ES2059366T3 - Compuestos macrolidos. - Google Patents

Compuestos macrolidos.

Info

Publication number
ES2059366T3
ES2059366T3 ES87302108T ES87302108T ES2059366T3 ES 2059366 T3 ES2059366 T3 ES 2059366T3 ES 87302108 T ES87302108 T ES 87302108T ES 87302108 T ES87302108 T ES 87302108T ES 2059366 T3 ES2059366 T3 ES 2059366T3
Authority
ES
Spain
Prior art keywords
group
compounds
substituted
ester phosphoric
macrolid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES87302108T
Other languages
English (en)
Inventor
Michael V J Ramsay
Edward P Tiley
Oswy Z Pereira
John B Ward
Neil Porter
Hazel M Noble
Richard A Fletton
David Noble
Derek R Sutherland
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth Holdings LLC
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB868606122A external-priority patent/GB8606122D0/en
Priority claimed from GB868614689A external-priority patent/GB8614689D0/en
Priority claimed from GB868616346A external-priority patent/GB8616346D0/en
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Application granted granted Critical
Publication of ES2059366T3 publication Critical patent/ES2059366T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
    • A01N57/10—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds
    • A01N57/16—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds containing heterocyclic radicals

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)

Abstract

SE DESCRIBEN COMPUESTOS DE FORMULA (I) EMI PA=00 FR=1 HE=90 WI=130 TI=CHE Y SALES DE LOS MISMOS, DONDE R1 ES UN GRUPO METILO, ETILO O ISOPROPILO; R2 ES -H, -OH, -OH SUSTITUIDO O UN GRUPO ESTER FOSFORICO) Y R3 ES -H, O R2 Y R3 JUNTOS CON EL ATOMO DE CARBONO AL QUE ESTAN UNIDOS REPRESENTAN UN GRUPO >C=O Y OR4 ES UN GRUPO OR5 COMO SE HA DEFINIDO ANTES; CON LA CONDICION DE QUE R2 REPRESENTE UN GRUPO OR5 (DONDE OR5 ES UN GRUPO ALCOXI OR7 EN EL QUE R7 REPRESENTA UN ALQUILO C1-6 SUSTITUIDO CON UN ATOMO DE HALOGENO O UN ALQUILO C2-6 INTERRUMPIDO POR UN -O- O -S-) O BIEN QUE AL MENOS UNO DE R2 Y OR4 SEA UN GRUPO ESTER FOSFORICO O UN GRUPO OCONR10R11 (DONDE R10 Y R11 SON -H O UN ALQUILO C1-4). ESTOS COMPUESTOS PUEDEN USARSE PARA COMBATIR INSECTOS, ACAROS, NEMATODOS Y OTRAS PLAGAS.
ES87302108T 1986-03-12 1987-03-11 Compuestos macrolidos. Expired - Lifetime ES2059366T3 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB868606122A GB8606122D0 (en) 1986-03-12 1986-03-12 Chemical compounds
GB868614689A GB8614689D0 (en) 1986-06-17 1986-06-17 Chemical compounds
GB868616346A GB8616346D0 (en) 1986-07-04 1986-07-04 Chemical compounds

Publications (1)

Publication Number Publication Date
ES2059366T3 true ES2059366T3 (es) 1994-11-16

Family

ID=27262948

Family Applications (1)

Application Number Title Priority Date Filing Date
ES87302108T Expired - Lifetime ES2059366T3 (es) 1986-03-12 1987-03-11 Compuestos macrolidos.

Country Status (10)

