ES2170101T3 - Compuesto ciclodepsipeptido. - Google Patents
Compuesto ciclodepsipeptido.Info
- Publication number
- ES2170101T3 ES2170101T3 ES94925614T ES94925614T ES2170101T3 ES 2170101 T3 ES2170101 T3 ES 2170101T3 ES 94925614 T ES94925614 T ES 94925614T ES 94925614 T ES94925614 T ES 94925614T ES 2170101 T3 ES2170101 T3 ES 2170101T3
- Authority
- ES
- Spain
- Prior art keywords
- compound
- salt
- lower alkyl
- cyclodepsipeptide
- cyclodepsipeptide compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 150000001875 compounds Chemical class 0.000 title abstract 3
- 108010002156 Depsipeptides Proteins 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 230000000590 parasiticidal effect Effects 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 241001465754 Metazoa Species 0.000 abstract 1
- 230000000507 anthelmentic effect Effects 0.000 abstract 1
- 229940124339 anthelmintic agent Drugs 0.000 abstract 1
- 239000000921 anthelmintic agent Substances 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 239000002297 parasiticide Substances 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biophysics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Manufacture Of Tobacco Products (AREA)
- Dental Preparations (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
UN COMPUESTO DE LA FORMULA: EN DONDE A ES UN GRUPO DE BENCILO QUE TIENE UN SUSTITUYENTE(S) ADECUADO (S), A{SUP,A}, B Y D SON CADA UNO ALQUILO BAJO, C ES HIDROGENO O ALQUILO BAJO, O UNA SAL DE LOS MISMOS. EL COMPUESTO O SU SAL DE LA PRESENTE INVENCION TIENE EXCELENTES ACTIVIDADES PARASITICIDAS COMO PARASITICIDAS (ANTIHELMINTICAS) PARA ANIMALES Y CUERPOS HUMANOS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP24632393 | 1993-09-06 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2170101T3 true ES2170101T3 (es) | 2002-08-01 |
Family
ID=17146855
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES94925614T Expired - Lifetime ES2170101T3 (es) | 1993-09-06 | 1994-08-31 | Compuesto ciclodepsipeptido. |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US5646244A (es) |
| EP (1) | EP0718293B1 (es) |
| JP (1) | JP3263947B2 (es) |
| KR (1) | KR100392172B1 (es) |
| CN (1) | CN1061039C (es) |
| AT (1) | ATE214379T1 (es) |
| AU (1) | AU686222B2 (es) |
| BR (1) | BR9407711A (es) |
| CA (1) | CA2171088A1 (es) |
| DE (1) | DE69430128T2 (es) |
| DK (1) | DK0718293T3 (es) |
| ES (1) | ES2170101T3 (es) |
| NZ (1) | NZ271739A (es) |
| PT (1) | PT718293E (es) |
| TW (1) | TW318844B (es) |
| WO (1) | WO1995007272A1 (es) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE69637876D1 (de) * | 1995-06-30 | 2009-04-30 | Astellas Pharma Inc | Ng und zwischenprodukt dafür |
| AU6860296A (en) * | 1995-09-07 | 1997-03-27 | Pharmacia & Upjohn Company | Cycloanthelmintic inhibitors |
| ATE237583T1 (de) | 1996-10-07 | 2003-05-15 | Fujisawa Pharmaceutical Co | Verfahren zur herstellung von depsipeptiden und zwischenprodukten davon |
| DE19713626A1 (de) | 1997-04-02 | 1998-10-08 | Bayer Ag | Neue Thiodepsipeptide zur Bekämpfung von Endoparasiten und ein einfaches Verfahren zu ihrer Herstellung |
| NZ501478A (en) * | 1997-06-04 | 2001-05-25 | Bayer Ag | 8,20-bis-(substituted benzyl)-desoxycyclodepsipeptides and their use for combatting endoparasites |
| CA2308067C (en) | 1997-11-10 | 2008-01-08 | Fujisawa Pharmaceutical Co., Ltd. | Novel crystals of depsipeptide derivative and a method for producing the same |
| DE19921887A1 (de) * | 1999-05-12 | 2000-11-16 | Bayer Ag | Endoparasitizide Mittel |
| DE19962145A1 (de) * | 1999-12-22 | 2001-06-28 | Bayer Ag | Schädlingsbekämpfungsmittel/Depsipeptide |
| DE19962147A1 (de) * | 1999-12-22 | 2001-06-28 | Bayer Ag | Schädlingsbekämpfungsmittel / PF 1022-221 |
| DE10031044A1 (de) * | 2000-06-26 | 2002-01-03 | Bayer Ag | Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere |
| DE102004055316A1 (de) * | 2004-11-16 | 2006-05-18 | Bayer Healthcare Ag | Verhinderung vertikaler Endoparasiten-Infektionen |
| DE102008022520A1 (de) * | 2008-05-07 | 2009-11-12 | Bayer Animal Health Gmbh | Feste Arzneimittelformulierung mit verzögerter Freisetzung |
| DE102008030764A1 (de) | 2008-06-28 | 2009-12-31 | Bayer Animal Health Gmbh | Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden |
| DE102008031283A1 (de) | 2008-07-02 | 2010-01-07 | Bayer Schering Pharma Aktiengesellschaft | Neue Bekämpfungsmöglichkeit von durch Trichomonadida hervorgerufenen Krankheiten |
