ES2057953T3 - Quinolilmetoxi-fenilacetamidas heterociclicamente substituidas como inhibidoras de la lipoxigenasa. - Google Patents

Quinolilmetoxi-fenilacetamidas heterociclicamente substituidas como inhibidoras de la lipoxigenasa.

Info

Publication number
ES2057953T3
ES2057953T3 ES92114428T ES92114428T ES2057953T3 ES 2057953 T3 ES2057953 T3 ES 2057953T3 ES 92114428 T ES92114428 T ES 92114428T ES 92114428 T ES92114428 T ES 92114428T ES 2057953 T3 ES2057953 T3 ES 2057953T3
Authority
ES
Spain
Prior art keywords
quinolylmetoxy
phenylacetamides
hetero
cyclically substituted
lipoxigenase
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES92114428T
Other languages
English (en)
Spanish (es)
Inventor
Siegfried Dr Raddatz
Klaus-Helmut Mohrs
Michael Dr Matzke
Romanis Fruchtmann
Armin Dr Hatzelmann
Christian Dr Kohlsdorfer
Reiner Prof Muller-Peddinghaus
Dr Theisen-Popp
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Application granted granted Critical
Publication of ES2057953T3 publication Critical patent/ES2057953T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Quinoline Compounds (AREA)
ES92114428T 1991-09-06 1992-08-25 Quinolilmetoxi-fenilacetamidas heterociclicamente substituidas como inhibidoras de la lipoxigenasa. Expired - Lifetime ES2057953T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4129742A DE4129742A1 (de) 1991-09-06 1991-09-06 Heterocyclisch substituierte chinolylmethoxy-phenylacetamide

Publications (1)

Publication Number Publication Date
ES2057953T3 true ES2057953T3 (es) 1994-10-16

Family

ID=6440067

Family Applications (1)

Application Number Title Priority Date Filing Date
ES92114428T Expired - Lifetime ES2057953T3 (es) 1991-09-06 1992-08-25 Quinolilmetoxi-fenilacetamidas heterociclicamente substituidas como inhibidoras de la lipoxigenasa.

Country Status (19)

Country Link
US (1) US5266578A (https=)
EP (1) EP0530639B1 (https=)
JP (1) JPH05194403A (https=)
KR (1) KR930006004A (https=)
CN (1) CN1070190A (https=)
AT (1) ATE110070T1 (https=)
AU (1) AU649351B2 (https=)
CA (1) CA2077465A1 (https=)
CZ (1) CZ276092A3 (https=)
DE (2) DE4129742A1 (https=)
DK (1) DK0530639T3 (https=)
ES (1) ES2057953T3 (https=)
FI (1) FI923968L (https=)
HU (1) HUT65660A (https=)
IL (1) IL103040A0 (https=)
MX (1) MX9204913A (https=)
NO (1) NO923181L (https=)
NZ (1) NZ244225A (https=)
TW (1) TW221431B (https=)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4219765A1 (de) * 1992-06-17 1993-12-23 Bayer Ag Substituierte (Benzothiazolyl- und Chinoxalyl-methoxy)phenylessigsäurederivate
ES2062943B1 (es) * 1993-03-23 1995-11-16 Uriach & Cia Sa J Nuevos derivados de la (2-metil-3-piridil) cianometilpiperazinas.
ATE188377T1 (de) * 1993-06-29 2000-01-15 Takeda Chemical Industries Ltd Chinoline oder chinazolin-derivate und deren verwendung zur herstellung eines medikaments für die behandlung von osteoporose
ES2103180B1 (es) * 1994-08-01 1998-04-01 Menarini Lab Fenilacetamidas con accion antagonista de los leucotrienos.
DE4443892A1 (de) * 1994-12-09 1996-06-13 Bayer Ag 4-(Chinolin-2-yl-methoxy)-phenyl-essigsäurederivate
EP0725063A1 (de) * 1995-02-01 1996-08-07 Ciba-Geigy Ag Chinolin-Derivate
US6121300A (en) 1998-11-10 2000-09-19 Wagle; Dilip R. Reversing advanced glycosylation cross-links using heterocyclic-substituted thiazolium salts
US6399641B1 (en) * 2000-07-13 2002-06-04 Hoffmann-La Roche Inc. 2H-tetrazole-amide compounds with therapeutic activity as metabotropic glutamate receptor agonists
ZA200602755B (en) * 2003-09-06 2007-06-27 Vertex Pharma Modulators of ATP-binding cassette transporters
KR102393675B1 (ko) * 2021-08-20 2022-05-11 (주)삼우공간건축사사무소 공동주택용 세대현관의 안전바닥패널

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS63503139A (ja) * 1986-03-13 1988-11-17 ローラー インターナショナル(オーバーシーズ)インコーポレーテッド 高血圧疾患治療剤としてのキノリニルエ−テル又はチオエ−テルテトラゾ−ル類
DE3900261A1 (de) * 1988-05-31 1989-12-07 Bayer Ag Substituierte 4-(chinolin-2-yl-methoxy) phenyl-essigsaeure-derivate
US5102881A (en) * 1988-06-27 1992-04-07 Merck Frosst Canada, Inc. Quinoline ether alkanoic acids
DE3916663A1 (de) * 1989-05-23 1990-11-29 Bayer Ag Substituierte (chinolin-2-yl-methoxy)phenyl-acyl-sulfonamide und -cyanamide, verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln
US5041453A (en) * 1990-05-30 1991-08-20 Rhone-Poulenc Rorer Pharmaceuticals Inc. Quinolinyl-benzoheterobicyclic derivatives as antagonists of leukotriene D4

Also Published As

Publication number Publication date
DE4129742A1 (de) 1993-03-11
DK0530639T3 (da) 1994-12-05
AU2205492A (en) 1993-03-11
US5266578A (en) 1993-11-30
EP0530639A1 (de) 1993-03-10
FI923968A7 (fi) 1993-03-07
IL103040A0 (en) 1993-02-21
NZ244225A (en) 1994-08-26
HUT65660A (en) 1994-07-28
FI923968A0 (fi) 1992-09-04
JPH05194403A (ja) 1993-08-03
FI923968L (fi) 1993-03-07
CN1070190A (zh) 1993-03-24
DE59200387D1 (de) 1994-09-22
CZ276092A3 (en) 1993-06-16
NO923181L (no) 1993-03-08
ATE110070T1 (de) 1994-09-15
MX9204913A (es) 1993-03-01
CA2077465A1 (en) 1993-03-07
TW221431B (https=) 1994-03-01
HU9202850D0 (en) 1992-11-30
KR930006004A (ko) 1993-04-20
NO923181D0 (no) 1992-08-14
AU649351B2 (en) 1994-05-19
EP0530639B1 (de) 1994-08-17

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