ES2001405A6 - Un procedimiento para la preparacion de derivados de 4-aminofenilo sustituidos - Google Patents

Un procedimiento para la preparacion de derivados de 4-aminofenilo sustituidos

Info

Publication number
ES2001405A6
ES2001405A6 ES8601414A ES8601414A ES2001405A6 ES 2001405 A6 ES2001405 A6 ES 2001405A6 ES 8601414 A ES8601414 A ES 8601414A ES 8601414 A ES8601414 A ES 8601414A ES 2001405 A6 ES2001405 A6 ES 2001405A6
Authority
ES
Spain
Prior art keywords
cycloalkyl
substituted
processfor
preparation
aminophenyl derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES8601414A
Other languages
English (en)
Inventor
Paolo Lombardi
Angelo Crugnola
Salle Enrico Di
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Publication of ES2001405A6 publication Critical patent/ES2001405A6/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/08—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions not involving the formation of amino groups, hydroxy groups or etherified or esterified hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
    • C07C205/56—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups bound to carbon atoms of six-membered aromatic rings and carboxyl groups bound to acyclic carbon atoms of the carbon skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/39—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by esterified hydroxy groups
    • C07C205/42—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by esterified hydroxy groups having nitro groups or esterified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/45—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by at least one doubly—bound oxygen atom, not being part of a —CHO group

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

UN PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE 4-AMINOFELICO SUSTITUIDOS. LOS COMPUESTOS (I) DONDE RFALQUILO, NF1 A 5, A Y BF-CO-, -O-, -NH- O -CH2- (SUJETOS A CIERTAS LIMITACIONES), SE OBTIENEN POR: 1) REACCION DE (II) CON (III); O 2) REDUCCION DE (IV); O 3) REDUCCION DE (I), DONDE O BIEN: I) A ES -CO- Y B ES -O- O -NH-, O II) A ES -O- O -NH- Y B ES -CO-, PARA DAR: (I) DONDE O BIEN: I) A ES -CH2- Y B ES -O- O -NH- O, RESPECTIVAMENTE, II) A ES -O- O -NH- Y B ES -CH2-; O 4) DESOXIGENAR (I) EN QUE A ES -CO- Y B ES -CH2- O A ES -CH2- Y B ES -CO- PARA DAR (I) DONDE A Y B SON AMBOS -CH2-. SON COMPUESTOS UTILES PARA TRATAR TUMORES E HIPERTROFIA O HIPERPLASIA PROSTATICA.
ES8601414A 1985-09-06 1986-08-27 Un procedimiento para la preparacion de derivados de 4-aminofenilo sustituidos Expired ES2001405A6 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858522186A GB8522186D0 (en) 1985-09-06 1985-09-06 Cycloalkyl-substituted 4-aminophenyl derivatives

Publications (1)

Publication Number Publication Date
ES2001405A6 true ES2001405A6 (es) 1988-05-16

Family

ID=10584835

Family Applications (1)

Application Number Title Priority Date Filing Date
ES8601414A Expired ES2001405A6 (es) 1985-09-06 1986-08-27 Un procedimiento para la preparacion de derivados de 4-aminofenilo sustituidos

Country Status (19)

Country Link
US (1) US4769483A (es)
EP (1) EP0215601B1 (es)
JP (1) JPS6259245A (es)
KR (1) KR870003054A (es)
CN (1) CN86105919A (es)
AT (1) ATE50982T1 (es)
AU (1) AU6213986A (es)
CA (1) CA1285287C (es)
DE (1) DE3669502D1 (es)
DK (1) DK420586A (es)
ES (1) ES2001405A6 (es)
FI (1) FI863566A (es)
GB (1) GB8522186D0 (es)
GR (1) GR862260B (es)
HU (1) HU198441B (es)
IL (1) IL79897A0 (es)
NZ (1) NZ217440A (es)
PT (1) PT83320B (es)
ZA (1) ZA866766B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8701080D0 (en) * 1987-01-19 1987-02-18 Erba Farmitalia Cycloalkyl-substituted 4-aminophenyl halo derivatives
GB2222588B (en) * 1988-09-09 1991-03-06 Erba Carlo Spa Cycloalkyl-substituted 4-aminophenyl derivatives and process for their preparation
GB2222589B (en) * 1988-09-09 1991-03-06 Erba Carlo Spa Cycloalkyl-substituted 4-aminophenyl derivatives and process for their preparation
US6031003A (en) * 1991-08-23 2000-02-29 Nps Pharmaceuticals, Inc. Calcium receptor-active molecules
US6011068A (en) * 1991-08-23 2000-01-04 Nps Pharmaceuticals, Inc. Calcium receptor-active molecules
US6313146B1 (en) 1991-08-23 2001-11-06 Nps Pharmaceuticals, Inc. Calcium receptor-active molecules
US6001884A (en) * 1991-08-23 1999-12-14 Nps Pharmaceuticals, Inc. Calcium receptor-active molecules
US5362911A (en) * 1993-12-30 1994-11-08 American Cyanamid Company Process for the preparation of o-aminophenyl cyclo-propyl ketone
UA55374C2 (uk) 1994-10-21 2003-04-15 Нпс Фармасьютікалз, Інк Сполуки, що мають активність по відношенню до рецепторів кальцію
ES2280460T3 (es) 1996-05-01 2007-09-16 Nps Pharmaceuticals, Inc. Compuestos activos frente a receptores de iones inorganicos.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2443342A1 (de) * 1974-09-11 1976-03-25 Basf Ag 1-amino-2-phenyl-propanverbindungen und verfahren zu ihrer herstellung
JPS58194814A (ja) * 1982-05-11 1983-11-12 Nippon Shinyaku Co Ltd 免疫調節作用を有する薬剤
GB8519261D0 (en) * 1985-07-31 1985-09-04 Roussel Lab Ltd Chemical compounds

Also Published As

Publication number Publication date
PT83320A (pt) 1986-10-01
HU198441B (en) 1989-10-30
GB8522186D0 (en) 1985-10-09
EP0215601A2 (en) 1987-03-25
JPS6259245A (ja) 1987-03-14
CA1285287C (en) 1991-06-25
EP0215601A3 (en) 1987-09-23
ATE50982T1 (de) 1990-03-15
KR870003054A (ko) 1987-04-14
DE3669502D1 (de) 1990-04-19
HUT44755A (en) 1988-04-28
US4769483A (en) 1988-09-06
PT83320B (en) 1988-10-07
DK420586A (da) 1987-03-07
EP0215601B1 (en) 1990-03-14
IL79897A0 (en) 1986-12-31
FI863566A (fi) 1987-03-07
GR862260B (en) 1987-01-02
ZA866766B (en) 1987-04-29
NZ217440A (en) 1989-10-27
CN86105919A (zh) 1987-03-04
AU6213986A (en) 1987-03-12
DK420586D0 (da) 1986-09-03
FI863566A0 (fi) 1986-09-04

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Legal Events

Date Code Title Description
SA6 Expiration date (snapshot 920101)

Free format text: 2006-08-27