ES2339791T3 - Ciclizacion de peptidos sobre resina. - Google Patents

Ciclizacion de peptidos sobre resina. Download PDF

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Publication number
ES2339791T3
ES2339791T3 ES05796237T ES05796237T ES2339791T3 ES 2339791 T3 ES2339791 T3 ES 2339791T3 ES 05796237 T ES05796237 T ES 05796237T ES 05796237 T ES05796237 T ES 05796237T ES 2339791 T3 ES2339791 T3 ES 2339791T3
Authority
ES
Spain
Prior art keywords
peptide
cysteine
resin
amino acid
solid phase
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES05796237T
Other languages
English (en)
Spanish (es)
Inventor
Stephane Varray
Oleg Werbitzky
Thomas Zeiter
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Lonza AG
Original Assignee
Lonza AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza AG filed Critical Lonza AG
Application granted granted Critical
Publication of ES2339791T3 publication Critical patent/ES2339791T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Polyamides (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ES05796237T 2004-10-19 2005-10-18 Ciclizacion de peptidos sobre resina. Expired - Lifetime ES2339791T3 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP04024813 2004-10-19
EP04024813 2004-10-19
EP05008979 2005-04-25
EP05008979 2005-04-25

Publications (1)

Publication Number Publication Date
ES2339791T3 true ES2339791T3 (es) 2010-05-25

Family

ID=36096370

Family Applications (1)

Application Number Title Priority Date Filing Date
ES05796237T Expired - Lifetime ES2339791T3 (es) 2004-10-19 2005-10-18 Ciclizacion de peptidos sobre resina.

Country Status (16)

Country Link
US (1) US7994280B2 (enExample)
EP (1) EP1805203B1 (enExample)
JP (1) JP4927746B2 (enExample)
KR (2) KR101222774B1 (enExample)
CN (1) CN101111510B (enExample)
AT (1) ATE455123T1 (enExample)
AU (1) AU2005298991B2 (enExample)
BR (1) BRPI0516929A (enExample)
CA (1) CA2588098A1 (enExample)
DE (1) DE602005018952D1 (enExample)
DK (1) DK1805203T3 (enExample)
ES (1) ES2339791T3 (enExample)
IL (1) IL182575A (enExample)
PT (1) PT1805203E (enExample)
TW (1) TW200628487A (enExample)
WO (1) WO2006045483A2 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101538316B (zh) * 2009-01-13 2012-09-05 深圳翰宇药业股份有限公司 一种固相法制备Eptifibatide的方法
WO2013112548A1 (en) * 2012-01-23 2013-08-01 University Of South Florida Gamma-aapeptides with potent and broad-spectrum antimicrobial activity
CN108218964A (zh) * 2018-01-30 2018-06-29 江南大学 一种固相载体上酶法合成环肽方法
WO2024234959A1 (en) * 2023-05-18 2024-11-21 Versitech Limited Late-stage peptide cyclization to form disulfide mimetics

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4606856A (en) * 1985-03-18 1986-08-19 Seyler Jay K [Des-1-amino, 8-glycine]calcitonin
US5770687A (en) * 1995-06-07 1998-06-23 Peptor Limited Comformationally constrained backbone cyclized somatostatin analogs
WO2003093302A2 (en) * 2002-05-03 2003-11-13 Avecia Limited Process for the synthesis of peptides amides by side-chain attachement to a solid phase
CN1222537C (zh) * 2002-11-14 2005-10-12 吉尔生化（上海）有限公司 一种制备依非巴特的工艺
WO2004092202A1 (en) 2003-04-07 2004-10-28 Novetide, Ltd. Process for production of cyclic peptides
EP1756141B1 (en) 2004-06-14 2009-12-09 USV Ltd. Process for the preparation of peptides
CN100500805C (zh) * 2006-11-07 2009-06-17 武汉钢铁集团鄂城钢铁有限责任公司 除尘焦粉回配煤炼焦方法及其工艺

Also Published As

Publication number Publication date
WO2006045483A3 (en) 2006-07-13
DK1805203T3 (da) 2010-05-17
IL182575A0 (en) 2007-07-24
KR20070084099A (ko) 2007-08-24
WO2006045483A2 (en) 2006-05-04
AU2005298991B2 (en) 2011-03-03
PT1805203E (pt) 2010-04-19
JP4927746B2 (ja) 2012-05-09
BRPI0516929A (pt) 2008-09-23
TW200628487A (en) 2006-08-16
US20080200647A1 (en) 2008-08-21
US7994280B2 (en) 2011-08-09
AU2005298991A1 (en) 2006-05-04
KR101222774B1 (ko) 2013-01-15
EP1805203A2 (en) 2007-07-11
ATE455123T1 (de) 2010-01-15
CN101111510A (zh) 2008-01-23
CA2588098A1 (en) 2006-05-04
KR101276463B1 (ko) 2013-06-19
DE602005018952D1 (de) 2010-03-04
KR20120088855A (ko) 2012-08-08
JP2008517016A (ja) 2008-05-22
EP1805203B1 (en) 2010-01-13
CN101111510B (zh) 2011-09-14
IL182575A (en) 2012-07-31

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