages
English (en)
Spanish (es)
Inventor
Michael Sander
Wolfgang Stirner
Frank Laschinski
Michael Konrad
Karsten Von Dem Bruch
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Saltigo GmbH
Original Assignee
Saltigo GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Saltigo GmbH filed Critical Saltigo GmbH
Application granted granted Critical
Publication of ES2471872T3 publication Critical patent/ES2471872T3/es
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES11175821.5T 2010-08-06 2011-07-28 Procedimiento para la preparación de compuestos de aminoarilalquilo Active ES2471872T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102010033690 2010-08-06
DE102010033690A DE102010033690A1 (de) 2010-08-06 2010-08-06 Verfahren zur Herstellung vom Aminoarylalkylverbindungen

Publications (1)

Publication Number Publication Date
ES2471872T3 true ES2471872T3 (es) 2014-06-27

Family

ID=44587696

Family Applications (1)

Application Number Title Priority Date Filing Date
ES11175821.5T Active ES2471872T3 (es) 2010-08-06 2011-07-28 Procedimiento para la preparación de compuestos de aminoarilalquilo

Country Status (6)

Country Link
US (1) US20120071662A1 (enExample)
EP (1) EP2415762B1 (enExample)
JP (1) JP2012062307A (enExample)
DE (1) DE102010033690A1 (enExample)
ES (1) ES2471872T3 (enExample)
PL (1) PL2415762T3 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20160145780A (ko) 2014-04-24 2016-12-20 노파르티스 아게 포스파티딜이노시톨 3-키나제 억제제로서의 아미노 피리딘 유도체
AU2014391610B2 (en) 2014-04-24 2018-01-25 Novartis Ag Pyrazine derivatives as phosphatidylinositol 3-kinase inhibitors
CA2945212A1 (en) 2014-04-24 2015-10-29 Novartis Ag Amino pyrazine derivatives as phosphatidylinositol 3-kinase inhibitors
CN107266357B (zh) * 2017-08-08 2018-07-17 九江善水科技股份有限公司 一种2,3-二氯吡啶的合成方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL112249A (en) * 1994-01-25 2001-11-25 Warner Lambert Co Pharmaceutical compositions containing di and tricyclic pyrimidine derivatives for inhibiting tyrosine kinases of the epidermal growth factor receptor family and some new such compounds
US7026478B2 (en) * 2002-05-10 2006-04-11 Studiengesellschaft Kohle Mbh Iron catalyzed cross coupling reactions of aromatic compounds
BRPI0417687A (pt) * 2003-12-19 2007-04-03 Pfizer derivados de benzenossulfonilamino-piridin-2-ila e compostos relacionados como inibidores de 11-beta-hidroxiesteróide desidrogenase tipo 1 (11-beta-hsd-1) para o tratamento de diabetes e obesidade
JP2006117568A (ja) * 2004-10-20 2006-05-11 Mitsubishi Pharma Corp チオフェン環を有する新規アミド誘導体及びその医薬としての用途
JP5203696B2 (ja) 2005-02-07 2013-06-05 田辺三菱製薬株式会社 光学活性なテトラヒドロナフタレン誘導体
JP5166747B2 (ja) 2007-03-09 2013-03-21 広栄化学工業株式会社 アルキルアミノピリジン類の精製方法
JP2010531358A (ja) * 2007-06-27 2010-09-24 メルク・シャープ・エンド・ドーム・コーポレイション ヒストン脱アセチル化酵素阻害剤としてのピリジル及びピリミジニル誘導体
US7928140B2 (en) * 2007-08-02 2011-04-19 Amgen Inc. Benzothiazole PI3 kinase modulators for cancer treatment

Also Published As

Publication number Publication date
EP2415762A3 (de) 2012-03-14
EP2415762B1 (de) 2014-04-23
PL2415762T3 (pl) 2014-11-28
DE102010033690A1 (de) 2012-02-09
JP2012062307A (ja) 2012-03-29
US20120071662A1 (en) 2012-03-22
EP2415762A2 (de) 2012-02-08

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