ES2061975T3 - Derivados de triazol, su preparacion y su uso como fungicidas. - Google Patents

Derivados de triazol, su preparacion y su uso como fungicidas.

Info

Publication number
ES2061975T3
ES2061975T3 ES89302244T ES89302244T ES2061975T3 ES 2061975 T3 ES2061975 T3 ES 2061975T3 ES 89302244 T ES89302244 T ES 89302244T ES 89302244 T ES89302244 T ES 89302244T ES 2061975 T3 ES2061975 T3 ES 2061975T3
Authority
ES
Spain
Prior art keywords
optionally
formula
fungicides
substituted phenyl
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES89302244T
Other languages
English (en)
Inventor
Sadao Oida
Yawara Tajima
Toshiyuki Konosu
Masayuki Iwata
Noriko Takeda
Takeo Miyaoka
Hideo Takeshiba
Toshiro Nakanishi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sankyo Co Ltd
Original Assignee
Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co Ltd filed Critical Sankyo Co Ltd
Application granted granted Critical
Publication of ES2061975T3 publication Critical patent/ES2061975T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/24—Halogenated aromatic hydrocarbons with unsaturated side chains
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46—Friedel-Crafts reactions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/82—Ketones containing a keto group bound to a six-membered aromatic ring containing hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

COMPUESTOS DE FORMULA(I), DONDE AR ES OPCIONALMENTE UN FENILO SUSTITUIDO; R1 ES H O ALQUILO; X ES OPCIONALMENTE UN ALQUILENO INSATURADO, CICLOALQUILENO O AMBOS; M ES 0 O 1; - YN - R2 ES ACIDO, FTALIMIDO, 1 - OXO - 2,3 - DIHIDRURO - 2 - ISOINDOLIL, HIDROXI PROTEGIDO O - OSO2R4 (EN DONDE R4 ES UN GRUPO ALQUILO, HALOALQUILO U OPCIONALMENTE UN FENILO SUSTITUIDO); O Y REPRESENTA UN GRUPO DE FORMULA - N(R5)CO -, - N(R5)CO - CH = CH -, O - CO -, - O - CO - CH = CH, - S - CO O - S - CO - CH = CH - (EN DONDE R5 ES H O ALQUILO); N ES 0 O 1; R2 ES ALQUILO, HALOALQUILO U OPCIONALMENTE FENILO SUSTITUIDO, NAFTILO O HETEROCICLICO; Y R3 ES H; O R3 Y - XM - YN R2 JUNTOS SON UN GRUPO DE FORMULA(II), DONDE R2 ES COMO SE DEFINE ARRIBA, Q ES 0 O 1, Y P ES 0 O 1; Y SALES DE ADICION ACIDAS DE ESTO SON FUNGICIDAS, Y SON DE CONSIDERABLE VALOR EN LA ERRADICACION DE HONGOS EN LA AGRICULTURA Y LA MEDICINA.
ES89302244T 1988-03-04 1989-03-06 Derivados de triazol, su preparacion y su uso como fungicidas. Expired - Lifetime ES2061975T3 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP5131288 1988-03-04
JP6868188 1988-03-23
JP25015888 1988-10-04
JP26121188 1988-10-17

Publications (1)

Publication Number Publication Date
ES2061975T3 true ES2061975T3 (es) 1994-12-16

Family

ID=27462619

Family Applications (1)

Application Number Title Priority Date Filing Date
ES89302244T Expired - Lifetime ES2061975T3 (es) 1988-03-04 1989-03-06 Derivados de triazol, su preparacion y su uso como fungicidas.

Country Status (11)