| DE102008031284A1 (de) | 2008-07-02 | 2010-01-07 | Bayer Schering Pharma Aktiengesellschaft | Neue Bekämpfungsmöglichkeit der Giardiose |
| WO2010058423A2 (en) | 2008-11-20 | 2010-05-27 | Panacea Biotec Ltd. | Novel antimicrobials |
| DE102009012423A1 (de) | 2009-03-10 | 2010-09-16 | Bayer Animal Health Gmbh | Zubereitung auf Ölbasis |
| MX2012000231A (es) | 2009-06-26 | 2012-03-07 | Panacea Biotec Ltd | Nuevos aza-biciclo-hexanos. |
| DE102010064245A1 (de) | 2010-12-28 | 2012-06-28 | Bayer Animal Health Gmbh | Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen |
| WO2012028556A1 (en) | 2010-08-31 | 2012-03-08 | Bayer Animal Health Gmbh | Macrocyclic lactones and their use and their combinations with other active substances |
| SG10202103403SA (en) | 2015-05-20 | 2021-05-28 | Boehringer Ingelheim Animal Health Usa Inc | Anthelmintic depsipeptide compounds |
| SG11201805368YA (en) | 2015-12-28 | 2018-07-30 | Merial Inc | Anthelmintic depsipeptide compounds |
| EP3541789A1 (en) | 2016-11-16 | 2019-09-25 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintic depsipeptide compounds |
| MX2020005573A (es) | 2017-11-29 | 2020-09-10 | Zoetis Services Llc | Depsipeptidos endoparasitarios. |
| NZ769696A (en) | 2018-05-10 | 2023-12-22 | Zoetis Services Llc | Endoparasitic depsipeptides |
| BR112021013488A2 (pt) | 2019-01-10 | 2021-09-14 | Zoetis Services Llc | Modelo animal de laboratório antelmíntico para dirofilariose |
| EP4262789A1 (en) | 2020-12-21 | 2023-10-25 | Boehringer Ingelheim Vetmedica GmbH | Parasiticidal collar comprising isoxazoline compounds |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO176766C (no) * | 1989-02-07 | 1995-05-24 | Meiji Seika Kaisha | Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet |
| JP3207870B2 (ja) * | 1991-04-15 | 2001-09-10 | 明治製菓株式会社 | 環状デプシペプチドおよびその製造法 |
| DK0634408T3 (da) * | 1992-03-17 | 2002-04-22 | Fujisawa Pharmaceutical Co | Depsipeptidderivater, fremstilling og anvendelse deraf |
| WO1994019334A1 (en) * | 1993-02-19 | 1994-09-01 | Meiji Seika Kaisha, Ltd. | Pf1022 derivative, cyclic depsipeptide |
| DE4317457A1 (de) * | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
-
1994
- 1994-08-31 WO PCT/JP1994/001446 patent/WO1995007272A1/ja active IP Right Grant
- 1994-08-31 CA CA002171088A patent/CA2171088A1/en not_active Abandoned
- 1994-08-31 DK DK94925614T patent/DK0718293T3/da active
- 1994-08-31 AU AU75463/94A patent/AU686222B2/en not_active Ceased
- 1994-08-31 KR KR1019960701109A patent/KR100392172B1/ko not_active IP Right Cessation
- 1994-08-31 NZ NZ271739A patent/NZ271739A/en not_active IP Right Cessation
- 1994-08-31 PT PT94925614T patent/PT718293E/pt unknown
- 1994-08-31 CN CN94193914A patent/CN1061039C/zh not_active Expired - Fee Related
- 1994-08-31 US US08/605,064 patent/US5646244A/en not_active Expired - Fee Related
- 1994-08-31 JP JP50857795A patent/JP3263947B2/ja not_active Expired - Fee Related
- 1994-08-31 EP EP94925614A patent/EP0718293B1/en not_active Expired - Lifetime
- 1994-08-31 AT AT94925614T patent/ATE214379T1/de not_active IP Right Cessation
- 1994-08-31 DE DE69430128T patent/DE69430128T2/de not_active Expired - Fee Related
- 1994-08-31 BR BR9407711A patent/BR9407711A/pt not_active Application Discontinuation
- 1994-08-31 ES ES94925614T patent/ES2170101T3/es not_active Expired - Lifetime
- 1994-09-05 TW TW083108159A patent/TW318844B/zh active
Also Published As
| Publication number | Publication date |
|---|---|
| CN1133592A (zh) | 1996-10-16 |
| EP0718293B1 (en) | 2002-03-13 |
| BR9407711A (pt) | 1997-02-12 |
| CA2171088A1 (en) | 1995-03-16 |
| JP3263947B2 (ja) | 2002-03-11 |
| KR100392172B1 (ko) | 2004-04-03 |
| DK0718293T3 (da) | 2002-04-22 |
| NZ271739A (en) | 1996-09-25 |
| DE69430128D1 (en) | 2002-04-18 |
| EP0718293A4 (en) | 1997-04-16 |
| AU686222B2 (en) | 1998-02-05 |
| ATE214379T1 (de) | 2002-03-15 |
| WO1995007272A1 (en) | 1995-03-16 |
| EP0718293A1 (en) | 1996-06-26 |
| AU7546394A (en) | 1995-03-27 |
| DE69430128T2 (de) | 2002-09-05 |
| TW318844B (es) | 1997-11-01 |
| CN1061039C (zh) | 2001-01-24 |
| US5646244A (en) | 1997-07-08 |
| PT718293E (pt) | 2002-08-30 |
| KR960704868A (ko) | 1996-10-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
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