EP3936190A4 - PENTACYCLIC HETEROCYCLIC COMPOUND - Google Patents
PENTACYCLIC HETEROCYCLIC COMPOUND Download PDFInfo
- Publication number
- EP3936190A4 EP3936190A4 EP20766918.5A EP20766918A EP3936190A4 EP 3936190 A4 EP3936190 A4 EP 3936190A4 EP 20766918 A EP20766918 A EP 20766918A EP 3936190 A4 EP3936190 A4 EP 3936190A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- heterocyclic compound
- pentacyclic heterocyclic
- pentacyclic
- compound
- heterocyclic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
- C07D491/147—Ortho-condensed systems the condensed system containing one ring with oxygen as ring hetero atom and two rings with nitrogen as ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2019039351 | 2019-03-05 | ||
PCT/JP2020/008881 WO2020179780A1 (ja) | 2019-03-05 | 2020-03-03 | 五環式複素環化合物 |
Publications (2)
Publication Number | Publication Date |
---|---|
EP3936190A1 EP3936190A1 (en) | 2022-01-12 |
EP3936190A4 true EP3936190A4 (en) | 2022-11-16 |
Family
ID=72336168
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP20766918.5A Pending EP3936190A4 (en) | 2019-03-05 | 2020-03-03 | PENTACYCLIC HETEROCYCLIC COMPOUND |
Country Status (21)
Country | Link |
---|---|
US (1) | US11358972B2 (zh) |
EP (1) | EP3936190A4 (zh) |
JP (1) | JP7504864B2 (zh) |
KR (1) | KR20210135224A (zh) |
CN (1) | CN113453762B (zh) |
AR (1) | AR118235A1 (zh) |
AU (1) | AU2020232044A1 (zh) |
BR (1) | BR112021015975A2 (zh) |
CA (1) | CA3129861A1 (zh) |
CL (1) | CL2021002144A1 (zh) |
CO (1) | CO2021010512A2 (zh) |
EA (1) | EA202191966A1 (zh) |
IL (1) | IL285511B1 (zh) |
JO (1) | JOP20210219A1 (zh) |
MA (1) | MA55221A (zh) |
MX (1) | MX2021009685A (zh) |
PE (1) | PE20211978A1 (zh) |
SG (1) | SG11202108780PA (zh) |
TW (1) | TWI821537B (zh) |
WO (1) | WO2020179780A1 (zh) |
ZA (1) | ZA202105729B (zh) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW202100531A (zh) | 2019-03-05 | 2021-01-01 | 日商衛材R&D企管股份有限公司 | 五環化合物之鹽及其等之結晶 |
Family Cites Families (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE258234C (zh) | ||||
US4187306A (en) | 1977-07-26 | 1980-02-05 | Bayer Aktiengesellschaft | Benzodiazepine-diones, a process for their production and their use as medicaments |
RU2117670C1 (ru) | 1988-10-31 | 1998-08-20 | Эйсай Ко., Лтд. | Производные триазоло[1,4]диазепина и способы их получения |
TW197442B (zh) | 1990-02-08 | 1993-01-01 | Pfizer | |
US5756494A (en) | 1992-07-24 | 1998-05-26 | Cephalon, Inc. | Protein kinase inhibitors for treatment of neurological disorders |
US5621100A (en) | 1992-07-24 | 1997-04-15 | Cephalon, Inc. | K-252a derivatives for treatment of neurological disorders |
US5736992A (en) * | 1994-10-31 | 1998-04-07 | Hewlett-Packard | Pressure regulated free-ink ink-jet pen |
KR100203456B1 (ko) | 1995-06-20 | 1999-06-15 | 한승수 | 디하이드로에보디아민-에이치씨1를 유효성분으로 함유하는 알츠하이머병에 의한 치매 치료제 |
CL2004000348A1 (es) | 1997-04-15 | 2005-01-14 | Cephalon Inc & Kyowa Hakko Kog | Compuesto derivado de estaurosporina bis-n-sustituida, util para potenciar la funcion de neuronas colinergicas, estriadas, del prosencefalo basal y sensoriales. |
CL2004000352A1 (es) | 1998-05-26 | 2005-05-27 | Cephalon Inc & Kyowa Hakko Kog | Uso de compuestos derivados de estaurosporina para potenciar la funcion de neuronas colinergicas, estriadas, de prosencefalo basal y sensoriales. |
FR2779652B1 (fr) | 1998-06-15 | 2001-06-08 | Sod Conseils Rech Applic | Utilisation de diazepines pour la preparation de medicaments destines a traiter les etats pathologiques ou les maladies dans lesquels un des recepteurs de la somatostatine est implique |
DE10246207B4 (de) * | 2002-10-04 | 2008-04-03 | Disetronic Licensing Ag | Mikrodialysesonde mit spiralförmiger Leitung |
AU2003299378A1 (en) | 2002-10-11 | 2004-05-04 | Board Of Regents, The University Of Texas System | Method and compounds for inhibiting hec1 activity for the treatment of proliferative diseases |
GB0308333D0 (en) * | 2003-04-10 | 2003-05-14 | Glaxo Group Ltd | Novel compounds |