Country Link
EP (1) EP0332387B1 (es)
KR (1) KR890014500A (es)
AU (1) AU622639B2 (es)
DE (1) DE68910853T2 (es)
DK (1) DK105189A (es)
ES (1) ES2061975T3 (es)
FI (1) FI97382C (es)
HU (1) HUT53889A (es)
IE (1) IE64189B1 (es)
NO (1) NO171272C (es)
NZ (1) NZ228236A (es)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8819308D0 (en) * 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents
US5206364A (en) * 1988-08-13 1993-04-27 Pfizer Inc. Triazole antifungal agents
IE903395A1 (en) * 1989-09-26 1991-04-10 Takeda Chemical Industries Ltd Triazole compounds, their production and use
TW206224B (es) * 1989-12-14 1993-05-21 Takeda Pharm Industry Co Ltd
CA2031892C (en) * 1989-12-25 2000-08-01 Minoru Tokizawa Triazole derivatives
US5278175A (en) * 1990-02-02 1994-01-11 Pfizer Inc. Triazole antifungal agents
GB9002375D0 (en) * 1990-02-02 1990-04-04 Pfizer Ltd Triazole antifungal agents
US5387599A (en) * 1990-03-15 1995-02-07 Takeda Chemical Industries, Ltd. Triazoles, their production and use
IT1240676B (it) * 1990-04-24 1993-12-17 Agrimont Spa Composizioni ad attivita' erbicida
ES2024332A6 (es) * 1990-10-08 1992-02-16 Uriach & Cia Sa J Procedimiento para la obtencion de nuevas sulfonamidas.
IL101372A0 (en) * 1991-03-27 1992-11-15 Schering Corp Preparation of chiral hydroxyketones
WO1992017433A1 (en) * 1991-03-27 1992-10-15 Schering Corporation Preparation of chiral hydroxyketones
KR920019763A (ko) * 1991-04-26 1992-11-19 모리다 가즈라 아졸 화합물, 그의 제조방법 및 용도
ES2038906B1 (es) * 1991-09-04 1994-02-16 Uriach & Cia Sa J Procedimiento para la obtencion de nuevas oxazoilidinas.
GB9121456D0 (en) * 1991-10-10 1991-11-27 Pfizer Ltd Triazole antifungal agents
US5426233A (en) * 1992-03-25 1995-06-20 Schering Corporation Preparation of chiral hydroxyketones
TW218017B (es) * 1992-04-28 1993-12-21 Takeda Pharm Industry Co Ltd
ES2051226B1 (es) * 1992-07-15 1994-12-16 Uriach & Cia Sa J Procedimiento para la obtencion del (-)-(2r,3r)-2-(2,4-diclorofenil)-3-(n-metanosulfonil-n-metilamino)-1-(1h-1,2,4-triazol-1-il)-2-butanol.
ES2099004B1 (es) * 1993-02-11 1998-01-16 Uriach & Cia Sa J Nuevos antifungicos activos por via oral.
ES2062941B1 (es) * 1993-03-15 1995-10-01 Uriach & Cia Sa J Nuevos derivados de azol activos por via oral.
TW297813B (es) * 1993-09-24 1997-02-11 Takeda Pharm Industry Co Ltd
US5349099A (en) * 1993-12-13 1994-09-20 Schering Corporation Process for preparing intermediates for the synthesis of antifungal agents
NZ270418A (en) * 1994-02-07 1997-09-22 Eisai Co Ltd Polycyclic triazole & imidazole derivatives, antifungal compositions
CA2145458A1 (en) * 1994-03-28 1995-09-29 Hiroki Kodama Triazole compound and production process and use thereof
WO1995034542A1 (fr) * 1994-06-10 1995-12-21 Tokyo Tanabe Company Limited Compose de triazole et agent antifongique contenant ledit compose en tant qu'ingredient actif
TW318841B (es) * 1995-02-17 1997-11-01 Takeda Pharm Industry Co Ltd
WO1996031491A1 (fr) * 1995-04-06 1996-10-10 Sankyo Company, Limited Agent antifongique de triazole
CA2180091A1 (en) * 1995-07-08 1997-01-09 Hiroki Kodama Optically active triazole derivative, process for producing the same, antifungal agent, and method for using the same
ES2112774B1 (es) * 1995-10-20 1999-05-16 Uriach & Cia Sa J Nuevos derivados azolicos con actividad antifungica.
JPH10507205A (ja) * 1995-08-02 1998-07-14 ホータ．ウリアッヒ イ シイア．エセ．アー． 抗真菌活性を有する新規カルボンアミド
US6133485A (en) * 1998-04-15 2000-10-17 Synphar Laboratories, Inc. Asymmetric synthesis of 2-(2,4-difluorophenyl)-1-heterocycl-1-yl butan-2,3-diols
GB9924692D0 (en) 1999-10-20 1999-12-22 Hoechst Schering Agrevo Gmbh Wood treatment
AU2007201000B2 (en) * 2000-09-05 2008-07-03 Donaldson Company, Inc. Polymer fine fiber and fine fiber layer
ATE508122T1 (de) * 2003-07-18 2011-05-15 Kaneka Corp Optisch aktives halogenhydrinderivat und verfahren zur herstellung eines optisch aktiven epoxyalkoholderivats davon
WO2007123853A2 (en) * 2006-04-20 2007-11-01 E. I. Du Pont De Nemours And Company Five-membered heterocyclic invertebrate pest control agents
WO2019216810A1 (en) * 2018-05-07 2019-11-14 Constantin Urban New antifungal compounds