Country Link
US (1) US4918098A (es)
EP (1) EP0238259B1 (es)
AU (1) AU609031B2 (es)
BR (1) BR8701121A (es)
CA (1) CA1288425C (es)
DE (1) DE3787548T2 (es)
ES (1) ES2059366T3 (es)
IE (1) IE62126B1 (es)
NZ (1) NZ219575A (es)
PH (1) PH24180A (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1301745C (en) * 1986-01-23 1992-05-26 Michael Vincent John Ramsay Macrolide antibiotics and their preparation
ES2055695T3 (es) * 1986-09-12 1994-09-01 American Cyanamid Co Derivados 23-desoxi de compuestos ll-f28249.
EP0259779B1 (en) * 1986-09-12 1994-08-10 American Cyanamid Company 23-Oxo (Keto) and 23-imino Derivatives of LL-F28249 Compounds
US4886829A (en) * 1987-03-06 1989-12-12 American Cyanamid Company 23-Oxo (keto) and 23-imino derivatives of mono- and diepoxy LL-F28249 compounds
GB8811036D0 (en) * 1988-05-10 1988-06-15 Glaxo Group Ltd Chemical compounds
GB8813150D0 (en) * 1988-06-03 1988-07-06 American Cyanamid Co Chemical compounds
US6826352B1 (en) 2000-03-29 2004-11-30 Macrovision Corporation Dynamic video copy protection system
EP2223600A1 (en) * 2009-02-19 2010-09-01 Urea Casale S.A. Granules containing filamentary fungi and method of preparation thereof
WO2012028556A1 (en) 2010-08-31 2012-03-08 Bayer Animal Health Gmbh Macrocyclic lactones and their use and their combinations with other active substances
DE102010064245A1 (de) 2010-12-28 2012-06-28 Bayer Animal Health Gmbh Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen
MX345501B (es) 2010-12-16 2017-02-02 Novo Nordisk As Composiciones solidas que comprenden agonista de glp-1 y sal del acido n-(8-(2-hidroxibenzoil)amino)caprilico.
MX355361B (es) 2011-04-12 2018-04-17 Novo Nordisk As Derivados de peptido 1 tipo glucagon (glp-1) doblemente acilados.
HUE042757T2 (hu) 2012-03-22 2019-07-29 Novo Nordisk As Szállító szert tartalmazó készítmények és elõállításuk
EP4331667A3 (en) 2012-03-22 2024-05-08 Novo Nordisk A/S Compositions comprising a delivery agent and preparation thereof
MY171146A (en) 2012-03-22 2019-09-27 Novo Nordisk As Compositions of glp-1 peptides and preparation thereof
EP2863895B1 (en) 2012-06-20 2021-04-14 Novo Nordisk A/S Tablet formulation comprising a peptide and a delivery agent
FR3023716A1 (fr) * 2014-07-18 2016-01-22 Univ Aix Marseille Compose et association de composes pour le traitement des poux
JP6621755B2 (ja) 2014-10-29 2019-12-18 学校法人東京理科大学 ユーシェアリライド類の製造方法
KR102647171B1 (ko) 2018-02-02 2024-03-15 노보 노르디스크 에이/에스 Glp-1 작용제 및 n-(8-(2-하이드록시벤조일)아미노)카프릴산의 염을 포함하는 고형 조성물

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4201861A (en) * 1977-10-03 1980-05-06 Merck & Co., Inc. Acyl derivatives of C-076 compounds
US4423209A (en) * 1982-02-26 1983-12-27 Merck & Co., Inc. Processes for the interconversion of avermectin compounds
JPS5920284A (ja) * 1982-07-23 1984-02-01 Sankyo Co Ltd ミルベマイシンｄの５−エ−テル誘導体及びその塩
US4469682A (en) * 1983-01-28 1984-09-04 Merck & Co., Inc. Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use
JPS60126289A (ja) * 1983-11-14 1985-07-05 Sankyo Co Ltd ミルベマイシン類の５−カ−ボネ−ト誘導体
PT80577B (pt) * 1984-06-05 1987-09-18 American Cyanamid Co Processo para a producao de novos agentes macrolidos ll-f28249 uteis no tratamento de infeccoes helminticas por ectoparasitas artropodes e por acarideos
AT396250B (de) * 1984-09-14 1993-07-26 American Cyanamid Co Verfahren zur herstellung von neuen antibiotisch wirkenden verbindungen
HUT39739A (en) * 1984-12-04 1986-10-29 Ciba Geigy Ag Process for production of derivatives of 13,3-milbemycin and medical preparatives containing thereof
US4587247A (en) * 1985-02-25 1986-05-06 Merck & Co., Inc. Substituted and unsubstituted 13-(alkoxy)methoxy derivatives of the avermectin aglycones, compositions and use
AU596586B2 (en) * 1985-04-30 1990-05-10 American Cyanamid Company Chemical derivatives of antibiotics S541
US4857544A (en) * 1987-03-06 1989-08-15 American Cyanamid Company 27-Halo derivatives of LL-F28249 compounds
US4956479A (en) * 1987-03-06 1990-09-11 American Cyanamid Company 23-deoxy-27-chloro derivatives of LL-F28249 compounds
US4806527A (en) * 1987-03-16 1989-02-21 Merck & Co., Inc. Avermectin derivatives

Also Published As

Publication number Publication date
PH24180A (en) 1990-03-22
BR8701121A (pt) 1988-01-05
AU6990887A (en) 1987-09-17
NZ219575A (en) 1990-04-26
DE3787548T2 (de) 1994-03-31
EP0238259A1 (en) 1987-09-23
EP0238259B1 (en) 1993-09-29
IE870627L (en) 1987-09-12
AU609031B2 (en) 1991-04-26
US4918098A (en) 1990-04-17
CA1288425C (en) 1991-09-03
DE3787548D1 (de) 1993-11-04
IE62126B1 (en) 1994-12-14

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