CN101084220B (zh) | 2004-10-20 | 2010-12-15 | 弗·哈夫曼-拉罗切有限公司 | 卤素取代的苯并二氮杂*衍生物 |
JP2009184924A (ja) | 2006-05-31 | 2009-08-20 | Eisai R & D Management Co Ltd | 生物学的試薬用化合物 |
GB201100181D0 (en) * | 2011-01-06 | 2011-02-23 | Eisai Ltd | Fused aminodihydrothiazine derivatives |
EP3144308B1 (en) * | 2014-05-16 | 2020-06-24 | Takeda Pharmaceutical Company Limited | Nitrogen-containing heterocyclic compound |
PL3680243T3 (pl) | 2017-09-07 | 2022-02-14 | Eisai R&D Management Co., Ltd. | Związek pentacykliczny |
TW202100531A (zh) | 2019-03-05 | 2021-01-01 | 日商衛材R&D企管股份有限公司 | 五環化合物之鹽及其等之結晶 |
-
2020
- 2020-03-03 BR BR112021015975-4A patent/BR112021015975A2/pt unknown
- 2020-03-03 JO JOP/2021/0219A patent/JOP20210219A1/ar unknown
- 2020-03-03 TW TW109106904A patent/TWI821537B/zh active
- 2020-03-03 AR ARP200100583A patent/AR118235A1/es unknown
- 2020-03-03 EA EA202191966A patent/EA202191966A1/ru unknown
- 2020-03-03 AU AU2020232044A patent/AU2020232044A1/en active Pending
- 2020-03-03 JP JP2021504107A patent/JP7504864B2/ja active Active
- 2020-03-03 IL IL285511A patent/IL285511B1/en unknown
- 2020-03-03 CA CA3129861A patent/CA3129861A1/en active Pending
- 2020-03-03 MX MX2021009685A patent/MX2021009685A/es unknown
- 2020-03-03 US US16/807,335 patent/US11358972B2/en active Active
- 2020-03-03 WO PCT/JP2020/008881 patent/WO2020179780A1/ja active Application Filing
- 2020-03-03 EP EP20766918.5A patent/EP3936190A4/en active Pending
- 2020-03-03 KR KR1020217025605A patent/KR20210135224A/ko active Search and Examination
- 2020-03-03 SG SG11202108780PA patent/SG11202108780PA/en unknown
- 2020-03-03 MA MA055221A patent/MA55221A/fr unknown
- 2020-03-03 PE PE2021001331A patent/PE20211978A1/es unknown
- 2020-03-03 CN CN202080014008.7A patent/CN113453762B/zh active Active
-
2021
- 2021-08-12 CO CONC2021/0010512A patent/CO2021010512A2/es unknown
- 2021-08-12 ZA ZA2021/05729A patent/ZA202105729B/en unknown
- 2021-08-12 CL CL2021002144A patent/CL2021002144A1/es unknown
Non-Patent Citations (1)
Title |
---|
No further relevant documents disclosed * |
Also Published As
Publication number | Publication date |
---|---|
EP3936190A1 (en) | 2022-01-12 |
PE20211978A1 (es) | 2021-10-05 |
AU2020232044A1 (en) | 2021-09-02 |
ZA202105729B (en) | 2022-08-31 |
CL2021002144A1 (es) | 2022-02-04 |
CN113453762A (zh) | 2021-09-28 |
SG11202108780PA (en) | 2021-09-29 |
JPWO2020179780A1 (zh) | 2020-09-10 |
TWI821537B (zh) | 2023-11-11 |
AR118235A1 (es) | 2021-09-22 |
JOP20210219A1 (ar) | 2023-01-30 |
MA55221A (fr) | 2022-01-12 |
KR20210135224A (ko) | 2021-11-12 |
MX2021009685A (es) | 2021-09-10 |
US11358972B2 (en) | 2022-06-14 |
US20200283452A1 (en) | 2020-09-10 |
TW202100528A (zh) | 2021-01-01 |
EA202191966A1 (ru) | 2021-12-08 |
BR112021015975A2 (pt) | 2021-10-05 |
IL285511A (en) | 2021-09-30 |
CA3129861A1 (en) | 2020-09-10 |
CN113453762B (zh) | 2024-06-07 |
WO2020179780A1 (ja) | 2020-09-10 |
CO2021010512A2 (es) | 2021-10-29 |
IL285511B1 (en) | 2024-06-01 |
JP7504864B2 (ja) | 2024-06-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE INTERNATIONAL PUBLICATION HAS BEEN MADE |
|
PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: REQUEST FOR EXAMINATION WAS MADE |
|
17P | Request for examination filed |
Effective date: 20210811 |
|
AK | Designated contracting states |
Kind code of ref document: A1 Designated state(s): AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR |
|
A4 | Supplementary search report drawn up and despatched |
Effective date: 20221018 |
|
RIC1 | Information provided on ipc code assigned before grant |
Ipc: A61K 31/551 20060101ALI20221012BHEP Ipc: C07D 495/22 20060101ALI20221012BHEP Ipc: C07D 491/22 20060101ALI20221012BHEP Ipc: C07D 491/147 20060101ALI20221012BHEP Ipc: A61P 43/00 20060101ALI20221012BHEP Ipc: A61P 25/28 20060101AFI20221012BHEP |
|
P01 | Opt-out of the competence of the unified patent court (upc) registered |
Effective date: 20230511 |