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4654332A (en) * 1979-03-07 1987-03-31 Imperial Chemical Industries Plc Heterocyclic compounds
US4482558A (en) * 1982-06-18 1984-11-13 Pfizer Inc. Antifungal amide and urea derivatives of (3-amino-2-aryl-2-hydroxyprop-1-yl)-1H-1,2,4-triazoles
DE3307218A1 (de) * 1983-03-02 1984-09-06 Bayer Ag, 5090 Leverkusen Substituierte diazolylalkyl-carbinole, verfahren zu ihrer herstellung und ihre verwendung als antimykotische mittel
CH658654A5 (de) * 1983-03-04 1986-11-28 Sandoz Ag Azolderivate, verfahren zu ihrer herstellung und mittel die diese verbindungen enthalten.
GB8306351D0 (en) * 1983-03-08 1983-04-13 Ici Plc Azole fungicides
US4483863A (en) * 1984-01-20 1984-11-20 Pfizer Inc. Triazole antifungal agents
GB8412750D0 (en) * 1984-05-18 1984-06-27 Ici Plc Heterocyclic compounds
DE3530799A1 (de) * 1985-08-29 1987-03-05 Hoechst Ag Azolyl-cyclopropyl-ethanol-derivate, verfahren zu ihrer herstellung und ihre verwendung
GB8819308D0 (en) * 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents

Also Published As

Publication number Publication date
IE64189B1 (en) 1995-07-12
NZ228236A (en) 1991-02-26
HUT53889A (en) 1990-12-28
AU622639B2 (en) 1992-04-16
KR890014500A (ko) 1989-10-24
NO171272C (no) 1993-02-17
AU3105189A (en) 1989-09-07
EP0332387A1 (en) 1989-09-13
DK105189A (da) 1989-09-05
FI891021A (fi) 1989-09-05
IE890712L (en) 1989-09-04
EP0332387B1 (en) 1993-11-24
FI97382B (fi) 1996-08-30
FI891021A0 (fi) 1989-03-03
DK105189D0 (da) 1989-03-03
NO890926D0 (no) 1989-03-03
DE68910853D1 (de) 1994-01-05
NO890926L (no) 1989-09-05
NO171272B (no) 1992-11-09
FI97382C (fi) 1996-12-10
DE68910853T2 (de) 1994-06-30

Similar Documents

Publication Publication Date Title
ES2061975T3 (es) Derivados de triazol, su preparacion y su uso como fungicidas.
EG18551A (en) Derivatives of acylic acid useful as fungicides insecticides,nematocides and plant growth regulators
HUT55951A (en) Fungicidal compositions comprising acrylic acid derivatives as active ingredient and process for producing the active ingredient
ES8701707A1 (es) Procedimiento para preparar derivados del acido acrilico conactividad fungicida
EP0378254A3 (en) 2-aminopyrimidinone derivatives
IL62905A0 (en) Aminopropiophenone derivatives,their preparation and their use as fungicides
EP0350237A3 (en) Triazole insecticides
MA20968A1 (fr) Compositions bactericides a base de derives de l'acide phosphoreux
EP0191724A3 (de) 1,4-Dihydropyridine, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zusammensetzungen
FR2515175B1 (fr) Nouveaux derives de l'acide 4-phenyl 4-oxo 2-butenoique, leurs sels, leur preparation, leur application comme medicaments et les compositions les renfermant
DK545385A (da) Triazolforbindelser, farmaceutiske praeparater og landbrugsfungicider indeholdende disse og fremgangsmaade til behandling af planter eller froe mod svampeinfektion
ATE84209T1 (de) Hautreinigungsmittel.
EP0315433A3 (en) 3-amino-5-methyl-1h-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics
NO883520L (no) Fremgangsmaate for fremstilling av et injeksjonspreparat.
ES8504434A1 (es) Procedimiento para preparar una composicion fungicida a base de una sal de acido alquil-fosforoso
IT1150707B (it) Metodo per la difesa di colture di interesse agrario dall'azione di erbicidi non selettivi
BG34607A3 (en) Fungicide means
NZ211736A (en) Beta-naphthylalkylamine derivatives and plant fungicidal compositions
GR880100854A (el) Υδατικές διαμορφώσεις που περιέχουν ενα παράγωγο πιπεριδινυλκυκλοπεντυλεπτενοικού οξέος.
BG79417A (bg) Съединения,съдържащи триазолова или имидазолова,тетрахидрофуранова и фенилна група,метод за тяхното получаване и приложение
ATE82861T1 (de) Physiologisch aktive, fluessige, allergenische zusammensetzungen aus biologischen rohmaterialien.
DK404584A (da) Triazolderivater og deres anvendelse som antifungale midler i farmaceutiske praeparater eller landbrugsfungicider
SE8702422D0 (sv) Improvements in or relating to fungicides
SE8004498L (sv) Pyridylaminotriazolderivat
BG90609A (bg) Производни на пирола, методи за получаване и приложение

Legal Events

Date Code Title Description
FG2A Definitive protection

Ref document number: 332387

Country of ref document: ES