ES2066879T3 - Procedimiento para la obtencion de derivados de 3-fenilpirrol. - Google Patents

Procedimiento para la obtencion de derivados de 3-fenilpirrol.

Info

Publication number
ES2066879T3
ES2066879T3 ES89810918T ES89810918T ES2066879T3 ES 2066879 T3 ES2066879 T3 ES 2066879T3 ES 89810918 T ES89810918 T ES 89810918T ES 89810918 T ES89810918 T ES 89810918T ES 2066879 T3 ES2066879 T3 ES 2066879T3
Authority
ES
Spain
Prior art keywords
alkyl
phenyl
hydrogen
procedure
methyltium
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES89810918T
Other languages
English (en)
Inventor
Rudolf Walter Dr Pfluger
Jean Dr Indermuhle
Franz Dr Felix
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Application granted granted Critical
Publication of ES2066879T3 publication Critical patent/ES2066879T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/323—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to the ring nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Luminescent Compositions (AREA)

Abstract

EL INVENTO SE REFIERE A UN DERIVADO DE 3-FENILPIROL DE FORMULA (I) Y TRATA DE UN PROCEDIMIENTO PARA SU PRODUCCION QUE CONSISTE EN: TRATAR LA N-(P-TOLIOLSULFONILO)-METILFORMAMIDA CON CLORURO DE FOSFOROXI, EN UN DISOLVENTE INERTE Y EN PRESENCIA DE UNA BASE ORGANICA; DILUIR LA SOLUCION DE REACCION CON AGUA PARA SEPARAR LA FASE ACUOSA DE LA SOLUCION Y TRATAR LA FASE ORGANICA DE LA SOLUCION QUE CONTIENE P-TOLIOL(SULFONILO)-METILISOCIAMIDA CON UN COMPUESTO DE FORMULA (II) EN PRESENCIA DE UNA BASE. SIENDO: R1 Y R2 INDEPENDIENTE UNO DE OTRO, HIDROGENO, ALQUILO DE C 1 A 6, ALCOXI DE C 1 A 6, ALQUILTIO DE C 1 A 6, NITRO, CIANO, HALOGENO,HALOGENOALQUILO DE C 1 A 6; O R1 Y R2 METILENODOXI, O DIFLUOROMETILENODOXI; R3 ALQUILO DE C 1 A 6, FENILO O BENZIKO O FENILO SUSTITUIDO A TRAVES DE HALOGENO, METILO, METOXI O METILTIO O BENCILO, R4 HIDROGENO ALQUILO DE C 1 A 6, TENILO O BENCILO, FENILO SUSTITUIDO A TRAVES DE HALOGENO, METILO, METOXI, METILTIO O BENCILO; R5 ALQUILO DE C 1 A 6, HALOGENOALQUILO DE C 1 A6, FENILO OBENCILO, FENILO SUSTITUIDO A TRAVES D HIDROGENO, METILO, METOXI O METILTIO O BENCILO; X CIANO, -CO-R3, -CO-OR3, -CO-NH-R4; E Y -CO-NH-R4, -COR5 O -SR5.
ES89810918T 1988-12-12 1989-12-05 Procedimiento para la obtencion de derivados de 3-fenilpirrol. Expired - Lifetime ES2066879T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US28334188A 1988-12-12 1988-12-12
US07/419,793 US4958030A (en) 1988-12-12 1989-10-11 Process for the preparation of 3-phenylpyrrole derivatives

Publications (1)

Publication Number Publication Date
ES2066879T3 true ES2066879T3 (es) 1995-03-16

Family

ID=26961991

Family Applications (1)

Application Number Title Priority Date Filing Date
ES89810918T Expired - Lifetime ES2066879T3 (es) 1988-12-12 1989-12-05 Procedimiento para la obtencion de derivados de 3-fenilpirrol.

Country Status (6)

Country Link
US (1) US4958030A (es)
EP (1) EP0378046B1 (es)
JP (1) JPH0717598B2 (es)
AT (1) ATE117293T1 (es)
DE (1) DE58908916D1 (es)
ES (1) ES2066879T3 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5252746A (en) * 1990-12-11 1993-10-12 American Cyanamid Company Process for the preparation of insecticidal, nematicidal and acaricidal 2-halo-3-substituted-5-arylpyrrole compounds
US6204397B1 (en) 1991-03-08 2001-03-20 Bayer Aktiengesellschaft Process for the preparation of 3-substituted 4-cyano-pyrrole compounds
DE4107398A1 (de) * 1991-03-08 1992-11-05 Bayer Ag Verfahren zur herstellung von in 3-stellung substituierten 4-cyano-pyrrolverbindungen
JP4161367B2 (ja) 2001-03-23 2008-10-08 日本曹達株式会社 ５−置換オキサゾール化合物および５−置換イミダゾール化合物の製造方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0111452A1 (de) * 1982-12-10 1984-06-20 Ciba-Geigy Ag Verwendung von Pyrrolen als Biocide für den Materialschutz
US4546099A (en) * 1983-07-22 1985-10-08 Ciba-Geigy Corporation N-Aminomethyl-3-phenyl-4-cyanopyrrole derivatives, compositions and use thereof as microbicides
US4705801A (en) * 1984-10-16 1987-11-10 Ciba-Geigy Corporation Production for producing 3-cyano-4-phenyl indoles and intermediates
US4687861A (en) * 1984-11-28 1987-08-18 Ciba-Geigy Corporation Microbicidal compositions
US4705800A (en) * 1985-06-21 1987-11-10 Ciba-Geigy Corporation Difluorbenzodioxyl cyanopyrrole microbicidal compositions
US4680413A (en) * 1986-01-17 1987-07-14 Nippon Soda Co., Ltd. Process for the production of 3-phenyl-4-cyanopyrroles
JPS6430571A (en) * 1987-07-24 1989-02-01 Sanwa Kosan Kk Expanded food and preparation thereof
DE3800387A1 (de) * 1988-01-09 1989-07-20 Bayer Ag Verfahren zur herstellung von 3-cyano-4-aryl-pyrrolen
JPH06130571A (ja) * 1992-10-21 1994-05-13 Konica Corp 錠剤状ハロゲン化銀写真感光材料用漂白定着剤及び処理方法

Also Published As

Publication number Publication date
DE58908916D1 (de) 1995-03-02
US4958030A (en) 1990-09-18
EP0378046A1 (de) 1990-07-18
EP0378046B1 (de) 1995-01-18
JPH02202871A (ja) 1990-08-10
ATE117293T1 (de) 1995-02-15
JPH0717598B2 (ja) 1995-03-01

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