ES2167377T3 - Derivados de piridina farmacologicamente activos y procedimientos para la preparacion de los mismos. - Google Patents

Derivados de piridina farmacologicamente activos y procedimientos para la preparacion de los mismos.

Info

Publication number
ES2167377T3
ES2167377T3 ES94927635T ES94927635T ES2167377T3 ES 2167377 T3 ES2167377 T3 ES 2167377T3 ES 94927635 T ES94927635 T ES 94927635T ES 94927635 T ES94927635 T ES 94927635T ES 2167377 T3 ES2167377 T3 ES 2167377T3
Authority
ES
Spain
Prior art keywords
derivatives
piridina
procedures
preparation
same
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES94927635T
Other languages
English (en)
Inventor
Jurg Zimmermann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis AG filed Critical Novartis AG
Application granted granted Critical
Publication of ES2167377T3 publication Critical patent/ES2167377T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/28—Compounds containing heavy metals
    • A61K31/305—Mercury compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

SE DESCRIBEN DERIVADOS DE N-FENIL-2-PIRIMIDINEAMINA DE FORMULA (I) DONDE LOS SUSTITUYENTES SON COMO SE DEFINE EN LA SOLICITUD 1. ESOS COMPUESTOS PUEDEN SER UTILIZADOS, POR EJEMPLO, EN EL TRATAMIENTO DE ENFERMEDADES TUMORALES.
ES94927635T 1993-10-01 1994-09-21 Derivados de piridina farmacologicamente activos y procedimientos para la preparacion de los mismos. Expired - Lifetime ES2167377T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH296993 1993-10-01
CH228194 1994-07-18

Publications (1)

Publication Number Publication Date
ES2167377T3 true ES2167377T3 (es) 2002-05-16

Family

ID=25690002

Family Applications (1)

Application Number Title Priority Date Filing Date
ES94927635T Expired - Lifetime ES2167377T3 (es) 1993-10-01 1994-09-21 Derivados de piridina farmacologicamente activos y procedimientos para la preparacion de los mismos.

Country Status (21)

Country Link
US (1) US5728708A (es)
EP (1) EP0672041B1 (es)
JP (1) JP2983636B2 (es)
KR (1) KR100330553B1 (es)
CN (1) CN1047776C (es)
AT (1) ATE208772T1 (es)
AU (1) AU691834B2 (es)
CA (1) CA2148928C (es)
CZ (1) CZ290681B6 (es)
DE (1) DE69429078T2 (es)
DK (1) DK0672041T3 (es)
ES (1) ES2167377T3 (es)
FI (1) FI112227B (es)
HU (1) HU228172B1 (es)
IL (1) IL111077A (es)
NO (1) NO308794B1 (es)
NZ (1) NZ273617A (es)
PL (1) PL179417B1 (es)
PT (1) PT672041E (es)
RU (1) RU2135491C1 (es)
WO (1) WO1995009853A1 (es)

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TW225528B (es) * 1992-04-03 1994-06-21 Ciba Geigy Ag
US5516775A (en) * 1992-08-31 1996-05-14 Ciba-Geigy Corporation Further use of pyrimidine derivatives

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HUT72609A (en) 1996-05-28
US5728708A (en) 1998-03-17
RU2135491C1 (ru) 1999-08-27
FI952607A (fi) 1995-05-29
NO308794B1 (no) 2000-10-30
JPH08504215A (ja) 1996-05-07
DE69429078T2 (de) 2002-07-11
CA2148928C (en) 2005-10-18
CA2148928A1 (en) 1995-04-13
DE69429078D1 (de) 2001-12-20
AU691834B2 (en) 1998-05-28
NO952132L (no) 1995-05-30
CN1115982A (zh) 1996-01-31
CZ290681B6 (cs) 2002-09-11
CN1047776C (zh) 1999-12-29
PL179417B1 (en) 2000-09-29
NO952132D0 (no) 1995-05-30
EP0672041B1 (en) 2001-11-14
FI112227B (fi) 2003-11-14
PT672041E (pt) 2002-04-29
EP0672041A1 (en) 1995-09-20
KR100330553B1 (ko) 2002-11-27
JP2983636B2 (ja) 1999-11-29
CZ172295A3 (en) 1996-03-13
IL111077A0 (en) 1994-11-28
FI952607A0 (fi) 1995-05-29
NZ273617A (en) 1996-11-26
HU228172B1 (en) 2013-01-28
WO1995009853A1 (en) 1995-04-13
DK0672041T3 (da) 2002-02-25
PL309225A1 (en) 1995-10-02
KR950704296A (ko) 1995-11-17
ATE208772T1 (de) 2001-11-15
IL111077A (en) 1999-10-28
AU7697794A (en) 1995-05-01
HU9501953D0 (en) 1995-09-28

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